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GluR6 antagonist-1

🥰Excellent

Catalog No. T9723Cas No. 323176-64-3

GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.

GluR6 antagonist-1

🥰Excellent

Purity: 99.89%

Catalog No. T9723Cas No. 323176-64-3

GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.

Pack Size	Price	USA Warehouse	Global Warehouse
2 mg	$32	In Stock	In Stock
5 mg	$53	In Stock	In Stock
10 mg	$83	In Stock	In Stock
25 mg	$140	In Stock	In Stock
50 mg	$208	In Stock	In Stock
100 mg	$310	In Stock	In Stock
200 mg	$433	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$59	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Batch Information

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Purity:99.89%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description

GluR6 antagonist-1 inhibits the pY binding site of tyrosine kinase p56lck SH2 domain.

Chemical Properties

Molecular Weight	302.78
Formula	C₁₅H₁₁ClN₂OS
Cas No.	323176-64-3
Smiles	ClC=1C=2C(SC1C(NCC=3C=CC=NC3)=O)=CC=CC2
Relative Density.	1.380 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 55 mg/mL (181.65 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.3027 mL	16.5136 mL	33.0273 mL	165.1364 mL
5 mM	0.6605 mL	3.3027 mL	6.6055 mL	33.0273 mL
10 mM	0.3303 mL	1.6514 mL	3.3027 mL	16.5136 mL
20 mM	0.1651 mL	0.8257 mL	1.6514 mL	8.2568 mL
50 mM	0.0661 mL	0.3303 mL	0.6605 mL	3.3027 mL
100 mM	0.0330 mL	0.1651 mL	0.3303 mL	1.6514 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc