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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9332 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9332 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
DNA/RNA Synthesis
COX
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Epigenetic Reader Domain
Reactive Oxygen Species
Calcium Channel
Antibiotic
Histamine Receptor
VEGFR
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
GABA Receptor
Parasite
TRP/TRPV Channel
JAK
PPAR
mTOR
Akt
ERK
Wnt/beta-catenin
AChR
HIV Protease
GPCR
Antifungal
PARP
Prostaglandin Receptor
PKC
Src
Estrogen Receptor/ERR
STAT
FLT
p38 MAPK
FGFR
Microtubule Associated
Adenosine Receptor
AMPK
PDGFR
GSK-3
Nucleoside Antimetabolite/Analog
Dehydrogenase
Topoisomerase
TNF
Estrogen/progestogen Receptor
Raf
Opioid Receptor
Glucocorticoid Receptor
Bcl-2 Family
Caspase
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Antioxidant
iGluR
Androgen Receptor
Ferroptosis
c-Met/HGFR
c-Kit
Sirtuin
HSP
Bcr-Abl
ALK
MMP
Cannabinoid Receptor
ATPase
Histone Demethylase
TGF-beta/Smad
Ras
Phosphatase
Aurora Kinase
IL Receptor
JNK
ROCK
PDE
DUB
Tyrosine Kinases
ROS
MAPK
MEK
P-gp
NO Synthase
p53
IκB/IKK
Mitophagy
RIP kinase
Virus Protease
NMDAR
Lipoxygenase
SARS-CoV
Serine/threonin kinase
S1P Receptor
PKA
HSV
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CXCR
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NOD
DNA-PK
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IGF-1R
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LPL Receptor
TLR
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c-RET
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ATM/ATR
S6 Kinase
P2X Receptor
FAK
Casein Kinase
HER
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PLK
HIF
Chloride channel
NOS
Pim
Mitochondrial Metabolism
Sigma receptor
TAM Receptor
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RAAS
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PDK
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transporter
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CFTR
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IRE1
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OX Receptor
ROS Kinase
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GRK
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GPX
Hydroxylase
APC/C
MLK
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CRM1
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
NAMPT
PYK2
Annexin A
PAFR
MT Receptor
Lipid
OAT
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LRRK2
CRFR
MELK
RSV
ribosome
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Apelin receptor
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TOPK
Cell Cycle Arrest
MTH1
DPP-4
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ACK1
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ASK
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Discoidin Domain Receptor (DDR)
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RANKL/RANK
IDO
Adiponectin Receptor
DNA gyrase
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TSH Receptor
PAI-1
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GST
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p97
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AAK1
VDAC
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HCN Channel
Epoxide Hydrolase
KSP
CD73
HuR
KLF
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DAPK
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EBI2/GPR183
MyD88
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gp120/CD4
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OXPHOS
PSMA
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AIM2
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IKZF
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Transketolase
Huntingtin
cGAS
hCE
NEDD4-1
Neprilysin
Glyoxalase
Sodium-dependent phosphate transporter
Vitamin

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