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CAY10471 Racemate

🥰Excellent
Catalog No. T7359Cas No. 844639-57-2
Alias TM30089 Racemate

CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective CRTH2/DP2 receptor antagonist. It binds to human CRTH2/DP2, DP1, and TP receptors with Ki values of 0.6, 1200, and >10,000 nM, respectively.

CAY10471 Racemate

CAY10471 Racemate

🥰Excellent
Purity: 99.08%
Catalog No. T7359Alias TM30089 RacemateCas No. 844639-57-2
CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective CRTH2/DP2 receptor antagonist. It binds to human CRTH2/DP2, DP1, and TP receptors with Ki values of 0.6, 1200, and >10,000 nM, respectively.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
5 mg$43In StockIn Stock
10 mg$68In StockIn Stock
25 mg$143In StockIn Stock
50 mg$213In StockIn Stock
100 mg$316In StockIn Stock
200 mg$457-In Stock
1 mL x 10 mM (in DMSO)$47In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.08%
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Product Introduction

Bioactivity
Description
CAY10471 Racemate (TM30089 Racemate) is a potent and highly selective CRTH2/DP2 receptor antagonist. It binds to human CRTH2/DP2, DP1, and TP receptors with Ki values of 0.6, 1200, and >10,000 nM, respectively.
Targets&IC50
DP:1200 nM(ki), CRTH2:0.6 nM(ki)
SynonymsTM30089 Racemate
Chemical Properties
Molecular Weight416.47
FormulaC21H21FN2O4S
Cas No.844639-57-2
Smiles[Na+].CN(C1CCc2c(C1)c1ccccc1n2CC([O-])=O)S(=O)(=O)c1ccc(F)cc1
Relative Density.1.41 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 150 mg/mL (360.17 mM), Sonication is recommended.
In Vivo Formulation
10% DMSO+40% PEG300+5% Tween 80+45% Saline: 4 mg/mL (9.6 mM), Sonication is recommended.
Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.4011 mL12.0057 mL24.0113 mL120.0567 mL
5 mM0.4802 mL2.4011 mL4.8023 mL24.0113 mL
10 mM0.2401 mL1.2006 mL2.4011 mL12.0057 mL
20 mM0.1201 mL0.6003 mL1.2006 mL6.0028 mL
50 mM0.0480 mL0.2401 mL0.4802 mL2.4011 mL
100 mM0.0240 mL0.1201 mL0.2401 mL1.2006 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

TM-30089TM30089TM 30089ProstaglandinReceptorProstaglandin ReceptorInhibitorinhibitCRTh2 (DP2) receptorCAY-10471 RacemateCAY10471 RacemateCAY-10471CAY10471CAY 10471
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