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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

We selected 3,230 drugs with demonstrated or potential anticancer activity—including FDA-approved drugs and those in clinical trials—to form an Anticancer Drug Library for tumor-related research and anticancer drug screening

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3660 drugs with anti-cancer activity or potential anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);;
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

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Apoptosis
Autophagy
Endogenous Metabolite
Antibacterial
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Antibiotic
Dopamine Receptor
COX
Histamine Receptor
Potassium Channel
NF-κB
Parasite
ROS
Sodium Channel
Calcium Channel
VEGFR
EGFR
PI3K
Reactive Oxygen Species
AChR
Cytochromes P450
Akt
CDK
Glucocorticoid Receptor
Topoisomerase
HIV Protease
FLT
p38 MAPK
Estrogen Receptor/ERR
PPAR
JAK
GABA Receptor
Virus Protease
mTOR
Antifungal
ERK
PDGFR
HDAC
FGFR
c-Met/HGFR
Estrogen/progestogen Receptor
c-Kit
Microtubule Associated
Prostaglandin Receptor
Ferroptosis
Interleukin
Caspase
SARS-CoV
Influenza Virus
iGluR
TNF
Ras
Nucleoside Antimetabolite/Analog
Dehydrogenase
Mitophagy
Androgen Receptor
Adenosine Receptor
Src
Tyrosine Kinases
Bcl-2 Family
STAT
Bcr-Abl
Epigenetic Reader Domain
Serotonin Transporter
PDE
HSV
PARP
Opioid Receptor
TRP/TRPV Channel
Raf
Wnt/beta-catenin
Drug Metabolite
MMP
P-gp
GPCR
HSP
ALK
ATPase
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MEK
PKC
Histone Methyltransferase
AMPK
JNK
Aurora Kinase
HIF/HIF Prolyl-Hydroxylase
Phosphatase
HBV
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Mitochondrial Metabolism
Beta Amyloid
MDM-2/p53
GSK-3
NMDAR
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DNA Alkylator/Crosslinker
RAAS
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c-RET
HER
TGF-beta/Smad
Nrf2
ROS Kinase
Kras
c-Fms
HCV Protease
Endothelin Receptor
IGF-1R
NO Synthase
Progesterone Receptor
GluR
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FAK
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CXCR
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PKA
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Molecular Glues
Cholinesterase (ChE)
Chk
Lipoxygenase
SGLT
ATM/ATR
Retinoid Receptor
HMG-CoA Reductase
CFTR
p53
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DHFR
LPL Receptor
GNRH Receptor
MAO
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MAPK
Monoamine Oxidase
S1P Receptor
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Guanylate cyclase
Vasopressin Receptor
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PERK
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IDO
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Isocitrate Dehydrogenase (IDH)
Angiotensin-converting Enzyme (ACE)
Indoleamine 2,3-Dioxygenase (IDO)
IκB/IKK
PLK
Neurokinin receptor
DNA Methyltransferase
NOD-like Receptor (NLR)
Kinesin
Chloride channel
Reductase
NADPH
Serine Protease
FXR
CSF-1R
Antifection
Sirtuin
Casein Kinase
Ligand for E3 Ligase
Phospholipase
IRAK
Mdm2
PROTACs
Leukotriene Receptor
RIP kinase
Smo
PAK
CCR
OX Receptor
CaMK
DNA
GPCR19
Melanocortin Receptor
Photosensitizer
Pim
Monoamine Transporter
Aromatase
Hydroxylase
Thrombin
PD-1/PD-L1
IKZF
IFNAR
Tie-2
CaSR
Cholecystokinin Receptor
Serine/threonin kinase
PYK2
UGT
Glucagon Receptor
DPP-4
Ephrin Receptor
RSV
ribosome
Aryl Hydrocarbon Receptor
Na-K-Cl cotransporter
Glucosidase
Fatty Acid Synthase
Bradykinin Receptor
Somatostatin
glycosidase
Telomerase
Wee1
OXPHOS
PGE Synthase
STING
Aminopeptidase
CRFR
PDK
Oxytocin Receptor
GHSR
AhR
NOS
Monocarboxylate transporter
CRM1
Amino Acids and Derivatives
YAP
LTR
TOPK
Melatonin Receptor
c-Myc
NAMPT
Glutaminase
Immunology/Inflammation related
IRE1
Annexin A
DNA gyrase
Neuropeptide Y Receptor
Xanthine Oxidase
DUB
GST
FKBP
CGRP Receptor
Cuproptosis
MLK
MicroRNA
ROR
NEDD8
Arginase
DYRK
Necroptosis
MIF
Rho
Cell Cycle Arrest
Cysteine Protease
Liver X Receptor
RANKL/RANK
MT Receptor
Hexokinase
PROTAC Linker
KSP
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Beta-Secretase
OAT
Acyltransferase
MNK
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transporter
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FOXO
Adenosine Deaminase
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Gap Junction Protein
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Thyroid hormone receptor(THR)
Ligands for Target Protein for PROTAC
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HCN Channel
FAAH
PTEN
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ASK
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p97
Imidazoline Receptor
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gp120/CD4
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OCT
N-Acetylglucosaminyltransferase
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Hck
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cAMP
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KLF
Aquaporin
RXFP receptor
Platelet aggregation
NADPH-oxidase
BMI-1
Liposome
Ferroportin
PGC-1α
Drug-Linker Conjugates for ADC

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