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Epetraborole hydrochloride

Name: Epetraborole hydrochloride
Brand: TargetMol
SKU: T4045
Price: 419 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T4045Cas No. 1234563-16-6

Alias GSK2251052 hydrochloride

Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.

Epetraborole hydrochloride

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🥰Excellent

Purity: 99.59%

Catalog No. T4045Alias GSK2251052 hydrochlorideCas No. 1234563-16-6

Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$56	In Stock	In Stock
5 mg	$113	In Stock	In Stock
10 mg	$189	In Stock	In Stock
25 mg	$419	In Stock	In Stock
50 mg	Preferential	In Stock	In Stock
1 mL x 10 mM (in DMSO)	$126	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.59%

Color:White

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.
Synonyms	GSK2251052 hydrochloride

Chemical Properties

Molecular Weight	273.52
Formula	C₁₁H₁₇BClNO₄
Cas No.	1234563-16-6
Smiles	Cl.NC[C@H]1OB(O)c2c1cccc2OCCCO
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 28 mg/mL (102.37 mM), Sonication is recommended.

DMSO: 150 mg/mL (548.41 mM)

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	3.6560 mL	18.2802 mL	36.5604 mL	182.8020 mL
5 mM	0.7312 mL	3.6560 mL	7.3121 mL	36.5604 mL
10 mM	0.3656 mL	1.8280 mL	3.6560 mL	18.2802 mL
20 mM	0.1828 mL	0.9140 mL	1.8280 mL	9.1401 mL
50 mM	0.0731 mL	0.3656 mL	0.7312 mL	3.6560 mL
100 mM	0.0366 mL	0.1828 mL	0.3656 mL	1.8280 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc