Shopping Cart
Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Membrane Protein-targeted Compound Library

Catalog No. L1520

Membrane proteins are a class of proteins widely found in biological cell membranes, playing essential roles in the structure and function of cells. Based on their location and function, membrane proteins can be classified into three main categories: peripheral membrane proteins, integral membrane proteins, and lipid-anchored proteins. Membrane proteins encompass a variety of functional proteins, including glycoproteins, carrier proteins, and enzymes. They are often linked to carbohydrate molecules, which can transmit signals into the cell by undergoing structural changes, participating in signal transduction processes.

Membrane proteins perform a range of critical functions, including substance transport, signal transduction, cell recognition, and energy conversion. In drug development, membrane proteins, especially G protein-coupled receptors (GPCRs), ion channels, and transporters, are of particular interest. Many diseases are related to the malfunction of specific membrane proteins. Therefore, drugs designed to target these proteins can regulate their activity, aiming to treat diseases.

TargetMol has collected 6422 compounds that target membrane proteins, which can be used for membrane protein-related scientific research and drug screening, suitable for high-throughput and high-content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L1520

Membrane Protein-targeted Compound Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 6422 small molecules targeting various membrane proteins.
  • Structurally diverse, highly effective, and cell-permeable.
  • Detailed compound information with structure, target, activity, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;
  • All compounds are in stock and continuously updated.

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Apoptosis
5-HT Receptor
Autophagy
AChR
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
Potassium Channel
Endogenous Metabolite
EGFR
Histamine Receptor
Ras
Sodium Channel
GABA Receptor
VEGFR
Antibacterial
GluR
TRP/TRPV Channel
p38 MAPK
Histone Methyltransferase
NF-κB
GPCR
iGluR
Cholinesterase (ChE)
Caspase
JAK
Prostaglandin Receptor
Src
Parasite
NO Synthase
Adenosine Receptor
FLT
ERK
Akt
PKC
ROS
Opioid Receptor
PDGFR
Estrogen Receptor/ERR
GSK-3
MMP
TLR
RAAS
FGFR
Raf
c-Met/HGFR
TNF
c-Kit
CDK
TGF-beta/Smad
COX
Cannabinoid Receptor
Bcr-Abl
HSP
ALK
ATPase
Wnt/beta-catenin
Cytochromes P450
P-gp
PKA
BTK
LPL Receptor
Reactive Oxygen Species
Antibiotic
NMDAR
Estrogen/progestogen Receptor
Interleukin
KRas
HIV Protease
Aurora Kinase
Serotonin Transporter
CCR
ROCK
STAT
Tyrosine Kinases
PI3K
CXCR
Drug Metabolite
Integrin
Neurokinin receptor
IGF-1R
Casein Kinase
P2X Receptor
S1P Receptor
Proton pump
DNA/RNA Synthesis
Sigma receptor
Trk receptor
FAK
c-RET
Antifungal
Hedgehog/Smoothened
IL Receptor
Influenza Virus
TAM Receptor
PDE
JNK
SARS-CoV
Angiotensin-converting Enzyme (ACE)
PPAR
c-Fms
Ferroptosis
Norepinephrine
CFTR
Bcl-2 Family
Virus Protease
HER
transporter
Chloride channel
mTOR
Syk
Beta Amyloid
Cysteine Protease
Protease-activated Receptor
AMPK
Leukotriene Receptor
Endothelin Receptor
Cholecystokinin Receptor
cAMP
Epigenetic Reader Domain
PARP
Mitophagy
P2Y Receptor
Glucagon Receptor
SGLT
Anti-infection
DYRK
ROS Kinase
LPA Receptor
MEK
Melanocortin Receptor
MRP
Smo
Neuropeptide Y Receptor
NOS
OX Receptor
Antioxidant
S6 Kinase
Vasopressin Receptor
Lipoxygenase
Guanylate cyclase
Bradykinin Receptor
GNRH Receptor
CaMK
Rho
Tyrosinase
Phospholipase
ABC Transporter
HSV
GTPase
Ephrin Receptor
Mitochondrial Metabolism
GPCR19
HCV Protease
Adenylate cyclase
HDAC
Serine Protease
MAPK
Monoamine Oxidase
Arrestin
Phosphatase
Nrf2
Neurotensin Receptor
BCRP
CSF-1R
PERK
Monoamine Transporter
HIF/HIF Prolyl-Hydroxylase
Dehydrogenase
CaSR
GHSR
Monocarboxylate transporter
Discoidin Domain Receptor (DDR)
Microtubule Associated
PAFR
Serine/threonin kinase
Somatostatin
Immunology/Inflammation related
GRK
Antiviral
MAO
Melatonin Receptor
Antifection
PGE Synthase
IκB/IKK
Glucocorticoid Receptor
Bombesin Receptor
Na+/Ca2+ Exchanger
MDM-2/p53
Topoisomerase
Tie-2
OAT
CRFR
Oxytocin Receptor
FXR
PYK2
Carbonic Anhydrase
HBV
Sirtuin
Apelin receptor
OCT
NOD-like Receptor (NLR)
CGRP Receptor
MLK
RIP kinase
Glucosidase
Beta-Secretase
Nucleoside Antimetabolite/Analog
Pim
Annexin A
MT Receptor
CRM1
Glutaminase
Melanin-concentrating Hormone Receptor (MCHR)
Neuropeptide FF Receptor
Acyltransferase
LTR
TSH Receptor
Hydroxylase
Chk
Transferase
BACE
DNA Methyltransferase
Thrombin
Progesterone Receptor
HCN Channel
HIF
IRAK
Aryl Hydrocarbon Receptor
LDL
p53
Fatty Acid Synthase
Androgen Receptor
Aquaporin
Reductase
Myosin
Histone Demethylase
RSV
IFNAR
NADPH
AhR
c-Myc
NOD
MyD88
Glutathione Peroxidase
PTEN
HMG-CoA Reductase
Proteasome
NPC1L1
FOXO
PROTACs
FAAH
glycosidase
DNA
Imidazoline Receptor
Gamma-secretase
PLK
Hck
Stearoyl-CoA Desaturase (SCD)
ACK1
PDK
SGK
PAK
Histone Acetyltransferase
GST
Reverse Transcriptase
Platelet aggregation
OXPHOS
Free radical scavengers
Pyroptosis
Survivin
Thyroid hormone receptor(THR)
VDAC
IAP
Adiponectin Receptor
Amino Acids and Derivatives
YAP
Na-K-Cl cotransporter
Lipid
Liver X Receptor
PAI-1
PD-1/PD-L1
Cadherin
MRGPR
LRRK2
Transaminase
UGT
Succinate Receptor 1 (SUCNR1)
Kisspeptin
ribosome
CRISPR/Cas9
ROR
Dynamin
PANoptosis
DUB
Piezo Channel
Necroptosis
IDO
EBI2/GPR183
Arginase
gp120/CD4
Photosensitizer
AIM2
MELK
Aromatase
IRE1
PACAP
DNA gyrase
STING
GluCls
Retinoid Receptor
RXFP receptor
NADPH-oxidase
Antifolate
GlyT
Indoleamine 2,3-Dioxygenase (IDO)
Wee1
Cuproptosis
DHFR
DNA-PK
NR4A
E1/E2/E3 Enzyme
PROTAC Linker
ATP Citrate Lyase
Porcupine
Lipase
Cell Cycle Arrest
Glucokinase
HCAR
MNK
Complement System
IKZF
RANKL/RANK
Phosphorylase
Telomerase
Mdm2
GSNOR
ASCT
NAMPT
Carboxypeptidase
Gap Junction Protein
Lysosomal Autophagy
RAR/RXR
Neuropeptide W
Amylase
FABP
Huntingtin
Acetyl-CoA Carboxylase
FKBP
GPX
PKM
ASBT
Glutaminyl Cyclase
MIF
PAD
Thrombopoietin Receptor
Aminopeptidase
Urea Transporter
DAPK
p97
Kinesin
Taste receptor
TOPK
AAK1
FLAP
Motilin Receptor
DNA Alkylation
Neprilysin
ATM/ATR
Adenosine Deaminase
Liposome
GDNF
N-Acetylglucosaminyltransferase
ATG
Anion Exchanger
cGAS
Hippo pathway
MicroRNA
Galectin
LIM Kinase
Haspin Kinase
DPP-4
Orphan Receptor
Protease
ADC Cytotoxin
IGF-2R
Sodium-dependent phosphate transporter

Keywords