Shopping Cart

Your shopping cart is currently empty

Pirenzepine dihydrochloride

Name: Pirenzepine dihydrochloride
Brand: TargetMol
SKU: T1542
Price: 33 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T1542Cas No. 29868-97-1

Alias Tabe, Pirenzepine HCl, LS519, Bisvanil

Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.

Pirenzepine dihydrochloride

🥰Excellent

Purity: 99.62%

Catalog No. T1542Alias Tabe, Pirenzepine HCl, LS519, BisvanilCas No. 29868-97-1

Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.

Pack Size	Price	USA Warehouse	Global Warehouse
100 mg	$33	In Stock	In Stock
500 mg	$65	In Stock	In Stock
1 g	$93	-	In Stock
1 mL x 10 mM (in H2O)	$36	In Stock	In Stock

Add to Cart

Add to Quotation

In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Questions

Batch Information

Select Batch

Purity:99.62%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.
Synonyms	Tabe, Pirenzepine HCl, LS519, Bisvanil

Chemical Properties

Molecular Weight	424.32
Formula	C₁₉H₂₁N₅O₂·2HCl
Cas No.	29868-97-1
Smiles	Cl.Cl.CN1CCN(CC(=O)N2c3ccccc3C(=O)Nc3cccnc23)CC1
Relative Density.	no data available

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: Insoluble

H2O: 10 mM, Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
1 mM	2.3567 mL	11.7836 mL	23.5671 mL	117.8356 mL
5 mM	0.4713 mL	2.3567 mL	4.7134 mL	23.5671 mL
10 mM	0.2357 mL	1.1784 mL	2.3567 mL	11.7836 mL

Calculator

Molarity Calculator
Dilution Calculator
Reconstitution Calculator
Molecular Weight Calculator

In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc