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Methiothepin mesylate

Name: Methiothepin mesylate
Brand: TargetMol
SKU: T2190
Price: 31 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T2190Cas No. 74611-28-2

Alias Ro 8-6837 mesylate, Metitepine mesylate

Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.

Methiothepin mesylate

🥰Excellent

Purity: 99.92%

Catalog No. T2190Alias Ro 8-6837 mesylate, Metitepine mesylateCas No. 74611-28-2

Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.

Pack Size	Price	Availability	Quantity
5 mg	$31	In Stock
10 mg	$50	In Stock

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Purity:99.92%

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Product Introduction

Bioactivity

Description	Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
Synonyms	Ro 8-6837 mesylate, Metitepine mesylate

Chemical Properties

Molecular Weight	452.65
Formula	C₂₁H₂₈N₂O₃S₃
Cas No.	74611-28-2
Smiles	CS(O)(=O)=O.CSc1ccc2Sc3ccccc3CC(N3CCN(C)CC3)c2c1
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 45 mg/mL (99.41 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.2092 mL	11.0461 mL	22.0921 mL	110.4606 mL
5 mM	0.4418 mL	2.2092 mL	4.4184 mL	22.0921 mL
10 mM	0.2209 mL	1.1046 mL	2.2092 mL	11.0461 mL
20 mM	0.1105 mL	0.5523 mL	1.1046 mL	5.5230 mL
50 mM	0.0442 mL	0.2209 mL	0.4418 mL	2.2092 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc