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ARC 239 dihydrochloride

Catalog No. T22033 CAS 55974-42-0

ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).

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ARC 239 dihydrochloride, CAS 55974-42-0

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).

Molecular Weight	480.43
Formula	C24H31Cl2N3O3
CAS No.	55974-42-0

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Suzana Assad Kahn, et al. The anti-hypertensive drug prazosin inhibits glioblastoma growth via the PKCδ-dependent inhibition of the AKT pathway. EMBO Mol Med. 2016 May 2;8(5):511-26.

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Keywords

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