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Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $47 | Backorder | |
10 mg | $77 | Backorder | |
25 mg | $128 | Backorder | |
50 mg | $189 | Backorder | |
100 mg | $273 | Backorder |
Description | Fesoterodine ((R) Fesoterodine) is an orally active, competitive mAChR antagonist with pKi values of 8.0, 7.7, 7.4, 7.3, 7.5 for M1, M2, M3, M4, M5 receptors, respectively. It is used for the overactive bladder (OAB). |
Targets&IC50 | M2 mAChR:7.7(pKi), M3 mAChR:7.4(pKi), M1 mAChR:8.0(pKi) |
In vivo | Fesoterodine (0.01-1 mg/kg; i.v.) decreases micturition pressure while increasing bladder capacity and ICIs (intercontraction intervals) even at the lowest dose of 0.01 mg/kg [3]. |
Alias | (R) Fesoterodine |
Molecular Weight | 411.58 |
Formula | C26H37NO3 |
Cas No. | 286930-02-7 |
Smiles | [C@H](CCN(C(C)C)C(C)C)(C1=C(OC(C(C)C)=O)C=CC(CO)=C1)C2=CC=CC=C2 |
Relative Density. | 1.043 g/cm3 |
Storage | Pure form: -20°C for 3 years | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
Solubility Information | Ethanol: 50 mg/mL (121.48 mM), Sonication is recommended. (The compound is unstable in solution, please use soon.) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
Ethanol
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