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TargetMol | Compound Library

Bioactive Compound Library

Catalog No. L4000

It contains more than 17100 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation. Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4000

Bioactive Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A collection of 17100 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Antibacterial
Endogenous Metabolite
Autophagy
Antibiotic
5-HT Receptor
AChR
Antifungal
Parasite
Adrenergic Receptor
COX
NF-κB
DNA/RNA Synthesis
Dopamine Receptor
CDK
HIV Protease
Calcium Channel
Potassium Channel
PI3K
EGFR
Antioxidant
Histamine Receptor
PDE
Reactive Oxygen Species
P450
Epigenetic Reader Domain
Dehydrogenase
Sodium Channel
VEGFR
GABA Receptor
GluR
Influenza Virus
Histone Methyltransferase
PPAR
Microtubule Associated
TRP/TRPV Channel
HDAC
TNF
GPR
mTOR
Phosphatase
Wnt/beta-catenin
JAK
AChE
p38 MAPK
Topoisomerase
Akt
Estrogen/progestogen Receptor
ERK
Prostaglandin Receptor
SARS-CoV
Src
Adenosine Receptor
Opioid Receptor
Antiviral
Ferroptosis
FLT
PKC
HCV Protease
PARP
RAAS
IL Receptor
STAT
NMDAR
Estrogen Receptor/ERR
PDGFR
iGluR
Caspase
AMPK
Nucleoside Antimetabolite/Analog
NO Synthase
GSK-3
Virus Protease
FGFR
Raf
MMP
BCL
Lipoxygenase
Ras
MAO
c-Kit
Glucocorticoid Receptor
Androgen Receptor
ATPase
Beta Amyloid
c-Met/HGFR
Bcr-Abl
Phospholipase
HSP
Cannabinoid Receptor
HBV
Proteasome
ROS
TLR
TGF-beta/Smad
Sirtuin
Mitochondrial Metabolism
ALK
Tyrosinase
HSV
Anti-infection
ADC Cytotoxin
JNK
Antifection
NOS
Aurora Kinase
DUB
MAPK
Mitophagy
BTK
Nrf2
HER
Integrin
Drug Metabolite
Histone Demethylase
PKA
E1/E2/E3 Enzyme
CCR
HIF/HIF Prolyl-Hydroxylase
ROCK
P-gp
Carbonic Anhydrase
Tyrosine Kinases
MEK
Transferase
Monoamine Oxidase
Casein Kinase
p53
Interleukin
IκB/IKK
Reverse Transcriptase
HIF
Immunology/Inflammation related
Gamma-secretase
Retinoid Receptor
Neurokinin receptor
Serotonin Transporter
CXCR
Serine/threonin kinase
Cysteine Protease
P2X Receptor
IGF-1R
Norepinephrine
Reductase
S1P Receptor
Serine Protease
Glucosidase
DNA-PK
CaMK
c-RET
Hedgehog/Smoothened
TAM Receptor
PROTACs
Trk receptor
Histone Acetyltransferase
Ligand for E3 Ligase
FAK
LPL Receptor
RIP kinase
Proton pump
FAAH
Sigma receptor
ribosome
PLK
S6 Kinase
Chloride channel
Glucokinase
Fatty Acid Synthase
Acyltransferase
NOD
Progesterone Receptor
transporter
ATM/ATR
NADPH
c-Fms
Syk
Amino Acids and Derivatives
Neuropeptide Y Receptor
Thrombin
DPP-4
Endothelin Receptor
HMG-CoA Reductase
CFTR
PERK
Pim
Rho
Chk
DNA Methyltransferase
Protease-activated Receptor
Thyroid hormone receptor(THR)
Mdm2
Aryl Hydrocarbon Receptor
Glucagon Receptor
cAMP
Kinesin
DNA Alkylator/Crosslinker
Smo
Complement System
DHFR
ROR
BACE
Lipase
Factor Xa
FXR
DNA
Indoleamine 2,3-Dioxygenase (IDO)
PDK
IRAK
cholecystokinin
P2Y Receptor
LTR
DYRK
Glutathione Peroxidase
Leukotriene Receptor
Guanylate cyclase
SGLT
STING
PD-1/PD-L1
Xanthine Oxidase
LRRK2
LPA Receptor
Platelet aggregation
AhR
MRP
Bradykinin Receptor
Epoxide Hydrolase
Melanocortin Receptor
Hydroxylase
GNRH Receptor
DNA Alkylation
OX Receptor
YAP
c-Myc
PAK
Vasopressin Receptor
Aromatase
GTPase
Liver X Receptor
PI4K
NOD-like Receptor (NLR)
IAP
Myosin
Ephrin Receptor
RSV
ROS Kinase
Antifolate
IRE1
Telomerase
Lipid
PGE Synthase
GHSR
ABC
Neurotensin Receptor
CSF-1R
LDL
DNA gyrase
Beta-Secretase
Aminopeptidase
Monoamine Transporter
Somatostatin
GPCR19
NADPH-oxidase
Monocarboxylate transporter
Arrestin
CETP
CaSR
ADC Linker
PAI-1
Acetyl-CoA Carboxylase
NAMPT
Glutaminase
IDO
GRK
Phosphorylase
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Free radical scavengers
Discoidin Domain Receptor (DDR)
Imidazoline Receptor
PKM
Ligands for Target Protein for PROTAC
Melatonin Receptor
UGT
Molecular Glues
Bombesin Receptor
BCRP
GST
GPX
MLK
Adenylyl cyclase
CAT
Dynamin
LIM Kinase
PAFR
MT Receptor
ATP Citrate Lyase
OAT
MNK
Neprilysin
SGK
Gap Junction Protein
Arginase
IFNAR
Tie-2
SIK
GlyT
Angiotensin-converting Enzyme (ACE)
PTEN
PAD
Wee1
Porcupine
ASK
Carboxypeptidase
Apelin receptor
Na+/Ca2+ Exchanger
OCT
Annexin A
AAK1 (AP2 associated kinase 1)
APC
MAGL
CRFR
p97
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
MyD88
RAR/RXR 
Cell wall
PYK2
FLAP
PROTAC Linker
Survivin
Decarboxylase
cGAS
TSH Receptor
MELK
Methionine Adenosyltransferase (MAT)
Drug-Linker Conjugates for ADC
CRISPR/Cas9
Oxytocin Receptor
Aquaporin
Adenosine deaminase
CGRP Receptor
DAPK
NPC1L1
MALT
DprE1
TOPK
Galectin
VDAC
cell cycle arrest
Amylase
MTH1
ACK
MRGPR
CD73
Pyroptosis
Hippo pathway
Protease
BMI-1
advanced glycation end products
CD38
NEDD8
gp120/CD4
Kisspeptin
Adiponectin receptor
Hexokinase
HCN Channel
KSP
Thrombopoietin Receptor
Liposome
Transaminase
Necroptosis
Hck
RANKL/RANK
Haspin Kinase
Na-K-Cl cotransporter
OXPHOS
Glutathione reductase
AIM2
CPT
GluCls
HuR
KLF
Taste receptor
GSNOR
NUDIX hydrolase
EBI2/GPR183
VDA
FOXO1
Prolyl Endopeptidase (PREP)
Fas/FasL
PACAP
Integrase
PGC-1α
hCE
RXFP receptor
ATTECs
lysosomal autophagy
LYTACs
stilbene oxidase
Hydrogenase
CYP19A1
Piezo Channel
Procollagen C Proteinase
Neuropeptide W
aconitase
LHRH
N-Acetylglucosaminyltransferase
Vitamin
Stemness kinase
Motilin Receptor
FABP
Anion Exchanger
Thioredoxin
Fer/FerT kinase
NMU2R
Glyoxalase

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