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Bisindolylmaleimide III

Catalog No. T77628 CAS 137592-43-9

Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively interacts with PKCα or ribosomal S6 protein kinase 1 upon activation of these kinases.

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Bisindolylmaleimide III Chemical Structure

Bisindolylmaleimide III, CAS 137592-43-9

Pack Size	Availability	Price/USD
5 mg	In stock	$ 71.00
10 mg	In stock	$ 116.00
25 mg	In stock	$ 195.00
50 mg	In stock	$ 289.00
100 mg	In stock	$ 429.00
1 mL * 10 mM (in DMSO)	In stock	$ 78.00

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Purity: 98.6%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Molecular Weight	384.43
Formula	C23H20N4O2
CAS No.	137592-43-9

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 20 mg/mL (52.02 mM), Sonication is recommended.

References and Literature

1. Brehmer D, et al. Proteome-wide identification of cellular targets affected by bisindolylmaleimide-type protein kinase C inhibitors. Mol Cell Proteomics. 2004 May;3(5):490-500. 2. Saito Y, et al. Role of ecto-kinase in phorbol ester-enhanced growth hormone-binding protein release from human IM-9 cells. Mol Cell Endocrinol. 1999 Jun 25;152(1-2):65-72.

Related compound libraries

This product is contained In the following compound libraries：

Inhibitor Library TGF-beta/Smad Compound Library Bioactive Compounds Library Max Kinase Inhibitor Library Bioactive Compound Library

Related Products

Related compounds with same targets

PKCβ inhibitor 1 Chelerythrine Chelerythrine chloride Daphnoretin Verbascoside HA-100 [Ala107]-MBP (104-118) acetate PKC β pseudosubstrate acetate

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Bisindolylmaleimide III 137592-43-9 Chromatin/Epigenetic Cytoskeletal Signaling PKC BisindolylmaleimideIII inhibitor inhibit

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