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KDM2B-IN-2

Catalog No. T39389 CAS 1965248-01-4

KDM2B-IN-2 is a potent <a href="/target/Histone_Demethylase" style="display: inline; color: #c13a36">Histone Demethylase</a> (kdm2b) inhibitor.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

KDM2B-IN-2, CAS 1965248-01-4

Pack Size	Availability	Price/USD
1 mg	In stock	$ 78.00
5 mg	In stock	$ 167.00
10 mg	In stock	$ 257.00
25 mg	In stock	$ 473.00
50 mg	In stock	$ 725.00
100 mg	In stock	$ 997.00
200 mg	In stock	$ 1,555.00
1 mL * 10 mM (in DMSO)	In stock	$ 195.00

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Purity: 97.57%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	KDM2B-IN-2 is a potent histone demethylase (kdm2b) inhibitor.
Targets&IC50	KDM2B:0.021 μM (IC50)
In vitro	In a KDM2B TR-FRET assay, KDM2B-IN-2 shows an IC50 of 0.021μM[1].

Molecular Weight	430.59
Formula	C21H26N4O2S2
CAS No.	1965248-01-4

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 28.8mg/mL (66.9mM), Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Brian K. Albrecht, et al. 4,5-dihydroimidazole derivatives and their use as histone demethylase (kdm2b) inhibitors. Patent WO2016112251A1.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Bioactive Compounds Library Max Inhibitor Library

Related Products

Related compounds with same targets

Methylstat Eicosapentaenoic Acid KDM2B-IN-2 GSK2879552 CP2 CPI-455 HCl KF21213 S2101

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Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

KDM2B-IN-2 1965248-01-4 Chromatin/Epigenetic Histone Demethylase KDM2B IN 2 KDM-2B-IN-2 KDM2BIN2 Inhibitor inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.