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Oxypeucedanin
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Catalog No. T3S0081Cas No. 737-52-0
Alias Oxypeucadanin, (+-)-Oxypeucedanin
1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocker of the hKv1.5 channel and it prolongs the APD; therefore, it is an excellent candidate as an antiarrhythmic drug for atrial fibrillation.
Oxypeucedanin
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Purity: 98.85%
Catalog No. T3S0081Alias Oxypeucadanin, (+-)-OxypeucedaninCas No. 737-52-0
1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocker of the hKv1.5 channel and it prolongs the APD; therefore, it is an excellent candidate as an antiarrhythmic drug for atrial fibrillation.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $52 | In Stock | In Stock | |
| 5 mg | $127 | In Stock | In Stock | |
| 10 mg | $198 | In Stock | In Stock | |
| 25 mg | $347 | In Stock | In Stock | |
| 50 mg | $515 | In Stock | In Stock | |
| 100 mg | $733 | In Stock | In Stock | |
| 200 mg | $987 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Batch Information
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Purity:98.85%
Color:White
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Product Introduction
Oxypeucedanin AI Summary
Oxypeucedanin displays a diverse range of bioactivities across various biological targets. It inhibits Human Jumonji Domain Containing 2E (JMJD2E) with a potency of 31622.8 nM and the interaction between Thyroid Hormone Receptor and Steroid Receptor Coregulator 2 at 70794.6 nM. Additionally, it inhibits Aldehyde Dehydrogenase 1 (ALDH1A1) with a potency of 39810.7 nM and modulates lipid storage in Drosophila S3 Cells at 3662.6 nM. Oxypeucedanin also exhibits potent inhibition of DNA Polymerase Beta with a potency of 1000.0 nM and affects Ran-regulated importin-beta cargo by inhibiting Importin beta complex formation with a potency of 125892.5 nM. The compound acts as a delayed death inhibitor of the malarial parasite plastid after a 96-hour incubation, with a potency of 369.6 nM, and inhibits the generation of Cell Surface uPA at 354.8 nM. Furthermore, it induces DNA re-replication in MCF 10a normal breast cells and SW480 colon adenocarcinoma cells with potencies of 580.5 nM and 14581.0 nM, respectively. Oxypeucedanin inhibits human tyrosyl-DNA phosphodiesterase 1 (TDP1) in the presence of CPT with a potency of 18356.4 nM and the PTHR with a potency of 39810.7 nM in a primary screen. It also demonstrates antiviral activity against HIV in human H9 cells, with an EC50 value of 1.0 µg/mL..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | 1. Oxypeucedanin ((+-)-Oxypeucedanin) has novel anticancer effect, mediated via induction of G2-M cell cycle arrest and apoptosis in human prostate carcinoma DU145 cells. 2. Oxypeucedanin is a kind of open-channel blocker of the hKv1.5 channel and it prolongs the APD; therefore, it is an excellent candidate as an antiarrhythmic drug for atrial fibrillation. |
| Synonyms | Oxypeucadanin, (+-)-Oxypeucedanin |
| Molecular Weight | 286.28 |
| Formula | C16H14O5 |
| Cas No. | 737-52-0 |
| Smiles | CC1(C)OC1COc1c2ccoc2cc2oc(=O)ccc12 |
| Relative Density. | 1.320 g/cm3 (Predicted) |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 6.88 mg/mL (24.03 mM), Sonication is recommended.  | |||||||||||||||||||||||||
| In Vivo Formulation | 10% DMSO+40% PEG300+5% Tween 80+45% Saline: 1 mg/mL (3.49 mM), Sonication is recommended. Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions. | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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