Powder: -20°C for 3 years | In solvent: -80°C for 1 year
IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | In stock | $ 51.00 | |
10 mg | In stock | $ 84.00 | |
25 mg | In stock | $ 172.00 | |
50 mg | In stock | $ 278.00 | |
100 mg | In stock | $ 452.00 |
Description | IK-930 is an orally active TEAD inhibitor (EC50 < 0.1 µM) with potent potency. |
Targets&IC50 | TEAD:<0.1 µM(EC50) |
In vitro | IK-930 (0-1 μM) is a potent and selective TEAD inhibitor.[2] |
In vivo | IK-930 (compound I-32) (10 mg/kg; p.o.) exhibits favorable pharmacokinetic parameters in BALB/c mice with Cmax of 1088 ng/mL and AUC 0-last of 4581 ng*h /mL.[1] |
Synonyms | compound I-32 |
Molecular Weight | 424.44 |
Formula | C19H19F3N4O2S |
CAS No. | 2563892-44-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 90.0 mg/mL (212.0 mM), Sonication and heating to 60℃ are recommended.
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
IK-930 2563892-44-2 Stem Cells YAP compound I-32 IK 930 IK930 inhibitor inhibit