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TargetMol | Compound Library

FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules.

TargetMol's FDA-Approved & Pharmacopeia Drug Library collects 3280 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1010

FDA-Approved & Pharmacopeia Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • 3280 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
  • All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

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Library Customization | TargetMol Library Composition

Antibacterial
Antibiotic
Autophagy
Endogenous Metabolite
Apoptosis
Adrenergic Receptor
5-HT Receptor
AChR
COX
Parasite
Dopamine Receptor
Histamine Receptor
Antifungal
HIV Protease
Sodium Channel
Calcium Channel
Potassium Channel
DNA/RNA Synthesis
Glucocorticoid Receptor
Estrogen/progestogen Receptor
NF-κB
Topoisomerase
Cytochromes P450
Influenza Virus
SARS-CoV
Reactive Oxygen Species
Ferroptosis
PDE
GABA Receptor
RAAS
EGFR
Estrogen Receptor/ERR
Dehydrogenase
VEGFR
Mitophagy
HCV Protease
c-Kit
HSV
Microtubule Associated
Cholinesterase (ChE)
PDGFR
PPAR
Serotonin Transporter
Nucleoside Antimetabolite/Analog
ribosome
Prostaglandin Receptor
Reverse Transcriptase
Antioxidant
MAO
Norepinephrine
Progesterone Receptor
Virus Protease
TRP/TRPV Channel
iGluR
Proteasome
ATPase
Carbonic Anhydrase
HBV
HDAC
FGFR
TNF
Androgen Receptor
Antifection
JAK
MMP
DNA Alkylator/Crosslinker
Monoamine Oxidase
Opioid Receptor
Bcr-Abl
FLT
HIF/HIF Prolyl-Hydroxylase
Proton pump
ROS
Src
Adenosine Receptor
Antiviral
DPP-4
IL Receptor
MRP
Thrombin
Transferase
Tyrosine Kinases
c-Met/HGFR
HMG-CoA Reductase
NMDAR
PKC
AMPK
Lipoxygenase
Phosphatase
ALK
CDK
Drug Metabolite
GluR
NO Synthase
PI3K
Raf
STAT
Thyroid hormone receptor(THR)
Antifolate
Beta Amyloid
Interleukin
Mitochondrial Metabolism
PARP
Tyrosinase
Amino Acids and Derivatives
c-RET
DHFR
ERK
MEK
Retinoid Receptor
SGLT
DNA Alkylation
HSP
Nrf2
P-gp
Phospholipase
Serine Protease
TLR
Akt
Endothelin Receptor
Factor Xa
ABC Transporter
Chloride channel
HIF
Monoamine Transporter
mTOR
P2Y Receptor
ROCK
S1P Receptor
ADC Cytotoxin
Aromatase
CaMK
Caspase
CFTR
DNA gyrase
DNA Methyltransferase
HER
Histone Methyltransferase
Integrin
NADPH
Neurokinin receptor
P2X Receptor
p38 MAPK
PKA
Reductase
Sigma receptor
Trk receptor
Cysteine Protease
DNA
FXR
Glutathione Peroxidase
GNRH Receptor
Guanylate cyclase
Hedgehog/Smoothened
Hydroxylase
IκB/IKK
LPL Receptor
PGE Synthase
ROS Kinase
TAM Receptor
TGF-beta/Smad
Vasopressin Receptor
Wnt/beta-catenin
Annexin A
Anti-infection
Bcl-2 Family
FAK
Fatty Acid Synthase
GPCR
GPCR19
GSK-3
NOS
Xanthine Oxidase
AhR
Aryl Hydrocarbon Receptor
Cannabinoid Receptor
CaSR
Cell wall
c-Fms
CGRP Receptor
Decarboxylase
Gap Junction Protein
Histone Demethylase
Isocitrate Dehydrogenase (IDH)
Ligand for E3 Ligase
Lipid
Melatonin Receptor
Molecular Glues
MT Receptor
Neprilysin
NOD
NOD-like Receptor (NLR)
Serine/threonin kinase
Smo
UGT
Adenosine Deaminase
Aminopeptidase
Arginase
Aurora Kinase
BTK
CCR
CETP
Cholecystokinin Receptor
Complement System
CXCR
Free radical scavengers
Gamma-secretase
GluCls
Glucosidase
Hexokinase
IGF-1R
Imidazoline Receptor
LDL
Leukotriene Receptor
Melanocortin Receptor
MicroRNA
Na-K-Cl cotransporter
OAT
Oxytocin Receptor
p53
PAK
Sirtuin
Syk
Acyltransferase
Adiponectin Receptor
Beta-Secretase
CRM1
CSF-1R
DUB
DYRK
Ephrin Receptor
Epigenetic Reader Domain
GHSR
Glutathione reductase
GlyT
GST
IFNAR
Immunology/Inflammation related
Indoleamine 2,3-Dioxygenase (IDO)
Integrase
IRE1
JNK
Kras
Ligands for Target Protein for PROTAC
LTR
MAPK
Monocarboxylate transporter
Na+/Ca2+ Exchanger
PAFR
PDK
PKM
Platelet aggregation
PLK
Protease-activated Receptor
Ras
Rho
ROR
RSV
S6 Kinase
Telomerase
Thrombopoietin Receptor
TOPK
Vitamin
YAP
ACK1
Advanced Glycation End Products
Angiotensin-converting Enzyme (ACE)
Anion Exchanger
Aquaporin
ATP Citrate Lyase
BACE
cAMP
Casein Kinase
Chk
CRFR
CRISPR/Cas9
DNA-PK
Dynamin
Epoxide Hydrolase
FAAH
Glucagon Receptor
Glucokinase
gp120/CD4
GRK
Hck
HCN Channel
Histone Acetyltransferase
Hydrogenase
IAP
IRAK
Lipase
Liver X Receptor
Mdm2
MTH1
Mucin
Myosin
N-Acetylglucosaminyltransferase
NADPH-oxidase
NPC1L1
PAD
PD-1/PD-L1
Phosphorylase
PROTAC Linker
Pyroptosis
RANKL/RANK
Somatostatin
STING
Taste receptor
transporter
VDA

Keywords