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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

We selected 3660 drugs with demonstrated or potential anticancer activity—including FDA-approved drugs and those in clinical trials—to form an Anticancer Drug Library for tumor-related research and anticancer drug screening

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library

size

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3660 drugs with anti-cancer activity or potential anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);;
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Antibiotic
Dopamine Receptor
COX
Histamine Receptor
Potassium Channel
ROS
NF-κB
Parasite
Sodium Channel
Calcium Channel
EGFR
VEGFR
PI3K
Reactive Oxygen Species
AChR
Cytochromes P450
Akt
CDK
Glucocorticoid Receptor
Topoisomerase
FLT
HIV Protease
JAK
PPAR
GABA Receptor
p38 MAPK
Estrogen Receptor/ERR
Virus Protease
mTOR
ERK
PDGFR
FGFR
Antifungal
HDAC
c-Met/HGFR
Estrogen/progestogen Receptor
Microtubule Associated
c-Kit
Ferroptosis
Prostaglandin Receptor
Caspase
SARS-CoV
Interleukin
Influenza Virus
Ras
TNF
iGluR
Nucleoside Antimetabolite/Analog
Dehydrogenase
Mitophagy
Androgen Receptor
Adenosine Receptor
Src
STAT
Bcr-Abl
Bcl-2 Family
Tyrosine Kinases
Epigenetic Reader Domain
BTK
Serotonin Transporter
HSV
PDE
PARP
Raf
MMP
TRP/TRPV Channel
Opioid Receptor
Drug Metabolite
Wnt/beta-catenin
P-gp
GPCR
ALK
HSP
ATPase
MEK
TLR
Histone Methyltransferase
PKC
AMPK
Aurora Kinase
HIF/HIF Prolyl-Hydroxylase
JNK
MDM-2/p53
HBV
Phosphatase
Norepinephrine
Mitochondrial Metabolism
Beta Amyloid
NMDAR
GSK-3
Trk receptor
HER
RAAS
c-RET
Proton pump
ROS Kinase
TGF-beta/Smad
DNA Alkylator/Crosslinker
Nrf2
Kras
c-Fms
IGF-1R
Endothelin Receptor
TAM Receptor
HCV Protease
NO Synthase
FAK
Progesterone Receptor
GluR
Antifolate
IL Receptor
Reverse Transcriptase
Carbonic Anhydrase
Antioxidant
E1/E2/E3 Enzyme
Cholinesterase (ChE)
CFTR
ROCK
CXCR
Chk
PKA
ATM/ATR
Molecular Glues
SGLT
Retinoid Receptor
LPL Receptor
HMG-CoA Reductase
Gamma-secretase
MAPK
S1P Receptor
GNRH Receptor
MAO
Lipoxygenase
DHFR
Monoamine Oxidase
p53
Vasopressin Receptor
HIF
Transferase
Antiviral
Anti-infection
Guanylate cyclase
Cannabinoid Receptor
MRP
P2X Receptor
NOD
DNA-PK
DNA Alkylation
ADC Cytotoxin
Tyrosinase
P2Y Receptor
Syk
IAP
ABC Transporter
Sigma receptor
Hedgehog/Smoothened
S6 Kinase
Indoleamine 2,3-Dioxygenase (IDO)
Kinesin
Angiotensin-converting Enzyme (ACE)
PLK
Isocitrate Dehydrogenase (IDH)
PROTACs
Histone Demethylase
Reductase
IκB/IKK
Neurokinin receptor
IDO
DNA Methyltransferase
NOD-like Receptor (NLR)
Glutathione Peroxidase
Antifection
Ligands for E3 Ligase
Serine Protease
Mdm2
IRAK
Casein Kinase
Integrin
CSF-1R
Phospholipase
CaMK
Chloride channel
FXR
RIP kinase
OX Receptor
GPCR19
PAK
Melanocortin Receptor
PERK
CCR
DNA
Sirtuin
Smo
NADPH
Leukotriene Receptor
DPP-4
PD-1/PD-L1
Hydroxylase
Proteasome
Pim
Thrombin
IKZF
PYK2
UGT
Glucagon Receptor
RSV
Photosensitizer
Ephrin Receptor
Aromatase
Oxytocin Receptor
Monoamine Transporter
ribosome
Tie-2
Cholecystokinin Receptor
IFNAR
Serine/threonin kinase
Fatty Acid Synthase
Somatostatin
Wee1
PGE Synthase
Aminopeptidase
CaSR
CRFR
GHSR
glycosidase
Glucosidase
Na-K-Cl cotransporter
Telomerase
AhR
Aryl Hydrocarbon Receptor
Bradykinin Receptor
Xanthine Oxidase
OXPHOS
STING
CRM1
Glutaminase
Cuproptosis
Amino Acids and Derivatives
Immunology/Inflammation related
DUB
NAMPT
GST
LTR
TOPK
YAP
Annexin A
Neuropeptide Y Receptor
PDK
Monocarboxylate transporter
Melatonin Receptor
IRE1
DNA gyrase
FKBP
CGRP Receptor
MLK
MIF
Thrombopoietin Receptor
BCRP
Survivin
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
MicroRNA
ROR
Cell Cycle Arrest
Hexokinase
OAT
MNK
Arginase
DYRK
c-Myc
Rho
Liver X Receptor
Gap Junction Protein
NEDD8
PROTAC Linker
ATP Citrate Lyase
Beta-Secretase
Acyltransferase
Decarboxylase
FOXO
Adenosine Deaminase
Necroptosis
RANKL/RANK
MT Receptor
transporter
NOS
Cysteine Protease
KSP
Free radical scavengers
PGC-1α
Adenylate cyclase
ASK
p97
Ligands for Target Protein for PROTAC
Galectin
PANoptosis
PI4K
Complement System
Na+/Ca2+ Exchanger
Factor Xa
HCN Channel
Histone Acetyltransferase
PAI-1
MELK
VDA
NR4A
FAAH
Porcupine
CD73
Imidazoline Receptor
Thyroid hormone receptor(THR)
Kisspeptin
GRK
Lipid
PSMA
LPA Receptor
SGK
LDL
PTEN
Cadherin
Huntingtin
Pyroptosis
Vitamin
Neurotensin Receptor
GlyT
PAD
Methionine Adenosyltransferase (MAT)
Aquaporin
Apelin receptor
Lipase
Glucokinase
PAFR
MTH1
HCAR
KLF
gp120/CD4
GTPase
cAMP
Dipeptidyl Peptidase
Platelet aggregation
Hydrogenase
Factor VIIa
N-Acetylglucosaminyltransferase
ATG
Adiponectin Receptor
Anion Exchanger
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
NPC1L1
SIK
Myosin
Thioredoxin
Glutathione reductase
Neprilysin
Liposome
Advanced Glycation End Products
BACE
Cell wall
OCT
Hck
Stemness kinase
Arp2/3 Complex
ACK1
BMI-1
MALT
MyD88
Prolyl Endopeptidase (PREP)
GluCls
RXFP receptor
NADPH-oxidase
Drug-Linker Conjugates for ADC
Ferroportin

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