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Esmolol hydrochloride

Name: Esmolol hydrochloride
Brand: TargetMol
SKU: T1503
Rating: 4.5 (1 reviews)

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Catalog No. T1503Cas No. 81161-17-3

Alias Esmolol HCl, ASL8052

Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instances of clinically apparent drug induced liver injury.

Esmolol hydrochloride

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Purity: 99.48%

Catalog No. T1503Alias Esmolol HCl, ASL8052Cas No. 81161-17-3

Pack Size	Price	Availability
25 mg	$1,520	4-6 weeks
50 mg	$1,980	4-6 weeks
100 mg	$2,500	4-6 weeks

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Bulk & Custom

This molecule is a custom-made product. TargetMol has an excellent synthesis team with the experience and capability to provide you with cost-effective products. However, due to objective factors, there is a small probability that the synthesis may not be successful during the R&D process. We appreciate your understanding. If you have any questions, please feel free to contact us. We are committed to serving you wholeheartedly.

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Batch Information

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Purity:99.48%

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COA

Product Introduction

Bioactivity

Description	Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to instances of clinically apparent drug induced liver injury.
In vitro	The main active site of Esmolol is the sinus node and AV node conduction system, and Esmolol has a rapid onset of action and inactivation.
In vivo	The main active site of Esmolol is the sinus node and AV node conduction system, and Esmolol has a rapid onset of action and inactivation.
Synonyms	Esmolol HCl, ASL8052

Chemical Properties

Molecular Weight	331.15
Formula	C₁₆H₂₅NO₄·HCl
Cas No.	81161-17-3
Smiles	c1(ccc(cc1)CCC(=O)OC)OCC(CNC(C)C)O.Cl
Relative Density.	1.026

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 198.9 mM, Sonication is recommended.

H2O: 150.68 mM, Sonication is recommended.

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	3.0198 mL	15.0989 mL	30.1978 mL	150.9890 mL
5 mM	0.6040 mL	3.0198 mL	6.0396 mL	30.1978 mL
10 mM	0.3020 mL	1.5099 mL	3.0198 mL	15.0989 mL
20 mM	0.1510 mL	0.7549 mL	1.5099 mL	7.5494 mL
50 mM	0.0604 mL	0.3020 mL	0.6040 mL	3.0198 mL
100 mM	0.0302 mL	0.1510 mL	0.3020 mL	1.5099 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc