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mAChR-IN-1 hydrochloride

Name: mAChR-IN-1 hydrochloride
Brand: TargetMol
SKU: T5655
Price: 34 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T5655Cas No. 119391-73-0

mAChR-IN-1 hydrochloride is a potent antagonist of muscarinic cholinergic receptors (mAChR) with an IC50 of 17 nM.

mAChR-IN-1 hydrochloride

🥰Excellent

Purity: 99.87%

Catalog No. T5655Cas No. 119391-73-0

mAChR-IN-1 hydrochloride is a potent antagonist of muscarinic cholinergic receptors (mAChR) with an IC50 of 17 nM.

Pack Size	Price	Availability
1 mg	$34	In Stock
5 mg	$83	In Stock
10 mg	$135	In Stock
25 mg	$239	In Stock
50 mg	$330	In Stock
100 mg	$413	In Stock
200 mg	$548	In Stock
1 mL x 10 mM (in DMSO)	$96	In Stock

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Purity:99.87%

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COA HPLC HNMR LCMS

Product Introduction

Bioactivity

Description	mAChR-IN-1 hydrochloride is a potent antagonist of muscarinic cholinergic receptors (mAChR) with an IC50 of 17 nM.
Targets&IC50	mAChR:17nM

Chemical Properties

Molecular Weight	524.82
Formula	C₂₃H₂₆ClIN₂O₂
Cas No.	119391-73-0
Smiles	Cl.Ic1ccc(CN2CCC(CC2)C2(CCC(=O)NC2=O)c2ccccc2)cc1
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 65 mg/mL (123.85 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	1.9054 mL	9.5271 mL	19.0542 mL	95.2708 mL
5 mM	0.3811 mL	1.9054 mL	3.8108 mL	19.0542 mL
10 mM	0.1905 mL	0.9527 mL	1.9054 mL	9.5271 mL
20 mM	0.0953 mL	0.4764 mL	0.9527 mL	4.7635 mL
50 mM	0.0381 mL	0.1905 mL	0.3811 mL	1.9054 mL
100 mM	0.0191 mL	0.0953 mL	0.1905 mL	0.9527 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc