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TOPRelated productsBioactivityChemical infoStorage&SolubilityCalculator

[Lys5,MeLeu9,Nle10]-NKA(4-10)

🥰Excellent
Catalog No. TP1883Cas No. 137565-28-7

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).

[Lys5,MeLeu9,Nle10]-NKA(4-10)
Other Forms of [Lys5,MeLeu9,Nle10]-NKA(4-10):
[Lys5,MeLeu9,Nle10]-NKA(4-10) TFAT75882
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[Lys5,MeLeu9,Nle10]-NKA(4-10)

🥰Excellent
Catalog No. TP1883Cas No. 137565-28-7
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
Pack SizePriceAvailabilityQuantity
1 mg$103In Stock
5 mg$257In Stock
10 mg$380In Stock
25 mg$592In Stock
50 mg$816In Stock
100 mg$1,090In Stock
200 mg$1,480In Stock
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Purity:>99.99%
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Product Introduction

Bioactivity
Description
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
Chemical Properties
Molecular Weight803.99
FormulaC39H65N9O9
Cas No.137565-28-7
Smiles[C@@H](CC1=CC=CC=C1)(NC([C@@H](NC([C@H](CC(O)=O)N)=O)CCCCN)=O)C(N[C@H](C(NCC(N([C@H](C(N[C@@H](CCCC)C(N)=O)=O)CC(C)C)C)=O)=O)C(C)C)=O
Relative Density.1.193 g/cm3 (Predicted)
ColorWhite
AppearanceSolid
Sequence ShortDKFVG{N(Me)Leu}{Nle}-NH2
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
H2O: 1 mg/mL (1.24 mM), Sonication is recommended.
Solution Preparation Table
H2O
1mg5mg10mg50mg
1 mM1.2438 mL6.2190 mL12.4380 mL62.1898 mL

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Keywords

Tachykinin receptorNK2NK receptorNeurokininreceptorNeurokinin receptorNeurokinin ReceptorInhibitorinhibit[Lys-5,MeLeu9,Nle10]-NKA(4-10)[Lys5,MeLeu9,Nle10]NKA(410)[Lys5,MeLeu9,Nle10]-NKA[Lys5,MeLeu9,Nle10] NKA(4 10)
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