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Acetyl-Calpastatin(184-210)(human)

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Catalog No. TP2056Cas No. 123714-50-1
Alias Acetyl-Calpastatin (184-210) (human)

Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.

Acetyl-Calpastatin(184-210)(human)
Other Forms of Acetyl-Calpastatin(184-210)(human):
Acetyl-Calpastatin (184-210)(human) acetateTP2056L
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Acetyl-Calpastatin(184-210)(human)

😃Good
Catalog No. TP2056Alias Acetyl-Calpastatin (184-210) (human)Cas No. 123714-50-1
Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$1,53035 days35 days
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction

Bioactivity
Description
Selective calpain inhibitor. Strongly inhibits calpain I (Ki = 0.2 nM) and II but does not inhibit papain, trypsin and cathepsin L (Ki = 6 μM). Increases secretion of amyoid β-protein (Aβ) 42, Aβ40 and Aβ42 ratio.
SynonymsAcetyl-Calpastatin (184-210) (human)
Chemical Properties
Molecular Weight3177.65
FormulaC142H230N36O44S
Cas No.123714-50-1
SmilesC(=O)([C@H]1N(C([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(CNC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CC2=CC=C(O)C=C2)NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC(=O)[C@H]3N(C([C@H](CC(O)=O)NC(C)=O)=O)CCC3)CCSC)=O)CO)=O)CO)=O)[C@@H](C)O)=O)=O)[C@H](CC)C)=O)CCC(O)=O)=O)CCC(O)=O)=O)CC(C)C)=O)=O)CCCCN)=O)CCCNC(=N)N)=O)CCC(O)=O)=O)[C@H](C)C)=O)[C@@H](C)O)=O)[C@H](CC)C)=O)CCC1)N4[C@H](C(N[C@H](C(N[C@@H](CC5=CC=C(O)C=C5)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N)=O)C)=O)CC(C)C)=O)CC(C)C)=O)CCC(O)=O)=O)CCCNC(=N)N)=O)=O)CCCCN)=O)CCC4
Relative Density.1.46 g/cm3 (Predicted)
SequenceAc-Asp-Pro-Met-Ser-Ser-Thr-Tyr-Ile-Glu-Glu-Leu-Gly-Lys-Arg-Glu-Val-Thr-Ile-Pro-Pro-Lys-Tyr-Arg-Glu-Leu-Leu-Ala-NH2
Sequence ShortAc-DPMSSTYIEELGKREVTIPPKYRELLA-NH2
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 5 mg/mL (1.57 mM), Sonication is recommended.
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM0.3147 mL1.5735 mL3.1470 mL15.7349 mL

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
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Keywords

AcetylCalpastatin(184210)(human)Acetyl-CalpastatinAcetyl Calpastatin(184 210)(human)
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