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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9332 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9332 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
DNA/RNA Synthesis
COX
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Epigenetic Reader Domain
Reactive Oxygen Species
Calcium Channel
Histamine Receptor
Antibiotic
VEGFR
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
GABA Receptor
TRP/TRPV Channel
Parasite
JAK
PPAR
mTOR
Akt
ERK
Wnt/beta-catenin
AChR
HIV Protease
GPCR
Antifungal
PARP
Prostaglandin Receptor
PKC
Src
Estrogen Receptor/ERR
FLT
STAT
p38 MAPK
FGFR
Microtubule Associated
Adenosine Receptor
AMPK
PDGFR
GSK-3
Dehydrogenase
Topoisomerase
TNF
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c-Kit
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Bcr-Abl
ALK
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ATPase
MMP
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TGF-beta/Smad
Ras
Aurora Kinase
Phosphatase
IL Receptor
JNK
ROCK
PDE
DUB
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MAPK
MEK
ROS
NO Synthase
p53
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Ligands for Target Protein for PROTAC
NAMPT
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ribosome
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NEDD4-1
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Glyoxalase
Sodium-dependent phosphate transporter

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