Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and <1 μM for ATP hydrolysis, respectively, with a selectivity ratio of <6.4 favoring cGAMP hydrolysis inhibition [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP hydrolysis, respectively, with a selectivity ratio of >6.4 favoring cGAMP hydrolysis inhibition [1]. |
Molecular Weight | 328.41 |
Formula | C18H24N4O2 |
CAS No. | 2289736-54-3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Enpp-1-IN-17 2289736-54-3 inhibitor inhibit