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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

We selected 3660 drugs with demonstrated or potential anticancer activity—including FDA-approved drugs and those in clinical trials—to form an Anticancer Drug Library for tumor-related research and anticancer drug screening

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3660 drugs with anti-cancer activity or potential anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);;
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Antibiotic
COX
Dopamine Receptor
Histamine Receptor
Potassium Channel
ROS
Parasite
NF-κB
Sodium Channel
Calcium Channel
EGFR
VEGFR
PI3K
Reactive Oxygen Species
AChR
Cytochromes P450
Akt
CDK
Glucocorticoid Receptor
Topoisomerase
FLT
HIV Protease
JAK
PPAR
p38 MAPK
Estrogen Receptor/ERR
GABA Receptor
ERK
Virus Protease
mTOR
PDGFR
Antifungal
HDAC
FGFR
c-Met/HGFR
c-Kit
Estrogen/progestogen Receptor
Microtubule Associated
Ferroptosis
Prostaglandin Receptor
Interleukin
SARS-CoV
TNF
Ras
iGluR
Caspase
Influenza Virus
Nucleoside Antimetabolite/Analog
Dehydrogenase
Mitophagy
Adenosine Receptor
Androgen Receptor
Src
STAT
Tyrosine Kinases
Epigenetic Reader Domain
Bcr-Abl
Bcl-2 Family
Serotonin Transporter
PDE
PARP
HSV
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Opioid Receptor
TRP/TRPV Channel
MMP
Wnt/beta-catenin
P-gp
Drug Metabolite
GPCR
ALK
HSP
TLR
MEK
ATPase
PKC
Histone Methyltransferase
AMPK
HIF/HIF Prolyl-Hydroxylase
JNK
Aurora Kinase
MDM-2/p53
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Phosphatase
Norepinephrine
Mitochondrial Metabolism
Beta Amyloid
NMDAR
GSK-3
Trk receptor
HER
Proton pump
RAAS
c-RET
ROS Kinase
DNA Alkylator/Crosslinker
Nrf2
TGF-beta/Smad
Kras
c-Fms
NO Synthase
IGF-1R
HCV Protease
Endothelin Receptor
TAM Receptor
Progesterone Receptor
GluR
FAK
Reverse Transcriptase
IL Receptor
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CFTR
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Chk
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Retinoid Receptor
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GNRH Receptor
MAO
Vasopressin Receptor
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Glutathione Peroxidase
IDO
DNA Methyltransferase
NOD-like Receptor (NLR)
IκB/IKK
Neurokinin receptor
Indoleamine 2,3-Dioxygenase (IDO)
Kinesin
Mdm2
IRAK
Serine Protease
Casein Kinase
Chloride channel
FXR
CaMK
Integrin
Reductase
CSF-1R
Phospholipase
Antifection
Ligands for E3 Ligase
PAK
Melanocortin Receptor
GPCR19
PERK
CCR
DNA
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Leukotriene Receptor
NADPH
Smo
RIP kinase
OX Receptor
Aromatase
PD-1/PD-L1
Hydroxylase
Pim
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IKZF
CaSR
Photosensitizer
Ephrin Receptor
Oxytocin Receptor
Glucagon Receptor
DPP-4
RSV
Monoamine Transporter
ribosome
Serine/threonin kinase
IFNAR
Tie-2
Cholecystokinin Receptor
PYK2
UGT
CRFR
GHSR
glycosidase
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Bradykinin Receptor
Xanthine Oxidase
OXPHOS
STING
Na-K-Cl cotransporter
Telomerase
AhR
Glucosidase
Fatty Acid Synthase
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Wee1
PGE Synthase
Aminopeptidase
NAMPT
GST
Amino Acids and Derivatives
Immunology/Inflammation related
DUB
LTR
Monocarboxylate transporter
Melatonin Receptor
IRE1
DNA gyrase
FKBP
CGRP Receptor
MLK
YAP
Annexin A
Neuropeptide Y Receptor
PDK
TOPK
CRM1
Glutaminase
Cuproptosis
Arginase
DYRK
c-Myc
Rho
Liver X Receptor
Gap Junction Protein
MicroRNA
ROR
Cell Cycle Arrest
Hexokinase
MNK
OAT
NEDD8
PROTAC Linker
ATP Citrate Lyase
NOS
Cysteine Protease
KSP
Free radical scavengers
Necroptosis
RANKL/RANK
MT Receptor
transporter
Beta-Secretase
Acyltransferase
Decarboxylase
FOXO
Adenosine Deaminase
MIF
Thrombopoietin Receptor
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Ligands for Target Protein for PROTAC
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VDA
NR4A
FAAH
Porcupine
CD73
Imidazoline Receptor
LDL
PTEN
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LPA Receptor
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gp120/CD4
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cAMP
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E3 Ligase Ligand-Linker Conjugates
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Neprilysin
Liposome
Neurotensin Receptor
GlyT
PAD
Methionine Adenosyltransferase (MAT)
Aquaporin
Ferroportin
Drug-Linker Conjugates for ADC
PGC-1α

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