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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3230 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3230 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Antibacterial
COX
Dopamine Receptor
Histamine Receptor
Antibiotic
DNA/RNA Synthesis
Sodium Channel
Potassium Channel
VEGFR
EGFR
Calcium Channel
AChR
Parasite
PI3K
Glucocorticoid Receptor
Reactive Oxygen Species
CDK
Cytochromes P450
Topoisomerase
FLT
HIV Protease
NF-κB
PDGFR
PPAR
GABA Receptor
JAK
HDAC
c-Kit
FGFR
Microtubule Associated
Estrogen/progestogen Receptor
c-Met/HGFR
Estrogen Receptor/ERR
Ferroptosis
Antifungal
Prostaglandin Receptor
Dehydrogenase
mTOR
Mitophagy
SARS-CoV
Src
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Nucleoside Antimetabolite/Analog
Androgen Receptor
Tyrosine Kinases
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iGluR
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MEK
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p38 MAPK
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Histone Methyltransferase
RAAS
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ERK
HIF/HIF Prolyl-Hydroxylase
Phosphatase
AMPK
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HBV
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GSK-3
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OX Receptor
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Hydroxylase
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ribosome
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transporter
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