Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Eleven-Nineteen-Leukemia Protein IN-1 is a potent inhibitor of the ENL YEATS domain, exhibiting an IC50 of 14.5 nM. It binds to the ENL protein, consequently increasing its thermal stability in vitro [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | Eleven-Nineteen-Leukemia Protein IN-1 is a potent inhibitor of the ENL YEATS domain, exhibiting an IC50 of 14.5 nM. It binds to the ENL protein, consequently increasing its thermal stability in vitro [1]. |
Targets&IC50 | Eleven-Nineteen-Leukemia YEATS domain:14.5 nM |
In vitro | The Eleven-Nineteen-Leukemia Protein IN-1 (compound 13) exhibits inhibitory effects on MOLM-13 and MV4-11 cells, with IC50 values of 39.6 µM and 45.1 µM respectively [1]. |
Molecular Weight | 487.6 |
Formula | C27H33N7O2 |
CAS No. | 2894121-68-5 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Eleven-Nineteen-Leukemia Protein IN-1 2894121-68-5 Chromatin/Epigenetic Epigenetic Reader Domain inhibitor inhibit