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Venuloside A

Name: Venuloside A
Brand: TargetMol
SKU: TN7256
Price: 195 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. TN7256Cas No. 1609278-97-8

Alias ESK246

Venuloside A (ESK246), a monoprostane glycoside from Pittosporum venulosum, is a LAT3 inhibitor and a leucine uptake inhibitor that inhibits the transporter of leucine through LAT3, and may be used in the study of prostate cancer.

Venuloside A

🥰Excellent

Purity: 99.7%

Catalog No. TN7256Alias ESK246Cas No. 1609278-97-8

Pack Size	Price	Availability
1 mg	$195	In Stock
5 mg	$483	In Stock
10 mg	$692	In Stock
25 mg	$1,080	In Stock
50 mg	$1,490	In Stock

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.7%

ee:100%

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COA CSFC HNMR LCMS ORP

Product Introduction

Bioactivity

Description	Venuloside A (ESK246), a monoprostane glycoside from Pittosporum venulosum, is a LAT3 inhibitor and a leucine uptake inhibitor that inhibits the transporter of leucine through LAT3, and may be used in the study of prostate cancer.
Targets&IC50	LNCaP cells:8.12 μM
Synonyms	ESK246

Chemical Properties

Molecular Weight	424.53
Formula	C₂₃H₃₆O₇
Cas No.	1609278-97-8
Smiles	O(C(C)(C)[C@@H]1CCC(C)=CC1)[C@H]2[C@H](OC(C)=O)[C@@H](OC(C=C(C)C)=O)[C@@H](O)[C@@H](C)O2
Relative Density.	no data available
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 245 mg/mL (577.11 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.3555 mL	11.7777 mL	23.5555 mL	117.7773 mL
5 mM	0.4711 mL	2.3555 mL	4.7111 mL	23.5555 mL
10 mM	0.2356 mL	1.1778 mL	2.3555 mL	11.7777 mL
20 mM	0.1178 mL	0.5889 mL	1.1778 mL	5.8889 mL
50 mM	0.0471 mL	0.2356 mL	0.4711 mL	2.3555 mL
100 mM	0.0236 mL	0.1178 mL	0.2356 mL	1.1778 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc