Powder: -20°C for 3 years | In solvent: -80°C for 1 year
NSD2-IN-1 (compound 38) serves as a potent and highly selective inhibitor of NSD2-PWWP1 (nuclear receptor-binding SET domain 2-PWWP1), demonstrating an IC50 value of 0.11 μM. By binding to NSD2-PWWP1, NSD2-IN-1 impacts the expression of genes under NSD2 regulation, leading to apoptosis and cell cycle arrest [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 10-14 weeks | $ 1,520.00 | |
50 mg | 10-14 weeks | $ 1,980.00 | |
100 mg | 10-14 weeks | $ 2,500.00 |
Description | NSD2-IN-1 (compound 38) serves as a potent and highly selective inhibitor of NSD2-PWWP1 (nuclear receptor-binding SET domain 2-PWWP1), demonstrating an IC50 value of 0.11 μM. By binding to NSD2-PWWP1, NSD2-IN-1 impacts the expression of genes under NSD2 regulation, leading to apoptosis and cell cycle arrest [1]. |
Molecular Weight | 449.59 |
Formula | C29H31N5 |
CAS No. | 2797183-37-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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NSD2-IN-1 2797183-37-8 inhibitor inhibit