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AP-III-a4 hydrochloride

Name: AP-III-a4 hydrochloride
Brand: TargetMol
SKU: T6759L
Rating: 4.5 (1 reviews)

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Catalog No. T6759LCas No. 2070014-95-6

Alias ENOblock hydrochloride, AP-III-a4 hydrochloride (1177827-73-4 free base)

AP-III-a4 hydrochloride (ENOblock hydrochloride) is a direct enolase (enolase) inhibitor with non-substrate analogs.AP-III-a4 hydrochloride inhibits metastasis of cancer cells in vivo and affects glucose homeostasis and can be used in bioassays.

AP-III-a4 hydrochloride

😃Good

Catalog No. T6759LAlias ENOblock hydrochloride, AP-III-a4 hydrochloride (1177827-73-4 free base)Cas No. 2070014-95-6

Pack Size	Price	Availability
2 mg	$98	Backorder
5 mg	$188	Backorder
10 mg	$302	Backorder
25 mg	$619	Backorder
50 mg	$873	Backorder
100 mg	Inquiry	Backorder
200 mg	Inquiry	Backorder
1 mL x 10 mM (in DMSO)	$260	Backorder

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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Product Introduction

Bioactivity

Description	AP-III-a4 hydrochloride (ENOblock hydrochloride) is a direct enolase (enolase) inhibitor with non-substrate analogs.AP-III-a4 hydrochloride inhibits metastasis of cancer cells in vivo and affects glucose homeostasis and can be used in bioassays.
Alias	ENOblock hydrochloride, AP-III-a4 hydrochloride (1177827-73-4 free base)

Chemical Properties

Molecular Weight	631.18
Formula	C₃₁H₄₄ClFN₈O₃
Cas No.	2070014-95-6
Smiles	O=C(CC1=CC=C(NC2=NC(NCC3CCCCC3)=NC(NCC4=CC=C(C=C4)F)=N2)C=C1)NCCOCCOCCN.Cl
Relative Density.	no data available

Storage & Solubility Information

Storage

keep away from direct sunlight | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 40 mg/mL (63.37 mM), Sonication is recommended.

H2O: 8 mg/mL (12.67 mM), Sonication is recommended.

Solution Preparation Table

H2O/DMSO

	1mg	5mg	10mg	50mg
1 mM	1.5843 mL	7.9217 mL	15.8433 mL	79.2167 mL
5 mM	0.3169 mL	1.5843 mL	3.1687 mL	15.8433 mL
10 mM	0.1584 mL	0.7922 mL	1.5843 mL	7.9217 mL

DMSO

	1mg	5mg	10mg	50mg
20 mM	0.0792 mL	0.3961 mL	0.7922 mL	3.9608 mL
50 mM	0.0317 mL	0.1584 mL	0.3169 mL	1.5843 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc