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Rapastinel

Name: Rapastinel
Brand: TargetMol
SKU: T3407
Price: 40 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T3407Cas No. 117928-94-6

Alias TPPT-amide, Thr-Pro-Pro-Thr-NH2, GLYX-13

Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.

Rapastinel

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Purity: 97.18%

Catalog No. T3407Alias TPPT-amide, Thr-Pro-Pro-Thr-NH2, GLYX-13Cas No. 117928-94-6

Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.

Pack Size	Price	USA Warehouse	Global Warehouse
1 mg	$40	In Stock	In Stock
5 mg	$82	In Stock	In Stock
10 mg	$117	In Stock	In Stock
25 mg	$243	In Stock	In Stock
50 mg	$359	-	In Stock
1 mL x 10 mM (in DMSO)	$82	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

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Purity:97.18%

Resource Download

COA HPLC MS

Product Introduction

Bioactivity

Description	Rapastinel (TPPT-amide) (GLYX-13) is an N-methyl-D-aspartate receptor (NMDAR) modulator.
Synonyms	TPPT-amide, Thr-Pro-Pro-Thr-NH2, GLYX-13

Chemical Properties

Molecular Weight	413.47
Formula	C₁₈H₃₁N₅O₆
Cas No.	117928-94-6
Smiles	C[C@@H](O)[C@H](N)C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N[C@@H]([C@@H](C)O)C(N)=O
Relative Density.	1.370 g/cm3 (Predicted)

Storage & Solubility Information

Storage

keep away from direct sunlight,store under nitrogen,store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 32 mg/mL (77.39 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4186 mL	12.0928 mL	24.1856 mL	120.9278 mL
5 mM	0.4837 mL	2.4186 mL	4.8371 mL	24.1856 mL
10 mM	0.2419 mL	1.2093 mL	2.4186 mL	12.0928 mL
20 mM	0.1209 mL	0.6046 mL	1.2093 mL	6.0464 mL
50 mM	0.0484 mL	0.2419 mL	0.4837 mL	2.4186 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc