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ERAP2-IN-1

Name: ERAP2-IN-1
Brand: TargetMol
SKU: T62861
Price: 52 USD
Availability: InStock
Rating: 5 (10 reviews)

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Synonyms:

Catalog No. T62861 Copy Product Info

Purity: 99.58%

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ERAP2-IN-1 is a non-competitive inhibitor of endoplasmic reticulum aminopeptidase 2 (ERAP2). ERAP2-IN-1 specifically inhibits the peptidase activity of ERAP2, blocking the hydrolysis of Arg-AMC (IC₅₀: 27 μM) and the hydrolysis of model peptides (IC₅₀: 44 μM).

Cas No. 2420551-38-6

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Pack Size	Price	USA Stock	Global Stock
1 mg	$52	-	In Stock
5 mg	$123	-	In Stock
10 mg	$198	-	In Stock
25 mg	$455	-	In Stock
50 mg	$789	-	In Stock
100 mg	$1,280	-	In Stock
1 mL x 10 mM (in DMSO)	$123	-	In Stock

For In stock only · Estimated delivery: USA Stock (1-2 days) Global Stock (5-7 days)

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With extensive experience in compound synthesis, we can provide rapid custom synthesis services for this product according to your research needs.

For research use only—not for human use. No sales to individuals. Use as intended only.

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Purity:99.58%

Appearance:Solid

Color:White

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COA HNMR LCMS

Product Introduction

Bioactivity

Description

Chemical Properties

Molecular Weight	458.45
Formula	C₂₀H₂₁F₃N₂O₅S
Cas No.	2420551-38-6
Smiles	O=C(O)C1=CC=C(OC)C(=C1)S(=O)(=O)NC2=CC=C(C=C2N3CCCCC3)C(F)(F)F

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 200 mg/mL (436.25 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.1813 mL	10.9063 mL	21.8126 mL	109.0631 mL
5 mM	0.4363 mL	2.1813 mL	4.3625 mL	21.8126 mL
10 mM	0.2181 mL	1.0906 mL	2.1813 mL	10.9063 mL
20 mM	0.1091 mL	0.5453 mL	1.0906 mL	5.4532 mL
50 mM	0.0436 mL	0.2181 mL	0.4363 mL	2.1813 mL
100 mM	0.0218 mL	0.1091 mL	0.2181 mL	1.0906 mL

Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 µL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 µL Tween 80 and mix well until fully clarified.

3) Add 450 µL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Related Tags: ERAP2-IN-1 chemical structure | ERAP2-IN-1 formula | ERAP2-IN-1 molecular weight