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TargetMol | Compound Library

Protease Inhibitor Library

Catalog No. L1100

Protease inhibitors are molecules that inhibit the function of proteases (enzymes that aid the breakdown of proteins), including proteins protease inhibitors, natural protease inhibitors, and synthetic protease inhibitors. (1). Antiprotozoal activity: protease inhibitors could be used against malaria and gastrointestinal protozoal infections; (2). Antiretrovirals: protease inhibitors were the second class of antiretroviral drugs developed widely used to treat HIV/AIDS and hepatitis C; (3). Anticancer activity: Researchers are investigating whether protease inhibitors could possibly be used to treat cancer. For example, nelfinavir and atazanavir are able to kill tumor cells in culture. Inhibitors of the proteasome, such as bortezomib are now front-line drugs for the treatment of multiple myeloma. Marimastat and batimastat are two of the matrix metalloproteinase inhibitors that can be used to treat cancer. The Protease Inhibitor Library by TargetMol, containing 507 small protease and proteasome inhibitors, can be used for research in Chemical Genomics and drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1100

Protease Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 507 protease and proteasome inhibitors for research in chemical genomics, and drug screening;
  • Targets include proteasome, DPP-4, Serine protease, cysteine protease, MMP, Aspartic proteinases, etc;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

MMP
Caspase
Proteasome
Apoptosis
Cysteine Protease
Gamma-secretase
Virus Protease
Autophagy
SARS-CoV
Serine Protease
HIV Protease
DPP-4
Thrombin
Antibacterial
HCV Protease
Bcl-2 Family
Endogenous Metabolite
PARP
NF-κB
p38 MAPK
Parasite
Beta Amyloid
COX
Factor Xa
Reactive Oxygen Species
Akt
Antibiotic
Cytochromes P450
IL Receptor
Protease
TNF
Antifungal
Antiviral
Carboxypeptidase
ERK
JNK
HSV
Immunology/Inflammation related
Influenza Virus
P-gp
PI3K
PPAR
Serine/threonin kinase
Antioxidant
Dehydrogenase
DNA/RNA Synthesis
DUB
Ferroptosis
ROS
5-HT Receptor
BACE
CDK
Drug Metabolite
Estrogen/progestogen Receptor
GABA Receptor
HDAC
HIF/HIF Prolyl-Hydroxylase
Interleukin
JAK
Lipoxygenase
NO Synthase
Nrf2
PKC
Prostaglandin Receptor
STAT
TRP/TRPV Channel
AChR
AMPK
Anti-infection
ATM/ATR
Beta-Secretase
Calcium Channel
DNA Methyltransferase
Epigenetic Reader Domain
Free radical scavengers
Histamine Receptor
IAP
MAPK
Mitophagy
mTOR
NOD-like Receptor (NLR)
p53
PAI-1
Phosphatase
Phospholipase
Potassium Channel
Pyroptosis
Rho
ribosome
Thrombopoietin Receptor
Tyrosinase
Wnt/beta-catenin
Adrenergic Receptor
AIM2
ALK
Amino Acids and Derivatives
Aminopeptidase
Antifection
ATPase
Aurora Kinase
CaMK
cAMP
Carbonic Anhydrase
CFTR
Complement System
DNA
DNA-PK
Dopamine Receptor
Dynamin
E1/E2/E3 Enzyme
FAK
Fatty Acid Synthase
gp120/CD4
GPR
GSK-3
IGF-1R
IκB/IKK
MAO
Neprilysin
NMDAR
Nucleoside Antimetabolite/Analog
Opioid Receptor
PAFR
PI4K
PKA
Platelet aggregation
Protease-activated Receptor
Proton pump
Ras
ROR
S1P Receptor
Sodium Channel
Somatostatin
Src
STING
TLR
UGT
BTK