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Fesoterodine

Name: Fesoterodine
Brand: TargetMol
SKU: T9419
Rating: 4.5 (1 reviews)

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Catalog No. T9419Cas No. 286930-02-7

Alias (R) Fesoterodine

Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB).

Fesoterodine

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Purity: 97.1%

Catalog No. T9419Alias (R) FesoterodineCas No. 286930-02-7

Pack Size	Price	Availability
5 mg	$47	Backorder
10 mg	$77	Backorder
25 mg	$128	Backorder
50 mg	$189	Backorder
100 mg	$273	Backorder

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Purity:97.1%

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COA HNMR LCMS

Product Introduction

Bioactivity

Description	Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB).
Targets&IC50	M2 mAChR:7.7(pKi), M3 mAChR:7.4(pKi), M1 mAChR:8.0(pKi)
In vivo	Fesoterodine (0.01-1 mg/kg; i.v.) decreases micturition pressure while increasing bladder capacity and ICIs (intercontraction intervals) even at the lowest dose of 0.01 mg/kg [3].
Alias	(R) Fesoterodine

Chemical Properties

Molecular Weight	411.58
Formula	C₂₆H₃₇NO₃
Cas No.	286930-02-7
Smiles	[C@H](CCN(C(C)C)C(C)C)(C1=C(OC(C(C)C)=O)C=CC(CO)=C1)C2=CC=CC=C2
Relative Density.	1.043 g/cm3

Storage & Solubility Information

Storage

Pure form: -20°C for 3 years | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

Ethanol: 50 mg/mL (121.48 mM), Sonication is recommended. (The compound is unstable in solution, please use soon.)

Solution Preparation Table

Ethanol

	1mg	5mg	10mg	50mg
1 mM	2.4297 mL	12.1483 mL	24.2966 mL	121.4831 mL
5 mM	0.4859 mL	2.4297 mL	4.8593 mL	24.2966 mL
10 mM	0.2430 mL	1.2148 mL	2.4297 mL	12.1483 mL
20 mM	0.1215 mL	0.6074 mL	1.2148 mL	6.0742 mL
50 mM	0.0486 mL	0.2430 mL	0.4859 mL	2.4297 mL
100 mM	0.0243 mL	0.1215 mL	0.2430 mL	1.2148 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc