Powder: -20°C for 3 years | In solvent: -80°C for 1 year
A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 52.00 | |
5 mg | In stock | $ 97.00 | |
10 mg | In stock | $ 155.00 | |
25 mg | In stock | $ 326.00 | |
50 mg | In stock | $ 497.00 | |
100 mg | In stock | $ 738.00 | |
500 mg | In stock | $ 1,550.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 65.00 |
Description | A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. |
Targets&IC50 | adenosine A2Areceptor:4 nM (Ki), A1receptor:264 nM (Ki) |
In vitro | A2A receptor anyagonist 1 is a potent adenosine A2A receptor antagonist, selective over the A1 receptor and demonstrate its binding activity with Ki values of 4 and 264 nM, respectively. [1] |
Synonyms | CPI-444 analog, A2A receptor antagonist 1 |
Molecular Weight | 309.3 |
Formula | C16H12FN5O |
CAS No. | 443103-97-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 20 mg/mL (64.66 mM), sonification is recommended.
You can also refer to dose conversion for different animals. More
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