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PKA inhibitor fragment (6-22) amide Acetate

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Catalog No. T21674L
Alias PKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)

PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).

PKA inhibitor fragment (6-22) amide Acetate
Other Forms of PKA inhibitor fragment (6-22) amide Acetate:
PKA Inhibitor Fragment (6-22) amide TFAT75888
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PKA inhibitor fragment (6-22) amide Acetate

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Purity: 99.30%
Catalog No. T21674LAlias PKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)
PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$87In StockIn Stock
2 mg$125In StockIn Stock
5 mg$178In StockIn Stock
10 mg$293In StockIn Stock
25 mg$491In StockIn Stock
50 mg$716In StockIn Stock
100 mg$987-In Stock
1 mL x 10 mM (in DMSO)$481In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
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Batch Information

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Purity:99.30%
Appearance:Solid
Color:White
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COA MS HPLC

Product Introduction

Bioactivity
Description
PKA inhibitor fragment (6-22) amide Acetate is a synthetic peptide which selectively inhibits PKA activity by binding to its substrate site (IC50 < 2 nM).
Targets&IC50
PKA:2.8 nM(ki)
SynonymsPKA inhibitor fragment (6-22) amide Acetate(121932-06-7 Free base)
Chemical Properties
Molecular Weight1928.11
FormulaC82H134N28O26
SmilesCC(O)=O.CC[C@H](C)[C@@H](C(N)=O)NC([C@H](C)NC([C@H](CC(N)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC(CNC([C@H]([C@H](O)C)NC([C@H](CCCNC(N)=N)NC(CNC([C@H](CO)NC([C@H](C)NC([C@H]([C@@H](C)CC)NC([C@H](CC1=CC=CC=C1)NC([C@H](CC(O)=O)NC([C@H](C)NC([C@H](CC2=CC=C(O)C=C2)NC([C@H]([C@H](O)C)N)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O
Relative Density.no data available
SequenceH-Thr-Tyr-Ala-Asp-Phe-lle-Ala-Ser-Gly-Arg-Thr-Gly-Arg-Arg-Asn-Ala-lle-NH2
Sequence ShortVAKHFAFLRUNHLQ-PEBJKXEYSA-N
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 55 mg/mL (28.53 mM), Sonication is recommended.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM0.5186 mL2.5932 mL5.1864 mL25.9321 mL
5 mM0.1037 mL0.5186 mL1.0373 mL5.1864 mL
10 mM0.0519 mL0.2593 mL0.5186 mL2.5932 mL
20 mM0.0259 mL0.1297 mL0.2593 mL1.2966 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
TargetMol | Animal experiments For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent 10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.
Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSOTargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSOTargetMol | reagent stock solution to 400 μL PEG300TargetMol | reagent and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH2OTargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PKA inhibitor fragment (622) amide AcetatePKA inhibitor fragment (6 22) amide AcetatePKA inhibitor fragment amide AcetatePKA
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