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(±)-Enitociclib

Name: (±)-Enitociclib
Brand: TargetMol
SKU: T13467
Price: 31 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T13467Cas No. 1610358-53-6

Alias (±)-BAY-1251152

(±)-Enitociclib ((±)-BAY-1251152) is a racemic mixture of BAY-1251152, a highly selective inhibitor of PTEF/CDK9.

(±)-Enitociclib

🥰Excellent

Purity: 99.29%

Catalog No. T13467Alias (±)-BAY-1251152Cas No. 1610358-53-6

(±)-Enitociclib ((±)-BAY-1251152) is a racemic mixture of BAY-1251152, a highly selective inhibitor of PTEF/CDK9.

Pack Size	Price	Availability
1 mg	$31	In Stock
5 mg	$81	In Stock
10 mg	$123	In Stock
25 mg	$228	In Stock
50 mg	$372	In Stock
100 mg	$596	In Stock
200 mg	$847	In Stock
1 mL x 10 mM (in DMSO)	$89	In Stock

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Batch Information

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Purity:99.29%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	(±)-Enitociclib ((±)-BAY-1251152) is a racemic mixture of BAY-1251152, a highly selective inhibitor of PTEF/CDK9.
Synonyms	(±)-BAY-1251152

Chemical Properties

Molecular Weight	404.43
Formula	C₁₉H₁₈F₂N₄O₂S
Cas No.	1610358-53-6
Smiles	COc1cc(F)ccc1-c1cc(Nc2cc(CS(C)(=N)=O)ccn2)ncc1F
Relative Density.	1.36 g/cm3 (Predicted)
Color	White
Appearance	Solid

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (123.63 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4726 mL	12.3631 mL	24.7262 mL	123.6308 mL
5 mM	0.4945 mL	2.4726 mL	4.9452 mL	24.7262 mL
10 mM	0.2473 mL	1.2363 mL	2.4726 mL	12.3631 mL
20 mM	0.1236 mL	0.6182 mL	1.2363 mL	6.1815 mL
50 mM	0.0495 mL	0.2473 mL	0.4945 mL	2.4726 mL
100 mM	0.0247 mL	0.1236 mL	0.2473 mL	1.2363 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc