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Anti-Cancer Drug Library

Catalog No. L2150
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 3080 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 3080 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

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Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2150)

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Library Composition

Autophagy (433)
Apoptosis (410)
5-HT Receptor (200)
Endogenous Metabolite (173)
Adrenergic Receptor (169)
Antibacterial (144)
COX (135)
Dopamine Receptor (126)
Histamine Receptor (125)
Antibiotic (119)
DNA/RNA Synthesis (116)
Sodium Channel (95)
Calcium Channel (86)
Potassium Channel (85)
VEGFR (81)
EGFR (76)
AChR (72)
Parasite (68)
PI3K (65)
Reactive Oxygen Species (61)
Glucocorticoid Receptor (61)
P450 (58)
FLT (55)
CDK (53)
Topoisomerase (53)
NF-κB (53)
HIV Protease (53)
PDGFR (52)
PPAR (51)
GABA Receptor (49)
c-Kit (48)
JAK (48)
FGFR (46)
HDAC (44)
Prostaglandin Receptor (42)
Ferroptosis (42)
Estrogen/progestogen Receptor (41)
Microtubule Associated (41)
Antifungal (41)
mTOR (41)
c-Met/HGFR (40)
Dehydrogenase (39)
Mitophagy (38)
Influenza Virus (37)
Estrogen Receptor/ERR (36)
Nucleoside Antimetabolite/Analog (34)
Src (34)
SARS-CoV (32)
iGluR (32)
Adenosine Receptor (31)
Tyrosine Kinases (31)
Androgen Receptor (31)
PDE (30)
GPR (30)
Opioid Receptor (29)
Bcr-Abl (28)
Raf (28)
Serotonin Transporter (25)
HER (25)
Akt (24)
ATPase (24)
Norepinephrine (24)
Aurora Kinase (23)
PARP (23)
TRP/TRPV Channel (22)
p38 MAPK (21)
MEK (21)
TNF (21)
HSV (21)
P-gp (21)
Epigenetic Reader Domain (21)
Proton pump (20)
PKC (20)
Virus Protease (20)
NMDAR (20)
HSP (20)
BTK (20)
DNA Alkylator/Crosslinker (19)
ALK (18)
HIF/HIF Prolyl-Hydroxylase (18)
RAAS (18)
ERK (18)
c-RET (17)
Trk receptor (17)
ROS (17)
HBV (17)
GSK-3 (16)
HCV Protease (16)
CXCR (16)
Phosphatase (16)
AMPK (16)
Caspase (15)
GNRH Receptor (15)
BCL (15)
SGLT (15)
Endothelin Receptor (15)
Drug Metabolite (15)
MMP (15)
Carbonic Anhydrase (15)
TAM Receptor (14)
Retinoid Receptor (14)
STAT (14)
Progesterone Receptor (14)
Histone Methyltransferase (14)
c-Fms (14)
Guanylate cyclase (13)
IL Receptor (13)
Chk (13)
E1/E2/E3 Enzyme (13)
Proteasome (13)
Reverse Transcriptase (13)
DNA-PK (13)
DNA Alkylation (12)
p53 (12)
TGF-beta/Smad (12)
MAO (12)
HIF (12)
S1P Receptor (12)
LPL Receptor (12)
CFTR (12)
Gamma-secretase (11)
Cannabinoid Receptor (11)
GluR (11)
Neurokinin receptor (11)
HMG-CoA Reductase (11)
Interleukin (11)
Mitochondrial Metabolism (11)
P2X Receptor (11)
MRP (11)
PKA (11)
Antifolate (11)
Lipoxygenase (11)
Monoamine Oxidase (11)
Transferase (11)
IGF-1R (11)
DHFR (11)
Hedgehog/Smoothened (11)
Nrf2 (10)
Antioxidant (10)
FAK (10)
Wnt/beta-catenin (10)
Syk (10)
Vasopressin Receptor (10)
AChE (10)
P2Y Receptor (10)
ROCK (10)
Indoleamine 2,3-Dioxygenase (IDO) (9)
Chloride channel (9)
S6 Kinase (9)
Beta Amyloid (9)
IAP (9)
Antifection (9)
TLR (9)
CSF-1R (9)
Phospholipase (8)
CaMK (8)
Sigma receptor (8)
ROS Kinase (8)
PLK (8)
Ras (8)
JNK (8)
ATM/ATR (8)
NADPH (8)
Smo (8)
DNA Methyltransferase (8)
OX Receptor (8)
Casein Kinase (8)
Kinesin (7)
Mdm2 (7)
Ligand for E3 Ligase (7)
Aromatase (7)
Monoamine Transporter (7)
Sirtuin (7)
Pim (7)
ABC (7)
Antiviral (7)
Integrin (7)
Thrombin (7)
cholecystokinin (7)
Glucagon Receptor (7)
IκB/IKK (6)
IRAK (6)
DNA (6)
NO Synthase (6)
PAK (6)
Histone Demethylase (6)
RIP kinase (6)
Leukotriene Receptor (6)
Isocitrate Dehydrogenase (IDH) (6)
Glutathione Peroxidase (6)
Bradykinin Receptor (6)
CCR (6)
Ephrin Receptor (5)
Hydroxylase (5)
DPP-4 (5)
Fatty Acid Synthase (5)
Tie-2 (5)
GHSR (5)
NOD (5)
ribosome (5)
PGE Synthase (5)
FXR (5)
IFNAR (5)
Serine Protease (5)
GPCR19 (5)
PDK (4)
Serine/threonin kinase (4)
Amino Acids and Derivatives (4)
Aminopeptidase (4)
Melanocortin Receptor (4)
AhR (4)
CRFR (4)
Tyrosinase (4)
Annexin A (4)
LTR (4)
IDO (4)
KSP (4)
Oxytocin Receptor (4)
Aryl Hydrocarbon Receptor (4)
Somatostatin (4)
Wee1 (4)
PD-1/PD-L1 (4)
Molecular Glues (4)
CaSR (4)
CGRP Receptor (4)
Xanthine Oxidase (4)
Melatonin Receptor (4)
RSV (3)
Reductase (3)
YAP (3)
Monocarboxylate transporter (3)
NAMPT (3)
GST (3)
DUB (3)
Neuropeptide Y Receptor (3)
Protease-activated Receptor (3)
Liver X Receptor (3)
Na-K-Cl cotransporter (3)
OAT (3)
UGT (3)
DNA gyrase (3)
NOD-like Receptor (NLR) (3)
MT Receptor (3)
MAPK (3)
Rho (3)
ROR (3)
Cysteine Protease (3)
STING (3)
Free radical scavengers (3)
Hexokinase (3)
Adenosine deaminase (3)
CRM1 (3)
PERK (2)
Discoidin Domain Receptor (DDR) (2)
Factor Xa (2)
LPA Receptor (2)
VDA (2)
Cell wall (2)
Gap Junction Protein (2)
PYK2 (2)
transporter (2)
Porcupine (2)
Glucosidase (2)
BCRP (2)
Imidazoline Receptor (2)
MLK (2)
Beta-Secretase (2)
Telomerase (2)
Acyltransferase (2)
PROTAC Linker (2)
LDL (2)
NEDD8 (2)
Lipid (2)
p97 (2)
CD73 (2)
Decarboxylase (2)
Ligands for Target Protein for PROTAC (2)
Arginase (2)
CAT (2)
IRE1 (2)
NOS (2)
PROTACs (2)
ATP Citrate Lyase (2)
NPC1L1 (1)
DYRK (1)
Platelet aggregation (1)
Lipase (1)
BMI-1 (1)
MALT (1)
RAR/RXR  (1)
Na+/Ca2+ Exchanger (1)
NADPH-oxidase (1)
BACE (1)
Hydrogenase (1)
ACK (1)
Complement System (1)
Survivin (1)
ASK (1)
Motilin Receptor (1)
Histone Acetyltransferase (1)
Adiponectin receptor (1)
PAFR (1)
MTH1 (1)
GRK (1)
MNK (1)
Glutathione reductase (1)
PAI-1 (1)
GlyT (1)
Anion Exchanger (1)
HCN Channel (1)
advanced glycation end products (1)
FAAH (1)
Thrombopoietin Receptor (1)
cAMP (1)
PAD (1)
GluCls (1)
Pyroptosis (1)
TOPK (1)
KLF (1)
SGK (1)
GTPase (1)
Galectin (1)
c-Myc (1)
Kisspeptin (1)
Aquaporin (1)
N-Acetylglucosaminyltransferase (1)
Hck (1)
PI4K (1)
MELK (1)
Glucokinase (1)
Stemness kinase (1)
Glutaminase (1)
Neprilysin (1)
Hippo pathway (1)
Immunology/Inflammation related (1)
Methionine Adenosyltransferase (MAT) (1)
Myosin (1)
Thioredoxin (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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