Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Membrane Protein-targeted Compound Library

Catalog No. L1520

Membrane proteins are a class of proteins widely found in biological cell membranes, playing essential roles in the structure and function of cells. Based on their location and function, membrane proteins can be classified into three main categories: peripheral membrane proteins, integral membrane proteins, and lipid-anchored proteins. Membrane proteins encompass a variety of functional proteins, including glycoproteins, carrier proteins, and enzymes. They are often linked to carbohydrate molecules, which can transmit signals into the cell by undergoing structural changes, participating in signal transduction processes. Membrane proteins perform a range of critical functions, including substance transport, signal transduction, cell recognition, and energy conversion. In drug development, membrane proteins, especially G protein-coupled receptors (GPCRs), ion channels, and transporters, are of particular interest. Many diseases are related to the malfunction of specific membrane proteins. Therefore, drugs designed to target these proteins can regulate their activity, aiming to treat diseases. TargetMol has collected 4175 compounds that target membrane proteins, which can be used for membrane protein-related scientific research and drug screening, suitable for high-throughput and high-content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L1520

Membrane Protein-targeted Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 4175 small molecules targeting various membrane proteins.
  • Structurally diverse, highly effective, and cell-permeable.
  • Detailed compound information with structure, target, activity, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are in stock and continuously updated.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

5-HT Receptor
AChR
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
Potassium Channel
Autophagy
Apoptosis
EGFR
Histamine Receptor
VEGFR
Sodium Channel
GABA Receptor
GluR
TRP/TRPV Channel
Endogenous Metabolite
GPR
Prostaglandin Receptor
Adenosine Receptor
Opioid Receptor
PDGFR
iGluR
RAAS
FGFR
c-Kit
c-Met/HGFR
TLR
ATPase
Antibacterial
Cannabinoid Receptor
ALK
FLT
Ras
NMDAR
CCR
P-gp
Parasite
Kras
P2X Receptor
NF-κB
CXCR
S1P Receptor
Src
HER
Neurokinin receptor
P450
LPL Receptor
Hedgehog/Smoothened
COX
TAM Receptor
Chloride channel
Proton pump
IGF-1R
Sigma receptor
HIV Protease
PDE
Norepinephrine
CFTR
Serotonin Transporter
Raf
Reactive Oxygen Species
Protease-activated Receptor
TGF-beta/Smad
AChE
c-Fms
Antibiotic
Glucagon Receptor
Endothelin Receptor
Bcr-Abl
SGLT
Trk receptor
P2Y Receptor
Neuropeptide Y Receptor
cAMP
c-RET
CDK
JAK
Bradykinin Receptor
LPA Receptor
TNF
Guanylate cyclase
Influenza Virus
Ferroptosis
Antifungal
PPAR
MRP
Vasopressin Receptor
GTPase
Leukotriene Receptor
ERK
IL Receptor
OX Receptor
SARS-CoV
NO Synthase
GNRH Receptor
PKC
Drug Metabolite
Aurora Kinase
Rho
ROS
Akt
DNA/RNA Synthesis
Melanocortin Receptor
Mitophagy
ABC
Ephrin Receptor
cholecystokinin
Monocarboxylate transporter
p38 MAPK
PI3K
CaSR
PKA
Neurotensin Receptor
CSF-1R
Monoamine Transporter
Smo
Somatostatin
GPCR19
Phospholipase
GHSR
HCV Protease
GRK
Lipoxygenase
CaMK
STAT
AMPK
Discoidin Domain Receptor (DDR)
ROS Kinase
Virus Protease
Melatonin Receptor
Tyrosine Kinases
Antioxidant
Mitochondrial Metabolism
BTK
BCRP
Arrestin
Glucocorticoid Receptor
HDAC
Tyrosinase
FAK
NOS
Carbonic Anhydrase
Dehydrogenase
LTR
Na+/Ca2+ Exchanger
JNK
OCT
Caspase
Annexin A
MT Receptor
Bombesin Receptor
HSV
OAT
IκB/IKK
Oxytocin Receptor
Phosphatase
ROCK
Topoisomerase
PAFR
Interleukin
MAPK
TSH Receptor
CRFR
Beta Amyloid
MEK
Syk
Monoamine Oxidase
Melanin-concentrating Hormone Receptor (MCHR)
Transferase
CRM1
GSK-3
VDAC
FXR
MMP
mTOR
Aquaporin
CGRP Receptor
Anti-infection
Microtubule Associated
Thrombin
Apelin receptor
NPC1L1
Histone Methyltransferase
Estrogen/progestogen Receptor
HBV
Wnt/beta-catenin
MAO
Adiponectin receptor
LDL
HCN Channel
FAAH
DNA
Beta-Secretase
HSP
transporter
HIF
Platelet aggregation
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
MLK
NADPH
Glutathione Peroxidase
Tie-2
Estrogen Receptor/ERR
Serine/threonin kinase
Immunology/Inflammation related
Na-K-Cl cotransporter
PROTAC Linker
BCL
Fatty Acid Synthase
Chk
ACK
Antiviral
Casein Kinase
RSV
GST
Reverse Transcriptase
Hydroxylase
HMG-CoA Reductase
AhR
Imidazoline Receptor
Proteasome
Adenylyl cyclase
Transaminase
ROR
EBI2/GPR183
Integrin
MyD88
Reductase
BACE
DYRK
Kisspeptin
PARP
Serine Protease
Cysteine Protease
PYK2
IRE1
Myosin
RIP kinase
Gamma-secretase
Antifection
PAK
Epigenetic Reader Domain
Androgen Receptor
Acyltransferase
LRRK2
Free radical scavengers
Histone Acetyltransferase
GluCls
PAI-1
CRISPR/Cas9
PDK
PLK
NADPH-oxidase
DNA Methyltransferase
NOD
IRAK
NOD-like Receptor (NLR)
PROTACs
CAT
GSNOR
Piezo Channel
Dynamin
Amino Acids and Derivatives
YAP
Neuropeptide W
RAR/RXR 
PERK
TOPK
Progesterone Receptor
c-Myc
N-Acetylglucosaminyltransferase
Antifolate
Hck
Amylase
IAP
FLAP
E1/E2/E3 Enzyme
UGT
DNA gyrase
GlyT
Glucosidase
Anion Exchanger
DNA Alkylation
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
PTEN
PAD
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
PGE Synthase
MNK
Aminopeptidase
Sirtuin
Nrf2
Hippo pathway
Neprilysin
GPX
Retinoid Receptor
ribosome
RXFP receptor
Adenosine deaminase
SGK
Gap Junction Protein
lysosomal autophagy
p53
PKM

Keywords