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Epetraborole hydrochloride

Name: Epetraborole hydrochloride
Brand: TargetMol
SKU: T4045
Price: 48 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T4045Cas No. 1234563-16-6

Alias GSK2251052 hydrochloride

Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.

Epetraborole hydrochloride

🥰Excellent

Purity: 99.59%

Catalog No. T4045Alias GSK2251052 hydrochlorideCas No. 1234563-16-6

Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.

Pack Size	Price	Availability
1 mg	$48	In Stock
5 mg	$102	In Stock
10 mg	$171	In Stock
25 mg	$381	In Stock
50 mg	$567	In Stock
1 mL x 10 mM (in DMSO)	$101	In Stock

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Batch Information

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Purity:99.59%

Resource Download

COA HNMR HPLC

Product Introduction

Bioactivity

Description	Epetraborole hydrochloride (GSK2251052 hydrochloride) is a potent and selective leucyl-tRNA synthetase inhibitor.
Synonyms	GSK2251052 hydrochloride

Chemical Properties

Molecular Weight	273.52
Formula	C₁₁H₁₇BClNO₄
Cas No.	1234563-16-6
Smiles	Cl.NC[C@H]1OB(O)c2c1cccc2OCCCO
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

H2O: 28 mg/mL (102.37 mM), Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	3.6560 mL	18.2802 mL	36.5604 mL	182.8020 mL
5 mM	0.7312 mL	3.6560 mL	7.3121 mL	36.5604 mL
10 mM	0.3656 mL	1.8280 mL	3.6560 mL	18.2802 mL
20 mM	0.1828 mL	0.9140 mL	1.8280 mL	9.1401 mL
50 mM	0.0731 mL	0.3656 mL	0.7312 mL	3.6560 mL
100 mM	0.0366 mL	0.1828 mL	0.3656 mL	1.8280 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc