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Notum pectinacetylesterase-1
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Catalog No. T60057Cas No. 460727-10-0
Notum pectinacetylesterase-1 is a Notum Pectinacetylesterase inhibitor with IC50 < 0.025 μM.
Notum pectinacetylesterase-1
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Purity: 99.89%
Catalog No. T60057Cas No. 460727-10-0
Notum pectinacetylesterase-1 is a Notum Pectinacetylesterase inhibitor with IC50 < 0.025 μM.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $117 | - | In Stock | |
| 2 mg | $175 | - | In Stock | |
| 5 mg | $269 | - | In Stock | |
| 10 mg | $395 | - | In Stock | |
| 25 mg | $592 | - | In Stock | |
| 50 mg | $834 | - | In Stock | |
| 100 mg | $1,120 | - | In Stock | |
| 500 mg | $2,260 | - | In Stock | |
| 1 mL x 10 mM (in DMSO) | $271 | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.89%
Appearance:Solid
Color:Yellow
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Product Introduction
Notum pectinacetylesterase-1 AI Summary
Notum pectinacetylesterase-1 exhibits multiple bioactivities across various biological targets. It is a potent IMPase inhibitor with a potency of 28183.8 nM. The compound acts as an antagonist of the Neuropeptide S receptor affecting cAMP signal transduction with a potency of 25118.9 nM, while also serving as an agonist of the Relaxin receptor RXFP1 with the same potency of 25118.9 nM. Notably, it inhibits delayed death in malarial parasite plastids after 96-hour incubation with a potency of 13115.4 nM and shows inhibitory activity against Polymerase Iota with a potency of 89125.1 nM. Furthermore, Notum pectinacetylesterase-1 is an effective inhibitor of Lassa Virus binding or entry into cells with a potency of 316.2 nM and inhibits the HIV-1 protein Vpr with a potency of 12589.3 nM..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | Notum pectinacetylesterase-1 is a Notum Pectinacetylesterase inhibitor with IC50 < 0.025 μM. |
| Molecular Weight | 334.42 |
| Formula | C14H14N4O2S2 |
| Cas No. | 460727-10-0 |
| Smiles | S(CC(NC=1C=C(C)ON1)=O)C2=C3C(SC(C)=C3C)=NC=N2 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | ||||||||||||||||||||
| Solubility Information | DMSO: 3.35 mg/mL (10.02 mM), Sonication is recommended.  | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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Calculator
In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:
For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, and a total of 10 animals are to be administered, using a formulation of 
10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH2O , the resulting working solution concentration would be 2 mg/mL.Stock Solution Preparation:
Dissolve 2 mg of the compound in 100 μL DMSO to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.
Preparation of the In Vivo Formulation:
1) Add 100 μL of the DMSO stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.
2) Add 50 μL Tween 80 and mix well until fully clarified.
3) Add 450 μL Saline,PBS or ddH2O and mix thoroughly until a homogeneous solution is obtained.
This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.
Dose Conversion
You can also refer to dose conversion for different animals. More Dose Conversion
Tech Support
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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