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Ajmaline

🥰Excellent
Catalog No. T4550Cas No. 4360-12-7
Alias Tachmalin, Raugalline, Cardiorythmine, (+)-Ajmaline

Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.

Ajmaline
Other Forms of Ajmaline:
Ajmaline hydrochlorideT4550L4410-48-4
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Ajmaline

🥰Excellent
Purity: 99.87%
Catalog No. T4550Alias Tachmalin, Raugalline, Cardiorythmine, (+)-AjmalineCas No. 4360-12-7
Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
100 mg$40In StockIn Stock
500 mg$92-In Stock
1 mL x 10 mM (in DMSO)$29In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.87%
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Product Introduction

Bioactivity
Description
Ajmaline (Cardiorythmine) is a class Ia anti-arrhythmic compound that is widely used for the diagnosis of Brugada syndrome and the acute treatment of atrial or ventricular tachycardia. Ajmaline inhibits cardiac Kv1.5 and Kv4.3 channels at therapeutic concentrations.
SynonymsTachmalin, Raugalline, Cardiorythmine, (+)-Ajmaline
Chemical Properties
Molecular Weight326.43
FormulaC20H26N2O2
Cas No.4360-12-7
SmilesO[C@H]1C23[C@]([C@]4(N5[C@@](C2)(C1C(C4)[C@H](CC)[C@H]5O)[H])[H])(N(C)C=6C3=CC=CC6)[H]
Relative Density.1.1117 g/cm3 (Estimated)
ColorWhite
AppearanceSolid
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 40 mg/mL (122.54 mM), Sonication is recommended.
Chloroform: Soluble
In Vivo Formulation
10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (6.13 mM), Sonication is recommended.
Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM3.0634 mL15.3172 mL30.6344 mL153.1722 mL
5 mM0.6127 mL3.0634 mL6.1269 mL30.6344 mL
10 mM0.3063 mL1.5317 mL3.0634 mL15.3172 mL
20 mM0.1532 mL0.7659 mL1.5317 mL7.6586 mL
50 mM0.0613 mL0.3063 mL0.6127 mL3.0634 mL
100 mM0.0306 mL0.1532 mL0.3063 mL1.5317 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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2 Enter the in vivo formulation:
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Keywords

ventriculartachyarrhythmiaSodiumChannelsodium channelSodium ChannelNa+ channelsNa channelsInhibitorinhibitcurrentanti-arrhythmicAjmaline
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