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Azasetron hydrochloride

Name: Azasetron hydrochloride
Brand: TargetMol
SKU: T1528
Price: 34 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T1528Cas No. 123040-16-4

Alias Y-25130 hydrochloride, Y-25130 HCl, Azasetron HCl

Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.

Azasetron hydrochloride

🥰Excellent

Purity: 99.50%

Catalog No. T1528Alias Y-25130 hydrochloride, Y-25130 HCl, Azasetron HClCas No. 123040-16-4

Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.

Pack Size	Price	USA Warehouse	Global Warehouse
5 mg	$34	In Stock	In Stock
10 mg	$53	In Stock	In Stock
25 mg	$96	In Stock	In Stock
50 mg	$174	In Stock	In Stock
100 mg	$296	In Stock	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

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Batch Information

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Purity:99.50%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.
Targets&IC50	5-HT3:0.33 nM
Synonyms	Y-25130 hydrochloride, Y-25130 HCl, Azasetron HCl

Chemical Properties

Molecular Weight	386.27
Formula	C₁₇H₂₀ClN₃O₃·HCl
Cas No.	123040-16-4
Smiles	Cl.CN1C(=O)COc2c1cc(Cl)cc2C(=O)NC1CN2CCC1CC2
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: Insoluble

H2O: 10 mM, Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	2.5889 mL	12.9443 mL	25.8886 mL	129.4431 mL
5 mM	0.5178 mL	2.5889 mL	5.1777 mL	25.8886 mL
10 mM	0.2589 mL	1.2944 mL	2.5889 mL	12.9443 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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