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mAChr-in-1

Name: mAChr-in-1
Brand: TargetMol
SKU: T5476
Rating: 4.5 (1 reviews)

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Catalog No. T5476Cas No. 119391-56-9

mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).

mAChr-in-1

😃Good

Catalog No. T5476Cas No. 119391-56-9

mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).

Pack Size	Price	Availability	Quantity
25 mg	$730	1-2 weeks
1 mL x 10 mM (in DMSO)	$223	1-2 weeks

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Product Introduction

Bioactivity

Description	mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Targets&IC50	mAChR:17 nM

Chemical Properties

Molecular Weight	488.36
Formula	C₂₃H₂₅IN₂O₂
Cas No.	119391-56-9
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 52 mg/mL (106.48 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0477 mL	10.2383 mL	20.4767 mL	102.3835 mL
5 mM	0.4095 mL	2.0477 mL	4.0953 mL	20.4767 mL
10 mM	0.2048 mL	1.0238 mL	2.0477 mL	10.2383 mL
20 mM	0.1024 mL	0.5119 mL	1.0238 mL	5.1192 mL
50 mM	0.0410 mL	0.2048 mL	0.4095 mL	2.0477 mL
100 mM	0.0205 mL	0.1024 mL	0.2048 mL	1.0238 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc