Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Nicotelline, also known as Nicotellin, is an alkaloid associated with nicotine and acts as a modest inhibitor of the enzyme human cDNA-expressed cytochrome P-450 2A6 (CYP2A6), which is responsible for coumarin 7-hydroxylation. However, Nicotelline does not show inhibitory effects at a concentration of 300 μM. It serves as a tracer and biomarker for particulate matter (PM) originating from tobacco smoke [1] [2].
Pack Size | Availability | Price/USD | Quantity |
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2 mg | 5 days | $ 41.00 |
Description | Nicotelline, also known as Nicotellin, is an alkaloid associated with nicotine and acts as a modest inhibitor of the enzyme human cDNA-expressed cytochrome P-450 2A6 (CYP2A6), which is responsible for coumarin 7-hydroxylation. However, Nicotelline does not show inhibitory effects at a concentration of 300 μM. It serves as a tracer and biomarker for particulate matter (PM) originating from tobacco smoke [1] [2]. |
Targets&IC50 | CYP26:≥300 μM (Ki) |
Synonyms | Nicotellin |
Molecular Weight | 233.27 |
Formula | C15H11N3 |
CAS No. | 494-04-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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Nicotelline 494-04-2 Nicotellin inhibitor inhibit