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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

We selected 3660 drugs with demonstrated or potential anticancer activity—including FDA-approved drugs and those in clinical trials—to form an Anticancer Drug Library for tumor-related research and anticancer drug screening

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library

sizeIn stock

  • 1 mg
  • 10 µL x 10 mM (in DMSO)
  • 20 µL x 10 mM (in DMSO)
  • 30 µL x 10 mM (in DMSO)
  • 50 µL x 10 mM (in DMSO)
  • 100 µL x 10 mM (in DMSO)
  • 250 µL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3660 drugs with anti-cancer activity or potential anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);;
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Antibiotic
Dopamine Receptor
COX
Histamine Receptor
Potassium Channel
Parasite
ROS
NF-κB
Sodium Channel
Calcium Channel
EGFR
VEGFR
PI3K
Reactive Oxygen Species
AChR
Cytochromes P450
Akt
CDK
Glucocorticoid Receptor
Topoisomerase
FLT
HIV Protease
JAK
p38 MAPK
Estrogen Receptor/ERR
PPAR
GABA Receptor
Virus Protease
ERK
mTOR
PDGFR
Antifungal
HDAC
FGFR
c-Met/HGFR
Estrogen/progestogen Receptor
c-Kit
Microtubule Associated
Ferroptosis
Caspase
Interleukin
SARS-CoV
Prostaglandin Receptor
iGluR
Influenza Virus
TNF
Ras
Nucleoside Antimetabolite/Analog
Dehydrogenase
Mitophagy
Adenosine Receptor
Androgen Receptor
Src
STAT
Tyrosine Kinases
Bcr-Abl
Epigenetic Reader Domain
Bcl-2 Family
Serotonin Transporter
PDE
HSV
PARP
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TRP/TRPV Channel
Opioid Receptor
MMP
Wnt/beta-catenin
Drug Metabolite
P-gp
GPCR
HSP
ALK
ATPase
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MEK
Histone Methyltransferase
PKC
AMPK
JNK
Aurora Kinase
HIF/HIF Prolyl-Hydroxylase
Phosphatase
HBV
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MDM-2/p53
Mitochondrial Metabolism
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GSK-3
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RAAS
Trk receptor
HER
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TGF-beta/Smad
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c-RET
ROS Kinase
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HCV Protease
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IGF-1R
TAM Receptor
Progesterone Receptor
GluR
FAK
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IL Receptor
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CFTR
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Chk
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Retinoid Receptor
HMG-CoA Reductase
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DHFR
LPL Receptor
GNRH Receptor
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S1P Receptor
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IDO
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Indoleamine 2,3-Dioxygenase (IDO)
IκB/IKK
PLK
Neurokinin receptor
DNA Methyltransferase
NOD-like Receptor (NLR)
Kinesin
Mdm2
Chloride channel
Integrin
Serine Protease
FXR
CSF-1R
Antifection
Ligands for E3 Ligase
CaMK
Casein Kinase
Phospholipase
IRAK
NADPH
PERK
Leukotriene Receptor
RIP kinase
Smo
PAK
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OX Receptor
DNA
GPCR19
Sirtuin
Melanocortin Receptor
Pim
Hydroxylase
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PD-1/PD-L1
IKZF
IFNAR
Tie-2
Cholecystokinin Receptor
Photosensitizer
Serine/threonin kinase
PYK2
UGT
Glucagon Receptor
Monoamine Transporter
DPP-4
Ephrin Receptor
RSV
Aromatase
ribosome
Oxytocin Receptor
CaSR
Aryl Hydrocarbon Receptor
Na-K-Cl cotransporter
Glucosidase
Fatty Acid Synthase
Bradykinin Receptor
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glycosidase
Telomerase
Wee1
OXPHOS
PGE Synthase
STING
Aminopeptidase
CRFR
GHSR
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Monocarboxylate transporter
CRM1
Amino Acids and Derivatives
YAP
LTR
TOPK
Melatonin Receptor
NAMPT
Glutaminase
Immunology/Inflammation related
IRE1
Annexin A
DNA gyrase
Neuropeptide Y Receptor
DUB
GST
FKBP
PDK
CGRP Receptor
Cuproptosis
MLK
MicroRNA
NOS
ROR
NEDD8
Arginase
DYRK
Necroptosis
MIF
c-Myc
Rho
Cell Cycle Arrest
Cysteine Protease
Liver X Receptor
RANKL/RANK
MT Receptor
Hexokinase
PROTAC Linker
KSP
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Beta-Secretase
OAT
MNK
Survivin
Acyltransferase
Free radical scavengers
transporter
Decarboxylase
FOXO
Adenosine Deaminase
Discoidin Domain Receptor (DDR)
Gap Junction Protein
Protease-activated Receptor
PGC-1α
Thyroid hormone receptor(THR)
Ligands for Target Protein for PROTAC
Na+/Ca2+ Exchanger
Factor Xa
VDA
Galectin
Kisspeptin
NR4A
Adenylate cyclase
LDL
GRK
HCN Channel
FAAH
PTEN
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CD73
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ASK
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OCT
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E3 Ligase Ligand-Linker Conjugates
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Neprilysin
Hippo pathway
KLF
Aquaporin
RXFP receptor
Platelet aggregation
NADPH-oxidase
BMI-1
Liposome
Ferroportin
Drug-Linker Conjugates for ADC

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