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TargetMol | Compound Library

Bioactive Compound Library

Catalog No. L4000

It contains more than 14439 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation. Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4000

Bioactive Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A collection of 14439 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Apoptosis
Antibacterial
Autophagy
Endogenous Metabolite
Antibiotic
5-HT Receptor
AChR
Antifungal
Parasite
COX
Adrenergic Receptor
DNA/RNA Synthesis
NF-κB
Dopamine Receptor
CDK
HIV Protease
PI3K
Potassium Channel
Calcium Channel
EGFR
Reactive Oxygen Species
P450
Histamine Receptor
PDE
VEGFR
Epigenetic Reader Domain
Dehydrogenase
Sodium Channel
Influenza Virus
Antioxidant
GABA Receptor
GluR
PPAR
Histone Methyltransferase
TRP/TRPV Channel
Microtubule Associated
HDAC
JAK
TNF
mTOR
GPR
Wnt/beta-catenin
Akt
ERK
p38 MAPK
FLT
Prostaglandin Receptor
Topoisomerase
Phosphatase
Src
Estrogen/progestogen Receptor
Ferroptosis
PDGFR
AChE
Adenosine Receptor
SARS-CoV
STAT
iGluR
PKC
Estrogen Receptor/ERR
HCV Protease
PARP
AMPK
FGFR
GSK-3
IL Receptor
Nucleoside Antimetabolite/Analog
RAAS
Opioid Receptor
Raf
Caspase
NMDAR
Virus Protease
NO Synthase
MMP
c-Kit
BCL
c-Met/HGFR
Ras
MAO
Glucocorticoid Receptor
Androgen Receptor
Antiviral
Lipoxygenase
Proteasome
TLR
HSP
Phospholipase
Sirtuin
HBV
Bcr-Abl
ATPase
Cannabinoid Receptor
HSV
Mitochondrial Metabolism
Anti-infection
Beta Amyloid
ROS
TGF-beta/Smad
Aurora Kinase
ALK
Mitophagy
Tyrosinase
Drug Metabolite
MAPK
JNK
HIF/HIF Prolyl-Hydroxylase
BTK
DUB
E1/E2/E3 Enzyme
MEK
Casein Kinase
Antifection
Tyrosine Kinases
HER
NOS
Nrf2
Carbonic Anhydrase
CCR
Monoamine Oxidase
Interleukin
PKA
ROCK
Transferase
Reverse Transcriptase
IκB/IKK
Histone Demethylase
p53
HIF
P-gp
Serine/threonin kinase
IGF-1R
Retinoid Receptor
Gamma-secretase
P2X Receptor
Serotonin Transporter
DNA-PK
Integrin
CXCR
c-RET
S1P Receptor
TAM Receptor
Norepinephrine
Cysteine Protease
Immunology/Inflammation related
Serine Protease
LPL Receptor
Reductase
S6 Kinase
Hedgehog/Smoothened
CaMK
ribosome
Histone Acetyltransferase
FAK
Trk receptor
Chloride channel
RIP kinase
FAAH
Glucosidase
PROTACs
PLK
Sigma receptor
Progesterone Receptor
Proton pump
c-Fms
NADPH
transporter
Fatty Acid Synthase
CFTR
NOD
Glucokinase
Thrombin
Syk
ATM/ATR
DPP-4
Aryl Hydrocarbon Receptor
Chk
Acyltransferase
Mdm2
Protease-activated Receptor
Kinesin
Rho
Pim
Amino Acids and Derivatives
Ligand for E3 Ligase
DNA Methyltransferase
Endothelin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
PERK
HMG-CoA Reductase
ROR
PDK
Smo
Lipase
Thyroid hormone receptor(THR)
DNA Alkylator/Crosslinker
Glutathione Peroxidase
SGLT
DNA
FXR
P2Y Receptor
AhR
IRAK
Epoxide Hydrolase
Glucagon Receptor
Factor Xa
LTR
MRP
DYRK
Guanylate cyclase
Neurokinin receptor
Complement System
Xanthine Oxidase
Hydroxylase
LRRK2
cAMP
STING
PAK
LPA Receptor
OX Receptor
PD-1/PD-L1
Leukotriene Receptor
Neuropeptide Y Receptor
DHFR
NOD-like Receptor (NLR)
IRE1
c-Myc
YAP
IAP
Antifolate
DNA Alkylation
BACE
Myosin
Lipid
Aromatase
PGE Synthase
CSF-1R
Platelet aggregation
Liver X Receptor
PI4K
GTPase
DNA gyrase
Ephrin Receptor
RSV
ABC
Vasopressin Receptor
Aminopeptidase
cholecystokinin
ROS Kinase
Beta-Secretase
Telomerase
CETP
NADPH-oxidase
Monoamine Transporter
Stearoyl-CoA Desaturase (SCD)
Neurotensin Receptor
Bradykinin Receptor
Discoidin Domain Receptor (DDR)
GHSR
Free radical scavengers
Acetyl-CoA Carboxylase
GPCR19
Monocarboxylate transporter
Phosphorylase
PAI-1
Isocitrate Dehydrogenase (IDH)
Melanocortin Receptor
LDL
PKM
IDO
Imidazoline Receptor
Melatonin Receptor
NAMPT
IFNAR
MT Receptor
BCRP
GRK
ATP Citrate Lyase
CaSR
SGK
UGT
CAT
MLK
Porcupine
Dynamin
GST
Adenylyl cyclase
Wee1
Neprilysin
ASK
Ligands for Target Protein for PROTAC
Glutaminase
Arrestin
Tie-2
Arginase
GlyT
Na+/Ca2+ Exchanger
OCT
Annexin A
PTEN
MNK
SIK
PAD
p97
Somatostatin
RAR/RXR 
MyD88
MAGL
Molecular Glues
Carboxypeptidase
GPX
FLAP
Adenosine deaminase
Aquaporin
MELK
OAT
CRISPR/Cas9
APC
CRM1
Decarboxylase
Methionine Adenosyltransferase (MAT)
Bombesin Receptor
DprE1
TOPK
NPC1L1
VDAC
PAFR
PYK2
BMI-1
cGAS
MTH1
Amylase
Hippo pathway
AAK1 (AP2 associated kinase 1)
LIM Kinase
CRFR
TSH Receptor
cell cycle arrest
CGRP Receptor
ACK
GNRH Receptor
Oxytocin Receptor
Angiotensin-converting Enzyme (ACE)
Gap Junction Protein
KSP
NEDD8
Pyroptosis
Cell wall
MALT
DAPK
Survivin
advanced glycation end products
Adiponectin receptor
PROTAC Linker
Thrombopoietin Receptor
Melanin-concentrating Hormone Receptor (MCHR)
Galectin
CD73
Glutathione reductase
Necroptosis
AIM2
CD38
Haspin Kinase
Hexokinase
CPT
RANKL/RANK
OXPHOS
Na-K-Cl cotransporter
Transaminase
HCN Channel
Hck
GluCls
KLF
GSNOR
ATTECs
Protease
Integrase
Apelin receptor
Prolyl Endopeptidase (PREP)
EBI2/GPR183
NUDIX hydrolase
Fas/FasL
Taste receptor
VDA
lysosomal autophagy
gp120/CD4
PGC-1α
hCE
stilbene oxidase
aconitase
Fer/FerT kinase
Piezo Channel
FOXO1
N-Acetylglucosaminyltransferase
HuR
NMU2R
Motilin Receptor
Anion Exchanger
Procollagen C Proteinase
FABP
RXFP receptor
Neuropeptide W
Thioredoxin
Hydrogenase
PACAP
Stemness kinase
CYP19A1

Keywords