Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM).CCG-273220 covalently binds the GRK5 subfamily-specific residue Cys474 and is more selective for GRK5 than GRK2.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 954.00 | |
50 mg | 6-8 weeks | $ 1,240.00 | |
100 mg | 6-8 weeks | $ 1,880.00 |
Description | CCG-273220 is a covalent inhibitor of G protein-coupled receptor (GPCR) kinase 5 (GRK5) (IC50: 220 nM).CCG-273220 covalently binds the GRK5 subfamily-specific residue Cys474 and is more selective for GRK5 than GRK2. |
Molecular Weight | 494.95 |
Formula | C26H24ClFN4O3 |
CAS No. | 2750414-35-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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CCG-273220 2750414-35-6 inhibitor inhibit