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PKA inhibitor fragment (6-22) amide Acetate

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Catalog No. T21674L
Alias PKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)

PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).

PKA inhibitor fragment (6-22) amide Acetate
Other Forms of PKA inhibitor fragment (6-22) amide Acetate:
PKA Inhibitor Fragment (6-22) amide TFAT75888
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PKA inhibitor fragment (6-22) amide Acetate

🥰Excellent
Purity: 99.30%
Catalog No. T21674LAlias PKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)
PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$87In StockIn Stock
2 mg$125In StockIn Stock
5 mg$178In StockIn Stock
10 mg$293In StockIn Stock
25 mg$491In StockIn Stock
50 mg$716In StockIn Stock
100 mg$987-In Stock
1 mL x 10 mM (in DMSO)$481In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
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Purity:99.30%
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COA MS HPLC

Product Introduction

Bioactivity
Description
PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).
Targets&IC50
PKA:2.8 nM(ki)
SynonymsPKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)
Chemical Properties
Molecular Weight1928.11
FormulaC82H134N28O26
SmilesCC(O)=O.CC[C@H](C)[C@@H](C(N)=O)NC([C@H](C)NC([C@H](CC(N)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC(CNC([C@H]([C@H](O)C)NC([C@H](CCCNC(N)=N)NC(CNC([C@H](CO)NC([C@H](C)NC([C@H]([C@@H](C)CC)NC([C@H](CC1=CC=CC=C1)NC([C@H](CC(O)=O)NC([C@H](C)NC([C@H](CC2=CC=C(O)C=C2)NC([C@H]([C@H](O)C)N)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O
Relative Density.no data available
SequenceH-Thr-Tyr-Ala-Asp-Phe-lle-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-lle-NH2
Sequence ShortVAKHFAFLRUNHLQ-PEBJKXEYSA-N
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 55 mg/mL (28.53 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM0.5186 mL2.5932 mL5.1864 mL25.9321 mL
5 mM0.1037 mL0.5186 mL1.0373 mL5.1864 mL
10 mM0.0519 mL0.2593 mL0.5186 mL2.5932 mL
20 mM0.0259 mL0.1297 mL0.2593 mL1.2966 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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2 Enter the in vivo formulation:
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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PKA inhibitor fragment (622) amide AcetatePKA inhibitor fragment (6 22) amide AcetatePKA inhibitor fragment amide AcetatePKA
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