Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 8700 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 8700 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
5-HT Receptor
Adrenergic Receptor
CDK
Dopamine Receptor
DNA/RNA Synthesis
EGFR
COX
PI3K
Histamine Receptor
Potassium Channel
VEGFR
Antibacterial
Calcium Channel
Sodium Channel
HDAC
mTOR
GPR
Antibiotic
TRP/TRPV Channel
P450
Src
FLT
JAK
PDGFR
GABA Receptor
Opioid Receptor
Raf
Wnt/beta-catenin
PPAR
Adenosine Receptor
GSK-3
FGFR
AChR
Prostaglandin Receptor
NF-κB
c-Kit
Nucleoside Antimetabolite/Analog
Reactive Oxygen Species
Estrogen Receptor/ERR
PARP
Epigenetic Reader Domain
c-Met/HGFR
Parasite
Glucocorticoid Receptor
Dehydrogenase
iGluR
Microtubule Associated
Histone Methyltransferase
Bcr-Abl
Akt
ERK
Androgen Receptor
HIV Protease
Estrogen/progestogen Receptor
Cannabinoid Receptor
HSP
Topoisomerase
Aurora Kinase
ALK
Kras
Endogenous Metabolite
Antifungal
STAT
Ras
Sirtuin
AMPK
HER
p38 MAPK
ROCK
DUB
Tyrosine Kinases
TGF-beta/Smad
BCL
Ferroptosis
Phosphatase
MAPK
MEK
Serine/threonin kinase
PDE
DNA-PK
PKC
CXCR
IκB/IKK
ATPase
Neurokinin receptor
p53
S1P Receptor
LPL Receptor
Caspase
RIP kinase
NMDAR
SARS-CoV
E1/E2/E3 Enzyme
P2X Receptor
BTK
Hedgehog/Smoothened
IGF-1R
Influenza Virus
c-RET
S6 Kinase
Sigma receptor
Drug Metabolite
ATM/ATR
PLK
TAM Receptor
Mitophagy
PKA
Serotonin Transporter
MMP
Norepinephrine
TNF
FAK
HIF/HIF Prolyl-Hydroxylase
ADC Cytotoxin
Casein Kinase
Proteasome
Proton pump
Rho
Chk
GluR
Trk receptor
HIF
Protease-activated Receptor
PERK
Endothelin Receptor
Mdm2
JNK
Neuropeptide Y Receptor
P-gp
Chloride channel
DNA Alkylator/Crosslinker
Pim
NOD
Glucagon Receptor
Guanylate cyclase
IRAK
Gamma-secretase
ROS
Melanocortin Receptor
Phospholipase
Carbonic Anhydrase
RAAS
Virus Protease
Mitochondrial Metabolism
HSV
Bradykinin Receptor
Lipoxygenase
SGLT
Retinoid Receptor
c-Fms
Syk
P2Y Receptor
IL Receptor
Interleukin
PDK
HCV Protease
Smo
DNA Alkylation
OX Receptor
LPA Receptor
cholecystokinin
CFTR
PROTACs
DHFR
DYRK
Histone Demethylase
GNRH Receptor
HBV
Vasopressin Receptor
PI4K
DNA Methyltransferase
Antioxidant
GTPase
c-Myc
Fatty Acid Synthase
DNA
Antiviral
Reverse Transcriptase
ROS Kinase
PD-1/PD-L1
Kinesin
Antifolate
Neurotensin Receptor
IRE1
TLR
Transferase
Progesterone Receptor
Leukotriene Receptor
Somatostatin
cAMP
CaMK
GHSR
YAP
NADPH
CSF-1R
Histone Acetyltransferase
Beta Amyloid
NO Synthase
Serine Protease
MAO
Nrf2
Ligand for E3 Ligase
Monocarboxylate transporter
Integrin
CaSR
IAP
GRK
Aromatase
NOD-like Receptor (NLR)
Monoamine Oxidase
Melatonin Receptor
ABC
Indoleamine 2,3-Dioxygenase (IDO)
Tyrosinase
Apelin receptor
NOS
MRP
LIM Kinase
Myosin
CCR
Telomerase
BCRP
STING
GPCR19
Ephrin Receptor
AhR
LTR
IFNAR
Arrestin
Na+/Ca2+ Exchanger
Tie-2
Glutathione Peroxidase
Aryl Hydrocarbon Receptor
SIK
Annexin A
Antifection
Monoamine Transporter
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Bombesin Receptor
Wee1
AChE
MNK
transporter
HMG-CoA Reductase
Thrombin
MLK
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
Ligands for Target Protein for PROTAC
Cysteine Protease
Glucokinase
PYK2
APC
PAK
PSMA
CRFR
MELK
GPX
Hydroxylase
Reductase
OCT
NAMPT
Glutaminase
MT Receptor
DPP-4
ACK
PGE Synthase
Acyltransferase
Survivin
Porcupine
LRRK2
Free radical scavengers
ASK
RSV
CGRP Receptor
SGK
BMI-1
BACE
TOPK
Kisspeptin
VDAC
Liver X Receptor
FXR
IDO
Immunology/Inflammation related
MTH1
FAAH
KSP
Lipid
Beta-Secretase
OAT
TSH Receptor
Methionine Adenosyltransferase (MAT)
Hippo pathway
ribosome
CRISPR/Cas9
Oxytocin Receptor
Aquaporin
Adenosine deaminase
Discoidin Domain Receptor (DDR)
p97
PKM
NPC1L1
Amino Acids and Derivatives
Galectin
Hck
Haspin Kinase
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Hexokinase
HCN Channel
PAD
Xanthine Oxidase
ATP Citrate Lyase
CD73
PAI-1
Carboxypeptidase
KLF
Complement System
Adenylyl cyclase
CAT
MALT
ROR
EBI2/GPR183
NEDD8
RAR/RXR 
VDA
Factor Xa
Adiponectin receptor
DNA gyrase
PTEN
Epoxide Hydrolase
OXPHOS
AIM2
Decarboxylase
HuR
GST
Protease
Gap Junction Protein
DAPK
Platelet aggregation
NADPH-oxidase
lysosomal autophagy
Imidazoline Receptor
advanced glycation end products
CD38
NUDIX hydrolase
Piezo Channel
MyD88
Neuropeptide W
Lipase
Necroptosis
N-Acetylglucosaminyltransferase
cell cycle arrest
Stemness kinase
RANKL/RANK
FLAP
Motilin Receptor
UGT
PAFR
LDL
GlyT
Anion Exchanger
Thioredoxin
Angiotensin-converting Enzyme (ACE)
Thrombopoietin Receptor
Glutathione reductase
Aminopeptidase
cGAS
GluCls
Pyroptosis
Neprilysin
RXFP receptor

Keywords