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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9019 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9019 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
COX
DNA/RNA Synthesis
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Reactive Oxygen Species
Calcium Channel
Histamine Receptor
VEGFR
Antibiotic
Cytochromes P450
Sodium Channel
HDAC
GABA Receptor
Parasite
PPAR
TRP/TRPV Channel
mTOR
Akt
GPR
AChR
ERK
JAK
Antifungal
Wnt/beta-catenin
Src
HIV Protease
Prostaglandin Receptor
FLT
Estrogen Receptor/ERR
PARP
STAT
p38 MAPK
Adenosine Receptor
Opioid Receptor
PDGFR
Microtubule Associated
AMPK
Dehydrogenase
GSK-3
Nucleoside Antimetabolite/Analog
Topoisomerase
FGFR
Raf
TNF
Caspase
Epigenetic Reader Domain
iGluR
Bcl-2 Family
Estrogen/progestogen Receptor
Influenza Virus
Antioxidant
Glucocorticoid Receptor
c-Met/HGFR
Androgen Receptor
c-Kit
Histone Methyltransferase
Ferroptosis
Bcr-Abl
HSP
Cannabinoid Receptor
PKC
MMP
ATPase
ALK
Sirtuin
IL Receptor
TGF-beta/Smad
Phosphatase
Aurora Kinase
Ras
JNK
PDE
HER
MAPK
P-gp
MEK
Tyrosine Kinases
DUB
IκB/IKK
NO Synthase
ROCK
Mitophagy
ROS
Lipoxygenase
SARS-CoV
p53
NMDAR
Virus Protease
Serine/threonin kinase
CXCR
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
DNA-PK
PKA
RIP kinase
Hedgehog/Smoothened
HSV
IGF-1R
P2X Receptor
Neurokinin receptor
LPL Receptor
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Drug Metabolite
TLR
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FAK
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Antiviral
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PLK
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NOS
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Interleukin
TAM Receptor
Chloride channel
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Serotonin Transporter
Norepinephrine
Casein Kinase
Tyrosinase
Proteasome
PERK
HBV
HCV Protease
RAAS
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Chk
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Phospholipase
Mdm2
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DNA Alkylator/Crosslinker
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PROTACs
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SGLT
Retinoid Receptor
PDK
Syk
P2Y Receptor
MAO
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Melanocortin Receptor
DHFR
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transporter
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Transferase
c-Myc
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LPA Receptor
Anti-infection
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CFTR
PD-1/PD-L1
Integrin
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OX Receptor
CaMK
DNA
GNRH Receptor
Leukotriene Receptor
IRE1
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ADC Cytotoxin
NADPH
Progesterone Receptor
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ABC Transporter
PI4K
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Monoamine Oxidase
YAP
GTPase
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Neurotensin Receptor
IAP
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Immunology/Inflammation related
CSF-1R
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STING
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PTEN
Oxytocin Receptor
Hydroxylase
MLK
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Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
NAMPT
PYK2
SIK
Annexin A
PAFR
MT Receptor
Lipid
Beta-Secretase
OAT
Survivin
CRFR
MELK
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ribosome
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MTH1
DPP-4
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ACK1
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ASK
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CGRP Receptor
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BMI-1
NPC1L1
MALT
ROR
TOPK
Kisspeptin
VDAC
Hck
IDO
Adiponectin Receptor
DNA gyrase
Hexokinase
PAD
ATP Citrate Lyase
LRRK2
Aminopeptidase
Decarboxylase
TSH Receptor
PAI-1
Hippo pathway
Aquaporin
Adenosine Deaminase
p97
PKM
Adenylyl Cyclase
RAR/RXR
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Galectin
AAK1
RANKL/RANK
Haspin Kinase
Na-K-Cl cotransporter
HCN Channel
Epoxide Hydrolase
KSP
CD73
Pyroptosis
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KLF
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NADPH-oxidase
Imidazoline Receptor
EBI2/GPR183
NEDD8
MyD88
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gp120/CD4
VDA
Amylase
OXPHOS
PSMA
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AIM2
GluCls
HuR
Protease
RXFP receptor
Gap Junction Protein
DAPK
Lysosomal Autophagy
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Thyroid hormone receptor(THR)
Advanced Glycation End Products
Transaminase
Hydrogenase
CD38
CYP19A1
Piezo Channel
NUDIX hydrolase
Dynamin
Neuropeptide W
Necroptosis
N-Acetylglucosaminyltransferase
Stemness kinase
FLAP
Phosphorylase
GlyT
Anion Exchanger
PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Transketolase
Thrombopoietin Receptor
cGAS
hCE
Neprilysin
Glyoxalase
Sodium-dependent phosphate transporter
IGF-2R

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