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Methuosis inducer 1

🥰Excellent
Catalog No. T7262Cas No. 2240205-30-3

Methuosis inducer 1 is a potent methuosis inducer with anticancer activity.

Methuosis inducer 1

Methuosis inducer 1

🥰Excellent
Purity: 99.34%
Catalog No. T7262Cas No. 2240205-30-3
Methuosis inducer 1 is a potent methuosis inducer with anticancer activity.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$81In StockIn Stock
5 mg$197In StockIn Stock
10 mg$297In StockIn Stock
25 mg$536In StockIn Stock
50 mg$787In StockIn Stock
100 mg$1,160In StockIn Stock
1 mL x 10 mM (in DMSO)$209In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.34%
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COA HNMR LCMS

Product Introduction

Bioactivity
Description
Methuosis inducer 1 is a potent methuosis inducer with anticancer activity.
In vivo
Methuosis inducer 1 exhibited substantial pharmacological efficacy in the suppression of tumor growth in a xenograft mouse model of MDA-MB-231 cells without apparent side effects, which makes this compound the first example of a methuosis inducer with potent in vivo efficacy.?These results demonstrate that methuosis inducers might serve as novel therapeutics for the treatment of cancer.
Chemical Properties
Molecular Weight487.48
FormulaC27H20F3N5O
Cas No.2240205-30-3
SmilesCc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1Nc1cc(nc2[nH]ccc12)-c1cccnc1
Relative Density.1.399 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 120 mg/mL (246.16 mM), Sonication is recommended.
In Vivo Formulation
10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (4.1 mM), Sonication is recommended.
Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.0514 mL10.2568 mL20.5137 mL102.5683 mL
5 mM0.4103 mL2.0514 mL4.1027 mL20.5137 mL
10 mM0.2051 mL1.0257 mL2.0514 mL10.2568 mL
20 mM0.1026 mL0.5128 mL1.0257 mL5.1284 mL
50 mM0.0410 mL0.2051 mL0.4103 mL2.0514 mL
100 mM0.0205 mL0.1026 mL0.2051 mL1.0257 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
mg/kg
g
μL
2 Enter the in vivo formulation:
% DMSO
%
% Tween 80
% Saline/PBS/ddH2O

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

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