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Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.

  • Tirzepatide Acetate(2023788-19-2 free base)
    TP1111L
    Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
    • $358
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  • Liraglutide
    T6876204656-20-2
    Liraglutide (Liraglutida) is a long-acting GLP-1 receptor agonist.
    • $119
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    TargetMol | Citations Cited
  • GLP-1(7-36), amide
    T3984107444-51-9
    GLP-1(7-36), amide (MKC 253) is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays various antidiabetic effects by potentiating glucose-induced secretion of insulin from pancreatic β-cells, increasing insulin expression.
    • $185
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  • Semaglutide
    T19850910463-68-2
    Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
    • $213
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  • Orforglipron
    T114082212020-52-3
    Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1 diabetes in adults.
    • $256
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  • NNC 92-1687
    T2818222903-37-3In house
    NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.
    • $397
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  • PF-06882961 Tris
    T88762230198-03-3
    PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
    • $133
    In Stock
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  • HAEGTFTSDVS acetate
    TP1382L
    HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.
    • $148
    In Stock
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  • Tirzepatide monosodium salt
    TP1111L1
    Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.
    • $263
    In Stock
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  • Semaglutide Acetate
    T19850L1997361-85-9
    Semaglutide Acetate is an agonist of a glucagon-like peptide 1 (GLP-1) receptor and can be used in studies about the treatment of type 2 diabetes.
    • $239
    In Stock
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  • Retatrutide sodium salt
    T76279L1
    Retatrutide sodium salt is a potent triple agonist peptide for glucagon receptor (GCGR), glucose-dependent proinsulinotropic polypeptide receptor (GIPR), and glucagon-like peptide-1 receptor (GLP-1R) Retatrutide sodium salt is used in the study of type 2 diabetes and obesity.
    • $247
    In Stock
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  • Glucagon (19-29), human acetate
    TP1863L
    Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
    • $59
    In Stock
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  • GLP-1(28-36)amide acetate
    T37890L
    GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
    • $129
    In Stock
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  • HAEGTFT acetate(926018-95-3 free base)
    TP1419L
    HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
    • $171
    In Stock
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  • Albiglutide TFA (782500-75-8 free base)
    TP1796
    Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
    • $167
    In Stock
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    TargetMol | Citations Cited
  • (S, R)-LSN 3318839
    T63166L2765539-92-0In house
    (S, R)-LSN 3318839 is an allosteric modulator of the glucagon-like peptide-3318839 receptor (GLP-1R) that has demonstrated powerful hypoglycemic effects in animal models alone or in combination with sitagliptin.
    • $195
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  • Secretin (33-59), rat
    TP1039121028-49-7
    Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.
    • $176
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  • Oxyntomodulin acetate
    TP1976L
    Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
    • $185
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  • Teduglutide acetate
    T35337L
    Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial function through an altered distribution of claudin-10, facilitating sodium recirculation for Na-coupled glucose transport and water absorption.
    • $112
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  • Bay 55-9837 acetate
    TP2071L
    Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
    • $539
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  • Mazdutide acetate(2259884-03-0 free base)
    T78097L
    Mazdutide acetate is a potent co-agonist of glucagon-like peptide (GLP-1R) and glucagon receptor (GCGR), a gastrin-regulating hormone analog.Mazdutide acetate stimulates insulin secretion from mouse pancreatic islets, and can be used in studies of obesity and type 2 diabetes (T2D).
    • $89
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  • Avexitide acetate
    TP2100L2051593-46-3
    Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.
    • $169
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  • GLP-1 receptor agonist 9 citrate
    T9579L
    GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
    • $195
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  • LGD-6972
    T118451207989-09-0In house
    LGD-6972 is an antagonist of glucagon receptor.
    • $81
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  • LSN3318839
    T631662764704-18-7In house
    LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be used to lower blood glucose.
    • $213
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  • GRA Ex-25
    T3422307983-31-9
    GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
    • $57
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    TargetMol | Citations Cited
  • Exendin-4
    T3967141758-74-9
    Exendin-4 (Exenatide) is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer half-life of 2.4 hours.
    • $57
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    TargetMol | Citations Cited
  • Glucagon-like peptide 1 (1-37), human acetate
    TP1148L
    Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
    • $397
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  • HAEGTFTSD acetate(926018-45-3 free base)
    TP1452L1
    HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from intestinal L-cells, in response to the ingestion of food.
    • $266
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  • V-0219
    T60047878453-71-5
    V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
    • $113
    5 days
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  • Semaglutide TFA (910463-68-2 free base)
    T12878
    Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
    • $232
    Backorder
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  • Teduglutide
    T35337197922-42-2
    Teduglutide is a useful organic compound for research related to life sciences. The catalog number is T35337 and the CAS number is 197922-42-2.
    • $183
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  • BETP
    TQ01241371569-69-5
    BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
    • $40
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  • Retatrutide
    T762792381089-83-2
    Retatrutide (LY3437943) is a triple agonist of the glucagon receptor, glucose-dependent insulinotropic polypeptide receptor, and glucagon-like peptide-1 receptor (GLP-1R), and inhibits GCGR, GIPR, and GLP-1R.Retatrutide can be used to study obesity.
    • $247
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  • GLP-1 (9-36) amide
    TP2252161748-29-4
    antagonist at the human GLP-1 receptor
    • $81
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  • GLP-1R Agonist DMB
    T36579281209-71-0
    GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
    • $47
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  • Shanzhiside methyl ester
    T389664421-28-9
    Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 MAPK signaling.
    • $30
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  • Lixisenatide acetate (320367-13-3 free base)
    TP14691997361-87-1
    Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
    • $97
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  • Tirzepatide
    TP11112023788-19-2
    Tirzepatide (LY-3298176) is a dual agonist of glucose-dependent polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) receptor with neuroprotective activity for the study of diabetes and obesity.
    • $266
    In Stock
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  • Avexitide
    TP2100133514-43-9
    Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.
    • $198
    In Stock
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  • GLP-1 receptor agonist 9
    T95792401892-71-3
    1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.
    • $148
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  • Cotadutide acetate
    TP1103
    Cotadutide acetate (MEDI0382 acetate) is a potent peptide dual agonist of glucagon-like peptide-1 (GLP-1) and glucagon receptor with EC50 of 6.9 pM and 10.2 pM, respectively.
    • $153
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  • 3-Deoxyglucosone
    T191174084-27-9
    3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with protein amino groups to form advanced glycosylated end proteins (AGEs).3-Deoxyglucosone inactivates glutathione peroxidase and synergizes with low glucose to enhance GLP-1 secretion.3-Deoxyglucosone is used as a biomarker for diabetes mellitus.3-Deoxyglucosone has been shown to be an inhibitor of GLP-1 secretion in the presence of low glucose. 3-Deoxyglucosone inactivates glutathione oxidase, synergizes with low glucose to enhance GLP-1 secretion, and can be used as a biologic marker for diabetes.
    • $188
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  • PF-06291874
    TQ02391393124-08-7
    PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
    • $55
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  • GLP-1(7-37) acetate(106612-94-6 free base)
    TP13761450806-98-0
    Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.
    • $113
    In Stock
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  • V-0219 hydrochloride
    T60047L
    V-0219 hydrochloride, an orally-active positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), is utilized in obesity-associated diabetes research.
    • $59
    In Stock
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  • GLP-1R modulator L7-028
    T402792648317-95-5
    GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.
    • $58
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  • GLP-1R modulator C5
    T61483421578-93-0
    GLP-1R modulator C5 is a small molecule GLP-1R orthosteric modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.
    • $35
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  • Adomeglivant
    T141301488363-78-5
    Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
    • $32
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  • GLP-1R agonist 3
    T639092428640-18-8
    GLP-1R agonist 3 is a thickened imidazole derivative compound that is a potent agonist of GLP-1R. GLP-1R agonist 3 has shown research potential in diabetes.
    • $128
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