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cholecystokinin

Cholecystokinin is a peptide hormone of the gastrointestinal system responsible for stimulating the digestion of fat and protein.

  • Ceruletide
    T1493217650-98-5
    Ceruletide (Caerulein) is a potent agonist of cholecystokinin receptor and it also is a safe and effective cholecystokinetic agent. It has a direct spasmogenic effect on the gallbladder muscle and bile ducts.
    • $162
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  • N-Cbz-DL-tryptophan
    T934313058-16-7
    N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
    • $35
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  • GV150013
    T27503167355-22-8In house
    GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
    • $329
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  • Gastrin I (human) acetate
    TP2030L1
    Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (CCK2) receptor.
    • $122
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  • PHA-767491
    T6206845714-00-3
    PHA-767491 (CAY10572) is a potent ATP-competitive dual Cdc7/CDK9 inhibitor with IC50 of 10 nM and 34 nM, respectively.
    • $30
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  • CCK Octapeptide, non-sulfated acetate
    TP2204L
    CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.
    • $131
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  • (Iso)-FK-480
    T10055167820-10-2In house
    (Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.
    • $1,520
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  • GI 181771
    T15382305366-98-7
    GI 181771 is an agonist of the cholecystokinin 1 receptor. GI 181771 can be used in studies about obesity.
    • $195
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  • [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
    TP1931L1
    [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate ([D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate (96736-12-8 free base)) is a broad spectrum neuropeptide inverse agonist and antagonist. Potent full inverse agonist for the ghrelin receptor (EC50 = 5.2 nM); diminishes constitutive ghrelin receptor signaling. Also antagonist at tachykinin, bradykinin, CCK and bombesin receptors. Induces apoptosis and inhibits cancer cell growth in vitro.
    • $143
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  • GV-150013X
    T27503L151386-96-8In house
    GV-150013X ((S)-1-(1-(adamantan-1-ylmethyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl)-3-phenylurea) is a potent CCKB antiagonist, pKi= 9.02.
    • $197
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  • Ceruletide Ammonium Salt
    T14932L1
    Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe and effective cholecystokinin receptor agonist with direct spasmodic effects on the gallbladder muscle and bile ducts. Ceruletide Ammonium Salt has sedative activity and has been used in the study of chronic schizophrenia.Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs.
    • $89
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  • XL413
    T33521169558-38-6In house
    XL-413 is an orally bioavailable cell division cycle 7 homolog (CDC7) kinase inhibitor with potential antineoplastic activity. XL-413 binds to and inhibits the activity of CDC7, which may result in the inhibition of DNA replication and mitosis, the induct
    • $48
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    TargetMol | Citations Cited
  • Mini Gastrin I, human acetate
    TP1821L
    Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.
    • $176
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  • Ceruletide Ammonium acetate
    T14932L
    Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stimulant.
    • $251
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  • A-65186
    T26483119295-94-2
    A-65186 is an A-type glutamatergic cholecystokinin (CCK) antagonist used to study inflammation and gastrointestinal tract injury.
    • $293
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  • Pranazepide
    T34123150408-73-4
    Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.
    • $543
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  • Loxiglumide
    T2312107097-80-3
    Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.
    • $34
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  • CCK-A receptor inhibitor 1
    T12404137004-80-9
    CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study of diseases related to the digestive system.
    • $700
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  • Gastrin/CCK antagonist 1
    T13260162271-52-5
    Gastrin/CCK antagonist 1 is a potent gastrin/CCK antagonist for the study of metabolic system-related diseases.
    • $700
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  • Spiroglumide
    T68016137795-35-8
    Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 (8.67-46.4) mg / kg, could be used to explore the physiological role of gastrin in the regulation of human gastric acid secretion.
    • $158
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  • XL413 hydrochloride
    T67352062200-97-7
    XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7, with an IC 50 of 3.4 nM. XL413 hydrochloride also exhibits potent effect with IC 50 s of 215, 42 nM on CK2, PIM1, respectively, and an EC 50 of 118 nM on pMCM.
    • $48
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  • Sincalide ammonium
    TP119870706-98-8
    Sincalide ammonium (CCK-8 ammonium) is a potent analog of the amino acid peptide hormone cholecystokinin (CCK), an active fragment that retains much of the biological activity of CCK.Sincalide ammonium promotes bile secretion, causes gallbladder contractions and relaxes the sphincter of Oddi, thereby facilitating bile drainage into the duodenum. Sincalide ammonium promotes bile secretion, contraction of the gallbladder and relaxation of the sphincter of Oddi, thereby facilitating the drainage of bile into the duodenum.Sincalide ammonium can be injected to promote gallbladder contraction, and is commonly used as an adjunct in the diagnosis of gallbladder and pancreatic diseases and in cholecystography.
    • $89
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  • Gastrin I, human
    TP203010047-33-3
    Gastrin I, human (Gastrin I (human)) is an endogenous peptide produced in the stomach that increases pepsinogen and acid secretion via the CCK2 receptor in the rat.
    • $109
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  • Itriglumide
    T27640201605-51-8
    Itriglumide (CR-2945) is a cholecystokinin (CCK)-2 receptor antagonist with antisecretory and antiulcerogenic properties.
    • $293
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  • Cholecystokinin (26-33) free acid
    TP2500103974-46-5
    Cholecystokinin (26-33) free acid, a part of cholecystokinin (CCK), is a highly selective ligand for CCKB-type receptors found in the vertebrate CNS and induces a mild taste aversion conditioned reflex in rats.
    • $40
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  • Nastorazepide
    TQ0062209219-38-5
    Nastorazepide (Z-360) is a selective, orally available antagonist of gastrin/cholecystokinin 2 (CCK-2) receptor with potential antineoplastic activity.
    • $48
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  • Lintitript
    T15759136381-85-6
    Lintitript (SR 27897) is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM for CCK1 and CCK2. The Ki value is 0.2 nM for CCK1.
    • $117
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  • Proglumide
    T10526620-60-6
    Proglumide (Binoside) is a cholecystokinin antagonist, which blocks both the CCKA and CCKB subtypes. Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. It is used clinically in the drug therapy of gastrointestinal ulcers.
    • $33
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  • WAY-620645
    T9991742116-45-6
    WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
    • $57
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  • Lorglumide sodium salt
    T118681021868-76-7
    Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).
    • $29
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  • Pentagastrin
    T45795534-95-2
    Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of salivary proteins.
    • $47
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