Powder: -20°C for 3 years | In solvent: -80°C for 1 year
MARK4 Inhibitor 2 is a potent inhibitor of Microtubule Affinity-Regulating Kinase 4 (MARK4), exhibiting a Kₘ of 6.3×10⁷ and an IC₅₀ of 0.82 μM. It effectively inhibits the growth of human cells, thereby offering potential for use in cancer research [1].
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Description | MARK4 Inhibitor 2 is a potent inhibitor of Microtubule Affinity-Regulating Kinase 4 (MARK4), exhibiting a Kₘ of 6.3×10⁷ and an IC₅₀ of 0.82 μM. It effectively inhibits the growth of human cells, thereby offering potential for use in cancer research [1]. |
In vitro | MARK4 inhibitor 2 (Compound 23a) at concentrations of 0-20 μM over 24 hours inhibits the proliferation of HeLa, U87MG, MDA-MB-435, U251, and HGFs cells, with EC50 values ranging from 1.76 μM to 7.98 μM [1]. |
Molecular Weight | 542.63 |
Formula | C34H30N4O3 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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MARK4 inhibitor 2 Chromatin/Epigenetic PI3K/Akt/mTOR signaling AMPK inhibitor inhibit