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Lartesertib

Name: Lartesertib
Brand: TargetMol
SKU: T62684
Price: 132 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T62684Cas No. 2495096-26-7

Alias M4076, ATM Inhibitor-5

Lartesertib (ATM Inhibitor-5) is an inhibitor of serine/threonine protein kinase ATM with potential anticancer activity for the study of lung cancer.

Lartesertib

🥰Excellent

Purity: 99.9%

Catalog No. T62684Alias M4076, ATM Inhibitor-5Cas No. 2495096-26-7

Lartesertib (ATM Inhibitor-5) is an inhibitor of serine/threonine protein kinase ATM with potential anticancer activity for the study of lung cancer.

Pack Size	Price	Availability
1 mg	$132	In Stock
2 mg	$196	In Stock
5 mg	$328	In Stock
10 mg	$562	In Stock
25 mg	$1,090	In Stock
50 mg	$1,820	In Stock
100 mg	$2,820	In Stock
1 mL x 10 mM (in DMSO)	$363	In Stock

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Batch Information

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Purity:99.9%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Lartesertib (ATM Inhibitor-5) is an inhibitor of serine/threonine protein kinase ATM with potential anticancer activity for the study of lung cancer.
Synonyms	M4076, ATM Inhibitor-5

Chemical Properties

Molecular Weight	448.45
Formula	C₂₃H₂₁FN₆O₃
Cas No.	2495096-26-7
Smiles	COc1cncc(F)c1-n1c2c(cnc3cc(OC)c(cc23)-c2cn(C)nc2C)n(C)c1=O
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

store at low temperature,keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 80 mg/mL (178.39 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.2299 mL	11.1495 mL	22.2990 mL	111.4951 mL
5 mM	0.4460 mL	2.2299 mL	4.4598 mL	22.2990 mL
10 mM	0.2230 mL	1.1150 mL	2.2299 mL	11.1495 mL
20 mM	0.1115 mL	0.5575 mL	1.1150 mL	5.5748 mL
50 mM	0.0446 mL	0.2230 mL	0.4460 mL	2.2299 mL
100 mM	0.0223 mL	0.1115 mL	0.2230 mL	1.1150 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc