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Atopaxar Hydrobromide
🥰Excellent
Catalog No. T1986LCas No. 474550-69-1
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome.
Atopaxar Hydrobromide
🥰Excellent
Catalog No. T1986LCas No. 474550-69-1
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $257 | In Stock | |
| 2 mg | $378 | In Stock | |
| 5 mg | $639 | In Stock | |
| 10 mg | $890 | In Stock | |
| 25 mg | $1,370 | In Stock | |
| 50 mg | $1,780 | In Stock |
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Product Introduction
Bioactivity
Chemical Properties
| Description | Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Artery Disease and Acute Coronary Syndrome. |
| Molecular Weight | 608.54 |
| Formula | C29H39BrFN3O5 |
| Cas No. | 474550-69-1 |
| Relative Density. | no data available |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||
| Solubility Information | DMSO: 10 mM, Sonication is recommended. | ||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||
DMSO
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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