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Quinaprilat
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Catalog No. T21049Cas No. 82768-85-2
Alias CI-928, CI928, CI 928
Quinaprilat is an orally active ACE inhibitor, the active metabolite of quinapril, and a substrate for OAT3. It blocks the conversion of angiotensin I to angiotensin II, exhibiting antihypertensive activity.
Quinaprilat
🥰Excellent
Catalog No. T21049Alias CI-928, CI928, CI 928Cas No. 82768-85-2
Quinaprilat is an orally active ACE inhibitor, the active metabolite of quinapril, and a substrate for OAT3. It blocks the conversion of angiotensin I to angiotensin II, exhibiting antihypertensive activity.
| Pack Size | Price | USA Warehouse | Global Warehouse | Quantity |
|---|---|---|---|---|
| 1 mg | $71 | - | In Stock | |
| 5 mg | Preferential | - | In Stock |
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Product Introduction
Bioactivity
Chemical Properties
| Description | Quinaprilat is an orally active ACE inhibitor, the active metabolite of quinapril, and a substrate for OAT3. It blocks the conversion of angiotensin I to angiotensin II, exhibiting antihypertensive activity. |
| In vitro | Quinaprilat (5μM) promotes its own active renal secretion by mediating the interaction with hOAT3, increasing the uptake by HEK293 cells to 25 times the original level, with a Km value of 13.4μM for its binding [1]. Quinaprilat (100 nM, 20 minutes) can activate the B1 receptor, thereby inhibiting PKC activity and leading to NO release from HLMVE cells [2]. |
| In vivo | Quinaprilat (3 mg/kg, once daily for 6 days) was administered via oral gavage and demonstrated certain antihypertensive effects in male SHR rats when used in combination with other medications [1]. |
| Synonyms | CI-928, CI928, CI 928 |
| Molecular Weight | 410.46 |
| Formula | C23H26N2O5 |
| Cas No. | 82768-85-2 |
| Smiles | C([C@@H](N[C@@H](CCC1=CC=CC=C1)C(O)=O)C)(=O)N2[C@H](C(O)=O)CC=3C(C2)=CC=CC3 |
| Relative Density. | 1.289 g/cm3 |
| Color | White |
| Appearance | Solid |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | DMSO: Soluble, Sonication is recommended. |
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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