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Fasentin

Name: Fasentin
Brand: TargetMol
SKU: T8616
Price: 34 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T8616Cas No. 392721-37-8

Alias N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide

Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.

Fasentin

🥰Excellent

Purity: 99.95%

Catalog No. T8616Alias N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamideCas No. 392721-37-8

Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.

Pack Size	Price	Availability
2 mg	$34	In Stock
5 mg	$55	In Stock
10 mg	$89	In Stock
25 mg	$163	In Stock
50 mg	$247	In Stock
100 mg	$369	In Stock
200 mg	$549	In Stock
1 mL x 10 mM (in DMSO)	$61	In Stock

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Batch Information

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Purity:99.95%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.
Targets&IC50	GLUT4:68 μM (IC50)
In vitro	Fasentin has been described as a modulator of GLUT-1 and GLUT-4 transporters, thus inhibiting glucose uptake in some cancer cells.
Synonyms	N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide

Chemical Properties

Molecular Weight	279.64
Formula	C₁₁H₉ClF₃NO₂
Cas No.	392721-37-8
Smiles	CC(=O)CC(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Relative Density.	1.411 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 25 mg/mL (89.4 mM), Sonication is recommended.

In Vivo Formulation

10% DMSO+40% PEG300+5% Tween 80+45% Saline: 2 mg/mL (7.15 mM), Sonication is recommended.

Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.5760 mL	17.8801 mL	35.7603 mL	178.8013 mL
5 mM	0.7152 mL	3.5760 mL	7.1521 mL	35.7603 mL
10 mM	0.3576 mL	1.7880 mL	3.5760 mL	17.8801 mL
20 mM	0.1788 mL	0.8940 mL	1.7880 mL	8.9401 mL
50 mM	0.0715 mL	0.3576 mL	0.7152 mL	3.5760 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc