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(S)-Amisulpride

🥰Excellent
Catalog No. T26375Cas No. 71675-92-8
Alias SEP-4199, Esamisulpride, (S) Amisulpride

(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist. (S)-Amisulpride is an antagonist at the 5-HT7 receptor with a Ki of 900 nM. (S)-Amisulpride has antipsychotic and antidepressant effects.

(S)-Amisulpride
Other Forms of (S)-Amisulpride:

(S)-Amisulpride

🥰Excellent
Purity: 98.38%
Catalog No. T26375Alias SEP-4199, Esamisulpride, (S) AmisulprideCas No. 71675-92-8
(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist. (S)-Amisulpride is an antagonist at the 5-HT7 receptor with a Ki of 900 nM. (S)-Amisulpride has antipsychotic and antidepressant effects.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$30In StockIn Stock
5 mg$81In StockIn Stock
10 mg$132In StockIn Stock
25 mg$251In StockIn Stock
50 mg$397In StockIn Stock
100 mg$538In StockIn Stock
200 mg$691-In Stock
1 mL x 10 mM (in DMSO)$90In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:98.38%
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COA LCMS HNMR HPLC

Product Introduction

Bioactivity
Description
(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist. (S)-Amisulpride is an antagonist at the 5-HT7 receptor with a Ki of 900 nM. (S)-Amisulpride has antipsychotic and antidepressant effects.
Targets&IC50
5-HT7:900 nM(Ki)
SynonymsSEP-4199, Esamisulpride, (S) Amisulpride
Chemical Properties
Molecular Weight369.48
FormulaC17H27N3O4S
Cas No.71675-92-8
SmilesCCN1CCC[C@H]1CNC(=O)c1cc(c(N)cc1OC)S(=O)(=O)CC
Relative Density.1.31g/cm3
ColorYellow
AppearanceViscous
Storage & Solubility Information
StoragePure form: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: 100 mg/mL (270.65 mM), Sonication is recommended.
In Vivo Formulation
10% DMSO+40% PEG300+5% Tween 80+45% Saline: 4 mg/mL (10.83 mM), Sonication is recommended.
Please add the solvents sequentially, clarifying the solution as much as possible before adding the next one. Dissolve by heating and/or sonication if necessary. Working solution is recommended to be prepared and used immediately. The formulation provided above is for reference purposes only. In vivo formulations may vary and should be modified based on specific experimental conditions.
Solution Preparation Table
DMSO
1mg5mg10mg50mg
1 mM2.7065 mL13.5325 mL27.0651 mL135.3253 mL
5 mM0.5413 mL2.7065 mL5.4130 mL27.0651 mL
10 mM0.2707 mL1.3533 mL2.7065 mL13.5325 mL
20 mM0.1353 mL0.6766 mL1.3533 mL6.7663 mL
50 mM0.0541 mL0.2707 mL0.5413 mL2.7065 mL
100 mM0.0271 mL0.1353 mL0.2707 mL1.3533 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
1 Enter information below:
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μL
2 Enter the in vivo formulation:
% DMSO
%
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Keywords

Serotonin ReceptorSEP4199SEP 4199InhibitorinhibitDopamineReceptorDopamine ReceptorD3D2antipsychoticantidepressantAmisulpride5-hydroxytryptamine Receptor5HTReceptor5-HT75-HT Receptor5HT Receptor(S)-Amisulpride(S)Amisulpride(R)-amisulpride
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