Select your Country or Region

  • TargetMol | Compound LibraryArgentinaArgentina
  • TargetMol | Compound LibraryAustraliaAustralia
  • TargetMol | Compound LibraryAustriaAustria
  • TargetMol | Compound LibraryBelgiumBelgium
  • TargetMol | Compound LibraryBrazilBrazil
  • TargetMol | Compound LibraryBulgariaBulgaria
  • TargetMol | Compound LibraryCroatiaCroatia
  • TargetMol | Compound LibraryCyprusCyprus
  • TargetMol | Compound LibraryCzechCzech
  • TargetMol | Compound LibraryDenmarkDenmark
  • TargetMol | Compound LibraryEgyptEgypt
  • TargetMol | Compound LibraryEstoniaEstonia
  • TargetMol | Compound LibraryFinlandFinland
  • TargetMol | Compound LibraryFranceFrance
  • TargetMol | Compound LibraryGermanyGermany
  • TargetMol | Compound LibraryGreeceGreece
  • TargetMol | Compound LibraryHong KongHong Kong
  • TargetMol | Compound LibraryHungaryHungary
  • TargetMol | Compound LibraryIcelandIceland
  • TargetMol | Compound LibraryIndiaIndia
  • TargetMol | Compound LibraryIrelandIreland
  • TargetMol | Compound LibraryIsraelIsrael
  • TargetMol | Compound LibraryItalyItaly
  • TargetMol | Compound LibraryJapanJapan
  • TargetMol | Compound LibraryKoreaKorea
  • TargetMol | Compound LibraryLatviaLatvia
  • TargetMol | Compound LibraryLebanonLebanon
  • TargetMol | Compound LibraryMalaysiaMalaysia
  • TargetMol | Compound LibraryMaltaMalta
  • TargetMol | Compound LibraryMoroccoMorocco
  • TargetMol | Compound LibraryNetherlandsNetherlands
  • TargetMol | Compound LibraryNew ZealandNew Zealand
  • TargetMol | Compound LibraryNorwayNorway
  • TargetMol | Compound LibraryPolandPoland
  • TargetMol | Compound LibraryPortugalPortugal
  • TargetMol | Compound LibraryRomaniaRomania
  • TargetMol | Compound LibrarySingaporeSingapore
  • TargetMol | Compound LibrarySlovakiaSlovakia
  • TargetMol | Compound LibrarySloveniaSlovenia
  • TargetMol | Compound LibrarySpainSpain
  • TargetMol | Compound LibrarySwedenSweden
  • TargetMol | Compound LibrarySwitzerlandSwitzerland
  • TargetMol | Compound LibraryTaiwan,ChinaTaiwan,China
  • TargetMol | Compound LibraryThailandThailand
  • TargetMol | Compound LibraryTurkeyTurkey
  • TargetMol | Compound LibraryUnited KingdomUnited Kingdom
  • TargetMol | Compound LibraryUnited StatesUnited States
  • TargetMol | Compound LibraryOther CountriesOther Countries
Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
Filter
TargetMol | Tags GPCR/G Protein
TargetMol | Tags Neuroscience

Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

  • Ritanserin
    T1675987051-43-2
    Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
    • $34
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
    TargetMol | Citations Cited
  • Syrosingopine
    TN225284-36-6
    Syrosingopine has selective depleting effect on brain amines is potentiated by combined treatment with disulfiram or fusaric acid, a dopamine beta-hydroxylase inhibitor.
    • $61
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
    TargetMol | Citations Cited
  • MPTP hydrochloride
    T408123007-85-4
    MPTP hydrochloride is a precursor of MPP+, a dopamine neurotoxin with blood-brain barrier permeability. MPTP hydrochloride is toxic to dopaminergic neurons, which can lead to Parkinson's disease, and is widely used in the construction of animal models of Parkinson's disease.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
  • CLOZAPINE N-OXIDE
    T449434233-69-7
    Clozapine N-oxide is the major metabolite of Clozapine and is blood-brain barrier permeable. Clozapine N-oxide is an agonist of DREADDs and activates the DREADD receptors hM3Dq and hM4Di. Clozapine N-oxide is also a dopamine antagonist and selective muscarinic M4 receptor agonist.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Hot
    TargetMol | Citations Cited
  • BL-1020 Mesylate
    T26834916898-61-8In house
    BL-1020 Mesylate (CYP-1020 Mesylate) is an orally available GABA A receptor agonist and D2 antagonist that decreases dopamine activity and enhances GABAA activity.BL-1020 Mesylate has been used in the study of schizophrenia, Alzheimer's disease, and bi-directional cognitive impairment.
    • $293 TargetMol
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • Ziprasidone hydrochloride monohydrate
    T0031138982-67-9
    Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
    • $50
    In Stock
    Size
    QTY
  • Dopamine hydrochloride
    T164462-31-7
    Dopamine hydrochloride (ASL279) is a naturally occurring catecholamine formed by decarboxylation of dihydroxyphenylalanine and a precursor of norepinephrine and epinephrine. Dopamine hydrochloride binds to alpha-1- and beta-1- adrenergic receptors.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
  • SKF 38393 hydrochloride
    T698862717-42-4
    SKF 38393 hydrochloride (SKF38393 HCl) is a selective dopamine D1 D5 receptor agonist.
    • $50
    In Stock
    Size
    QTY
  • L-(R,S)-Tetrahydropalmatine
    T271410097-84-4
    L-(R,S)-Tetrahydropalmatine (Rotundine) is extracted from Corydalis yanhusuo W. T. Wang.
    • $50
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • N-0500 HCl
    T60107100935-99-7In house
    N-0500 HCl ((-)-Propyl-9-hydroxynaphthoxazine Hydrochloride) is a very potent centrally acting DA receptor agonist. N-0500 HCl is a potent displacer of the specific [3H]DP_x0002_5,6-ADTN binding with IC50 of 3nM.
    • $30
    In Stock
    Size
    QTY
  • Mianserin hydrochloride
    T078321535-47-7
    Mianserin hydrochloride (Org GB 94) is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin receptors. It may cause drowsiness and hematological problems.
    • $32
    In Stock
    Size
    QTY
  • A 77636 hydrochloride
    T21782145307-34-2In house
    A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM). A 77636 hydrochloride shows antiparkinsonian activity. A 77636 hydrochloride is functionally inactive at dopamine D2 receptor.
    • $97
    In Stock
    Size
    QTY
  • LE 300
    T22921274694-98-3In house
    dopamine D1 receptor antagonist
    • $108
    In Stock
    Size
    QTY
  • Perphenazine
    T109058-39-9
    Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
    • $29
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
  • Citicoline
    T0136987-78-0
    Citicoline (CDP-Choline) is an intermediate in the synthesis of phosphatidylcholine, a component of cell membranes. Citicoline exerts neuroprotective effects.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
  • Pridopidine
    T7352346688-38-8In house
    Pridopidine (FR310826), a dopamine (DA) stabilizer, acts as a low affinity dopamine D2 receptor (D2R) antagonist, improves motor performance and shows neuroprotective effects in Huntington disease R6 2 mouse model.
    • $34
    In Stock
    Size
    QTY
  • PF-00217830
    T24613846032-02-8In house
    PF-00217830 is a serotonin 1A receptor agonist, dopamine D2 receptor agonist, and serotonin 2A receptor antagonist.PF-00217830 may be used in the study of schizophrenia.
    • $143
    In Stock
    Size
    QTY
  • carfenazine
    T98272622-30-2
    carfenazine targets the Dopamine receptor and is used for schizophrenia research.
    • $187
    In Stock
    Size
    QTY
  • 3-CPMT
    T2250814008-79-8
    3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
    • $37
    In Stock
    Size
    QTY
  • Rotigotine
    T923792206-54-7In house
    Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.
    • $38
    In Stock
    Size
    QTY
    TargetMol | Citations Cited
  • Pimethixene
    T12489314-03-4
    Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
    • $35
    In Stock
    Size
    QTY
  • Dopamine D2 receptor agonist-2
    T600751610591-93-9
    Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
    • $53
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • PNU-177864 hydrochloride
    T125101783978-03-9In house
    PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor. PNU-177864 hydrochloride is structurally consistent with a cationic amphiphilic drug (CAD). PNU-177864 hydrochloride induces phospholipidosis in vivo. PNU-177864 hydrochloride exhibits antischizophrenic activity.
    • $30
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • Neuromedin N acetate(92169-45-4 free base)
    TP1085L
    Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.Neuromedin N is a potent modulator of dopamine D2 receptor agonist binding in rat neostriatal membranes.
    • $47
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • L-745870 trihydrochloride
    T22904866021-03-6
    L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
    • $68
    In Stock
    Size
    QTY
  • SLV-310
    T28809264869-71-8In house
    SLV-310 is a potent dopamine D2 receptor antagonist and 5-HT reuptake receptor inhibitor used in the study of neurological disorders such as bipolar disorder and schizophrenia.
    • $293 TargetMol
    In Stock
    Size
    QTY
  • Lensiprazine
    T32633327026-93-7In house
    Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and schizophrenia.
    • $191
    In Stock
    Size
    QTY
  • BP 897
    T9100192384-87-5
    BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2 receptor antagonist, with Kis of 0.92 nM and 61 nM for D3 and D2 receptors, and shows low affinities at D1 and D4 receptors (Kis, 3 and 0.3 μM, respectively).
    • $121
    In Stock
    Size
    QTY
  • Aplindore Fumarate
    T30098189681-71-8In house
    Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-HT2), and α1-adrenergic receptors.Aplindore Fumarate is used in the study of Parkinson's disease and schizophrenia. Fumarate can be used to study Parkinson's and schizophrenia.
    • $293
    In Stock
    Size
    QTY
  • Tedatioxetine
    T34795508233-95-2In house
    Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Tedatioxetine acts as a CYP2D6 substrate.
    • $293
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • NGD 94-1
    T23066178928-68-2In house
    NGD 94-1 is a selective D4 receptor antagonist with an affinity of 3 nM for the D4 receptor and greater than 2 pM for the D1, D2, D3, and D5 receptors.NGD 94-1 can be used in the study of cognitive disorders and other psychiatric disorders.
    • $85
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • Tolnapersine TFA
    T68023L
    Tolnapersine TFA is a mixed dopamine agonist and alpha adrenergic receptor antagonist.
    • $195
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • 5-HT6/7 antagonist 1
    T61807131999-28-5In house
    5-HT6 7 antagonist 1 is a dual 5-HT6 7 2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.
    • $700 TargetMol
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • Abaperidone
    T14083183849-43-6In house
    Abaperidone is a potent 5-HT2A receptor and dopamine D2 receptor antagonist with an IC50 of 6.2 for 5-HT2A receptors and 17 nM for dopamine D2 receptors.Abaperidone is a potentially atypical anti-psychotropic compound that reduces basal hsp70 mRNA expression in rat striatum and prefrontal cortex. expression in the striatum and prefrontal cortex of rats.
    • $350
    In Stock
    Size
    QTY
  • WAY-260022
    T23711850692-43-2
    WAY-260022 is an orally available and selective norepinephrine transporter protein inhibitor that displays inhibitory effects on serotonin and dopamine transporter proteins.
    • $293 TargetMol
    In Stock
    Size
    QTY
  • PF-184298
    T28380813447-40-4In house
    PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.
    • $293 TargetMol
    In Stock
    Size
    QTY
  • PNU-96391
    T28435146798-66-5In house
    PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.
    • $195
    In Stock
    Size
    QTY
  • Ordopidine
    T33816871351-60-9In house
    Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity. Ordopidine acts as a dopamine D2 receptor antagonist in vitro and, despite its low affinity, its specific state-dependent behavioral effect characteristics are not generally shared by D2 receptor antagonists.
    • $142
    In Stock
    Size
    QTY
  • Trazpiroben
    T387541352993-39-5In house
    Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.
    • $293 TargetMol
    In Stock
    Size
    QTY
  • Tiaspirone hydrochloride
    T24885L87691-92-7In house
    Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity. Tiaspirone hydrochloride influences the electrophysiological activity of dopaminergic neurons in the substantia nigra zona compacta (A9 DA cells) and ventral tegmental area (A10 DA cells) in the brain of the rat.
    • $195
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • Molindone
    T214327416-34-4In house
    Molindone ((±)-Molindone) is a therapeutic antipsychotic used to treat schizophrenia by blocking the action of dopamine in the brain. molindone is often used in combination with serotonin in a dose-dependent manner to increase errors and decrease response rates.
    • $350
    In Stock
    Size
    QTY
  • DOPEXAMINE
    T865386197-47-9
    Dopexamine is a dopaminergic agonist
    • $133
    In Stock
    Size
    QTY
  • Romergoline 2HCl
    T71707L In house
    Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.
    • $195 TargetMol
    In Stock
    Size
    QTY
  • U 99194 maleate
    T23483234757-41-6
    U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.
    • $84
    In Stock
    Size
    QTY
  • JNJ-37822681
    T27677935776-74-2In house
    JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.
    • $148
    In Stock
    Size
    QTY
  • Liafensine
    T327371198790-53-2In house
    Liafensine(BMS-820836) is a novel and selective triple monoamine reuptake inhibitor with inhibitory effects on the reuptake of serotonin, norepinephrine, and dopamine for the study of major depressive disorder and central nervous system disorders.
    • $387
    In Stock
    Size
    QTY
  • SB-277011
    T12861215803-78-4In house
    SB-277011 (SB-277011A) is a specific antagonist of the dopamine D3 receptor with pKi values of 8.0, 6.0, 5.0, and <5.2 for D3 receptor, D2 receptor, 5-HT1D, and 5-HT1B respectively.
    • $39
    In Stock
    Size
    QTY
  • Mesoridazine Besylate
    T308632672-69-8
    Mesoridazine Besylate (Serentil) is a piperidine neuroleptic drug belonging to the class of drugs called phenothiazines, used in the treatment of schizophrenia. It is a metabolite of thioridazine.
    • $70
    In Stock
    Size
    QTY
  • Tiospirone
    T2488587691-91-6In house
    Tiospirone (BMY 13859-1 free base) is a 5-HT2 receptor antagonist and dopamine blocker that inhibits D2, 5-HT1a, 5-HT7, and sigma receptors.Tiospirone is used in the study of neurological disorders such as schizophrenia.
    • $132 TargetMol
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale
  • SK609 HCl
    T247971092797-77-7
    SK609 HCl (SK609 hydrochloride) is a dopamine D3 receptor (D3R) selective agonist that inhibits norepinephrine transporter proteins and can be used to study Parkinson's disease and cognitive disorders.
    • $80
    In Stock
    Size
    QTY
    TargetMol | Inhibitor Sale