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Pellitorine
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Catalog No. T21165Cas No. 18836-52-7
Alias Pellitorin, AI3-19560
Pellitorine (Pellitorin) is an extract of Tetradium daniellii, and acts as a TRPV1 antagonist.
Pellitorine
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Purity: 97.54%
Catalog No. T21165Alias Pellitorin, AI3-19560Cas No. 18836-52-7
Pellitorine (Pellitorin) is an extract of Tetradium daniellii, and acts as a TRPV1 antagonist.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $64 | In Stock | In Stock | |
| 5 mg | $189 | In Stock | In Stock | |
| 10 mg | $313 | In Stock | In Stock | |
| 25 mg | $528 | In Stock | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Batch Information
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Purity:97.54%
Appearance:Solid
Color:White
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Product Introduction
Pellitorine AI Summary
Pellitorine exhibits a range of biological activities across different assays. It shows a dose-dependent inhibition of D-galactosamine/TNF-alpha-induced cell death in ddY mouse hepatocytes, with 19.0%, 25.0%, and 42.0% inhibition at 3 µM, 10 µM, and 30 µM concentrations, respectively, determined by the MTT assay. Additionally, it exhibits strong bioactivity in inhibiting the sICAM1/LFA1 interaction-mediated adhesion in human THP1 cells, with an IC50 value of 13.5 µg/mL and up to 80.6% inhibition at 25 µg/mL. In mouse 3T3L1 cells, it enhances triglyceride accumulation indicative of antidiabetic activity, with the highest activity of 18.2% observed at 3 µM. The compound shows hepatoprotective effects in various assays, including inhibition of D-galactosamine-induced cytotoxicity (IC50 = 9300 nM) and TNF-alpha-induced cytotoxicity in mouse L929 cells. It also exhibits antimicrobial activity against Mycobacterium tuberculosis H37Ra with a MIC of 50 µg/mL and antitrypanosomal activity against Trypanosoma cruzi Y with an IC50 of 57100 nM. Furthermore, it has significant insecticidal and larvicidal activities, demonstrated by an LD90 of 184.56 µg and an LD50 of 91.19 µg against Diatraea saccharalis and an LC50 of 0.92 ppm against Aedes aegypti. Lastly, it displays antineuroinflammatory activity in mouse BV2 cells, with an IC50 for inhibiting LPS-induced NO production of 45000 nM..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Pellitorine (Pellitorin) is an extract of Tetradium daniellii, and acts as a TRPV1 antagonist. |
| Synonyms | Pellitorin, AI3-19560 |
| Molecular Weight | 223.35 |
| Formula | C14H25NO |
| Cas No. | 18836-52-7 |
| Smiles | CCCCC\C=C\C=C\C(=O)NCC(C)C |
| Relative Density. | 0.882 g/cm3 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | DMSO: Soluble |
Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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