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N,N-Didesethyl Sunitinib

Name: N,N-Didesethyl Sunitinib
Brand: TargetMol
SKU: T60128
Price: 139 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T60128Cas No. 873077-70-4

Alias AMPK-IN-4

N,N-Didesethyl Sunitinib is a potent AMPK inhibitor with IC50 of 393 nM and 141 nM for AMPKα1 and AMPK2,respectively.

N,N-Didesethyl Sunitinib

🥰Excellent

Purity: 97.1%

Catalog No. T60128Alias AMPK-IN-4Cas No. 873077-70-4

N,N-Didesethyl Sunitinib is a potent AMPK inhibitor with IC50 of 393 nM and 141 nM for AMPKα1 and AMPK2,respectively.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$139	-	In Stock
5 mg	$347	-	In Stock
10 mg	$488	-	In Stock
25 mg	$793	-	In Stock
50 mg	$1,080	-	In Stock
100 mg	$1,480	-	In Stock
1 mL x 10 mM (in DMSO)	$355	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Batch Information

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Purity:97.1%

Resource Download

COA HPLC HNMR

Product Introduction

Bioactivity

Description	N,N-Didesethyl Sunitinib is a potent AMPK inhibitor with IC50 of 393 nM and 141 nM for AMPKα1 and AMPK2,respectively.
Synonyms	AMPK-IN-4

Chemical Properties

Molecular Weight	342.37
Formula	C₁₈H₁₉FN₄O₂
Cas No.	873077-70-4
Smiles	C(=C\1/C=2C(NC1=O)=CC=C(F)C2)\C3=C(C)C(C(NCCN)=O)=C(C)N3
Relative Density.	1.345 g/cm3 (Predicted)
Color	Orange
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 4.5 mg/mL (11.88 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.9208 mL	14.6041 mL	29.2082 mL	146.0408 mL
5 mM	0.5842 mL	2.9208 mL	5.8416 mL	29.2082 mL
10 mM	0.2921 mL	1.4604 mL	2.9208 mL	14.6041 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc