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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3404 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence. Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Autophagy
Autophagy
Apoptosis
Apoptosis
Apoptosis
Antibacterial
Antibacterial
Antibacterial
Antibiotic
Antibiotic
Antibiotic
Endogenous Metabolite
Endogenous Metabolite
Endogenous Metabolite
5-HT Receptor
5-HT Receptor
5-HT Receptor
Adrenergic Receptor
Adrenergic Receptor
Adrenergic Receptor
DNA/RNA Synthesis
DNA/RNA Synthesis
DNA/RNA Synthesis
HIV Protease
HIV Protease
HIV Protease
AChR
AChR
AChR
Dopamine Receptor
Dopamine Receptor
Dopamine Receptor
COX
COX
COX
VEGFR
VEGFR
VEGFR
Histamine Receptor
Histamine Receptor
Histamine Receptor
Parasite
Parasite
Parasite
Sodium Channel
Sodium Channel
Sodium Channel
Calcium Channel
EGFR
Calcium Channel
EGFR
Calcium Channel
EGFR
PI3K
PI3K
PI3K
Antifungal
Antifungal
Antifungal
Potassium Channel
Potassium Channel
Potassium Channel
PDE
PDE
PDE
FLT
FLT
FLT
Topoisomerase
Topoisomerase
Topoisomerase
CDK
HCV Protease
CDK
HCV Protease
CDK
HCV Protease
P450
PDGFR
P450
PDGFR
PDGFR
P450
c-Kit
JAK
c-Kit
JAK
c-Kit
JAK
Dehydrogenase
Dehydrogenase
Dehydrogenase
FGFR
PPAR
Microtubule Associated
Reactive Oxygen Species
FGFR
Microtubule Associated
PPAR
Reactive Oxygen Species
FGFR
Microtubule Associated
Reactive Oxygen Species
PPAR
SARS-CoV
SARS-CoV
SARS-CoV
HDAC
Ferroptosis
Ferroptosis
HDAC
HDAC
Ferroptosis
Glucocorticoid Receptor
mTOR
Glucocorticoid Receptor
mTOR
Glucocorticoid Receptor
mTOR
c-Met/HGFR
Influenza Virus
c-Met/HGFR
Influenza Virus
c-Met/HGFR
Influenza Virus
Estrogen/progestogen Receptor
Estrogen/progestogen Receptor
Estrogen/progestogen Receptor
NF-κB
Src
Mitophagy
NF-κB
Mitophagy
Src
NF-κB
Mitophagy
Src
Prostaglandin Receptor
RAAS
Prostaglandin Receptor
RAAS
Prostaglandin Receptor
RAAS
HBV
Nucleoside Antimetabolite/Analog
GABA Receptor
GABA Receptor
HBV
Nucleoside Antimetabolite/Analog
HBV
GABA Receptor
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
Reverse Transcriptase
Reverse Transcriptase
GPR
Tyrosine Kinases
GPR
Tyrosine Kinases
GPR
Tyrosine Kinases
Adenosine Receptor
Adenosine Receptor
Adenosine Receptor
ADC Cytotoxin
Raf
Bcr-Abl
ADC Cytotoxin
Bcr-Abl
Raf
ADC Cytotoxin
Bcr-Abl
Raf
BTK
Proteasome
BTK
Proteasome
BTK
Proteasome
Androgen Receptor
Androgen Receptor
Androgen Receptor
Akt
PARP
Serotonin Transporter
iGluR
Akt
iGluR
PARP
Serotonin Transporter
Akt
iGluR
PARP
Serotonin Transporter
Epigenetic Reader Domain
Aurora Kinase
HER
Virus Protease
Aurora Kinase
Epigenetic Reader Domain
HER
Virus Protease
Aurora Kinase
Epigenetic Reader Domain
HER
Virus Protease
HSV
MEK
ROS
HSV
MEK
ROS
ROS
HSV
MEK
GluR
Transferase
Norepinephrine
Progesterone Receptor
Estrogen Receptor/ERR
p38 MAPK
Estrogen Receptor/ERR
Norepinephrine
GluR
Progesterone Receptor
p38 MAPK
Transferase
GluR
Estrogen Receptor/ERR
p38 MAPK
Transferase
Norepinephrine
Progesterone Receptor
HSP
Phosphatase
IL Receptor
IL Receptor
HSP
Phosphatase
HSP
Phosphatase
IL Receptor
HIF/HIF Prolyl-Hydroxylase
ALK
NMDAR
Beta Amyloid
c-RET
Opioid Receptor
TNF
ALK
Beta Amyloid
c-RET
HIF/HIF Prolyl-Hydroxylase
Opioid Receptor
NMDAR
TNF
ALK
Beta Amyloid
c-RET
HIF/HIF Prolyl-Hydroxylase
NMDAR
TNF
Opioid Receptor
Antifection
P-gp
ERK
DPP-4
Trk receptor
Antifection
ERK
DPP-4
P-gp
Trk receptor
Antifection
ERK
DPP-4
P-gp
Trk receptor
Antioxidant
Carbonic Anhydrase
ribosome
ATPase
TRP/TRPV Channel
Antioxidant
Carbonic Anhydrase
ATPase
ribosome
TRP/TRPV Channel
Antioxidant
ATPase
Carbonic Anhydrase
ribosome
TRP/TRPV Channel
GSK-3
AChE
c-Fms
PKC
DNA Alkylator/Crosslinker
Thrombin
AChE
c-Fms
DNA Alkylator/Crosslinker
GSK-3
PKC
Thrombin
AChE
c-Fms
DNA Alkylator/Crosslinker
GSK-3
PKC
Thrombin
Antiviral
Endothelin Receptor
Gamma-secretase
Proton pump
CXCR
Interleukin
TLR
Retinoid Receptor
Mitochondrial Metabolism
TAM Receptor
Antiviral
CXCR
Gamma-secretase
Endothelin Receptor
Interleukin
Mitochondrial Metabolism
Retinoid Receptor
Proton pump
TAM Receptor
TLR
Antiviral
CXCR
Endothelin Receptor
Interleukin
Mitochondrial Metabolism
Proton pump
TLR
TAM Receptor
Gamma-secretase
Retinoid Receptor
Chk
E1/E2/E3 Enzyme
MMP
CCR
DNA-PK
BCL
STAT
AMPK
Phospholipase
S1P Receptor
MAO
CCR
BCL
Chk
AMPK
DNA-PK
E1/E2/E3 Enzyme
MMP
MAO
Phospholipase
S1P Receptor
STAT
AMPK
CCR
BCL
Chk
DNA-PK
MAO
MMP
Phospholipase
S1P Receptor
STAT
E1/E2/E3 Enzyme
Histone Methyltransferase
HIF
Caspase
Syk
NO Synthase
SGLT
LPL Receptor
Thyroid hormone receptor(THR)
Caspase
Histone Methyltransferase
HIF
NO Synthase
LPL Receptor
Syk
SGLT
Thyroid hormone receptor(THR)
Caspase
Histone Methyltransferase
HIF
LPL Receptor
NO Synthase
SGLT
Thyroid hormone receptor(THR)
Syk
CFTR
Antifolate
Guanylate cyclase
p53
DNA Alkylation
Antifolate
CFTR
Guanylate cyclase
DNA Alkylation
p53
Antifolate
CFTR
DNA Alkylation
Guanylate cyclase
p53
CSF-1R
Nrf2
Hedgehog/Smoothened
Integrin
IGF-1R
NADPH
CSF-1R
Hedgehog/Smoothened
Integrin
IGF-1R
Nrf2
NADPH
CSF-1R
Hedgehog/Smoothened
Integrin
Nrf2
IGF-1R
NADPH
Cannabinoid Receptor
FAK
Glutathione Peroxidase
HMG-CoA Reductase
Monoamine Oxidase
P2X Receptor
Lipoxygenase
MRP
PKA
Hydroxylase
S6 Kinase
CETP
TGF-beta/Smad
PLK
Wnt/beta-catenin
Cannabinoid Receptor
CETP
FAK
Hydroxylase
Glutathione Peroxidase
Lipoxygenase
HMG-CoA Reductase
MRP
S6 Kinase
Monoamine Oxidase
PKA
P2X Receptor
PLK
Wnt/beta-catenin
TGF-beta/Smad
Cannabinoid Receptor
FAK
CETP
Glutathione Peroxidase
Lipoxygenase
HMG-CoA Reductase
MRP
Monoamine Oxidase
PKA
P2X Receptor
TGF-beta/Smad
PLK
Wnt/beta-catenin
Hydroxylase
S6 Kinase
ATM/ATR
DHFR
Drug Metabolite
Indoleamine 2,3-Dioxygenase (IDO)
Neurokinin receptor
Sirtuin
Glucosidase
IAP
JNK
Kras
Mdm2
ROCK
ROS Kinase
P2Y Receptor
Vasopressin Receptor
Reductase
ATM/ATR
DHFR
Drug Metabolite
Glucosidase
IAP
JNK
Indoleamine 2,3-Dioxygenase (IDO)
Kras
Mdm2
Neurokinin receptor
ROS Kinase
ROCK
Sirtuin
P2Y Receptor
Vasopressin Receptor
Reductase
ATM/ATR
DHFR
Drug Metabolite
Glucosidase
Indoleamine 2,3-Dioxygenase (IDO)
IAP
JNK
Kras
Neurokinin receptor
Mdm2
ROCK
P2Y Receptor
ROS Kinase
Reductase
Vasopressin Receptor
Sirtuin
Casein Kinase
Aminopeptidase
FXR
Aryl Hydrocarbon Receptor
Histone Demethylase
Kinesin
DNA Methyltransferase
RSV
CAT
OX Receptor
RIP kinase
Smo
Beta-Secretase
Sigma receptor
GNRH Receptor
Serine Protease
Xanthine Oxidase
Aryl Hydrocarbon Receptor
Casein Kinase
CAT
DNA Methyltransferase
Beta-Secretase
Aminopeptidase
FXR
Histone Demethylase
Kinesin
GNRH Receptor
OX Receptor
Sigma receptor
RIP kinase
Smo
Serine Protease
Xanthine Oxidase
RSV
Aryl Hydrocarbon Receptor
Casein Kinase
Aminopeptidase
CAT
Beta-Secretase
DNA Methyltransferase
FXR
Histone Demethylase
GNRH Receptor
Kinesin
OX Receptor
RSV
RIP kinase
Smo
Serine Protease
Sigma receptor
Xanthine Oxidase
Amino Acids and Derivatives
Bradykinin Receptor
DNA
Glucokinase
Glucagon Receptor
AhR
BACE
Pim
Ligand for E3 Ligase
PAK
Isocitrate Dehydrogenase (IDH)
ROR
IRAK
IκB/IKK
AhR
Amino Acids and Derivatives
Bradykinin Receptor
BACE
DNA
Glucokinase
Glucagon Receptor
Isocitrate Dehydrogenase (IDH)
Ligand for E3 Ligase
PAK
IRAK
IκB/IKK
ROR
Pim
Amino Acids and Derivatives
AhR
Bradykinin Receptor
BACE
DNA
Glucokinase
Glucagon Receptor
Ligand for E3 Ligase
IRAK
IκB/IKK
Isocitrate Dehydrogenase (IDH)
Pim
ROR
PAK
Factor Xa
Complement System
Fatty Acid Synthase
IDO
Ephrin Receptor
Leukotriene Receptor
Tie-2
Acyltransferase
DNA gyrase
Acyltransferase
Ephrin Receptor
Factor Xa
Fatty Acid Synthase
DNA gyrase
Complement System
Leukotriene Receptor
IDO
Tie-2
Acyltransferase
Factor Xa
Complement System
Ephrin Receptor
DNA gyrase
Fatty Acid Synthase
Leukotriene Receptor
IDO
Tie-2
Chloride channel
Decarboxylase
CGRP Receptor
Acetyl-CoA Carboxylase
cholecystokinin
LTR
Molecular Glues
NADPH-oxidase
CaMK
CRFR
DprE1
GHSR
Liver X Receptor
Melatonin Receptor
Neprilysin
Ras
Gap Junction Protein
IFNAR
MT Receptor
FAAH
PGE Synthase
KSP
Monoamine Transporter
NOS
Wee1
Acetyl-CoA Carboxylase
CaMK
CGRP Receptor
cholecystokinin
CRFR
DprE1
Gap Junction Protein
GHSR
FAAH
IFNAR
Chloride channel
Decarboxylase
Liver X Receptor
Melatonin Receptor
MT Receptor
LTR
Neprilysin
PGE Synthase
Ras
Molecular Glues
NADPH-oxidase
KSP
Monoamine Transporter
NOS
Wee1
Acetyl-CoA Carboxylase
CaMK
CRFR
CGRP Receptor
cholecystokinin
Chloride channel
Decarboxylase
DprE1
FAAH
Gap Junction Protein
GHSR
Liver X Receptor
Melatonin Receptor
IFNAR
LTR
KSP
MT Receptor
Molecular Glues
NADPH-oxidase
Monoamine Transporter
NOS
PGE Synthase
Wee1
Neprilysin
Ras
Annexin A
CRM1
DUB
GlyT
ABC
Arginase
CaSR
Free radical scavengers
LPA Receptor
Adenosine deaminase
Cell wall
Myosin
PDK
Telomerase
Imidazoline Receptor
Tyrosinase
PD-1/PD-L1
NAMPT
NOD-like Receptor (NLR)
OAT
Cysteine Protease
Protease-activated Receptor
Rho
STING
YAP
PERK
GPCR19
Melanocortin Receptor
Neuropeptide Y Receptor
Serine/threonin kinase
Somatostatin
Adenosine deaminase
ABC
Arginase
Cell wall
CaSR
Free radical scavengers
Cysteine Protease
Annexin A
CRM1
Imidazoline Receptor
NAMPT
LPA Receptor
PD-1/PD-L1
GPCR19
DUB
NOD-like Receptor (NLR)
OAT
PERK
Melanocortin Receptor
Rho
Neuropeptide Y Receptor
Protease-activated Receptor
GlyT
STING
YAP
Tyrosinase
Serine/threonin kinase
Somatostatin
Myosin
PDK
Telomerase
Adenosine deaminase
ABC
Arginase
Annexin A
Cell wall
CaSR
CRM1
DUB
Cysteine Protease
Imidazoline Receptor
GPCR19
GlyT
LPA Receptor
Melanocortin Receptor
NAMPT
Rho
Neuropeptide Y Receptor
Myosin
PDK
NOD-like Receptor (NLR)
OAT
PERK
STING
YAP
Protease-activated Receptor
Serine/threonin kinase
Somatostatin
Telomerase
Tyrosinase
Free radical scavengers
PD-1/PD-L1
Galectin
Hexokinase
CD73
GST
ATP Citrate Lyase
Drug-Linker Conjugates for ADC
Epoxide Hydrolase
p97
Porcupine
PYK2
Discoidin Domain Receptor (DDR)
BCRP
IRE1
LDL
MLK
Oxytocin Receptor
Integrase
Ligands for Target Protein for PROTAC
MAPK
Na-K-Cl cotransporter
NEDD8
PAI-1
PROTACs
UGT
Stearoyl-CoA Desaturase (SCD)
transporter
VDA
Lipid
Taste receptor
ATP Citrate Lyase
BCRP
CD73
Discoidin Domain Receptor (DDR)
Drug-Linker Conjugates for ADC
Epoxide Hydrolase
Galectin
Integrase
GST
IRE1
LDL
MLK
Ligands for Target Protein for PROTAC
MAPK
Oxytocin Receptor
Na-K-Cl cotransporter
NEDD8
Lipid
PAI-1
p97
Porcupine
Stearoyl-CoA Desaturase (SCD)
transporter
VDA
PROTACs
Hexokinase
PYK2
Taste receptor
UGT
ATP Citrate Lyase
BCRP
CD73
Galectin
Discoidin Domain Receptor (DDR)
GST
Hexokinase
Integrase
Lipid
Ligands for Target Protein for PROTAC
MAPK
Na-K-Cl cotransporter
NEDD8
p97
Porcupine
UGT
PAI-1
PROTACs
PYK2
Stearoyl-CoA Desaturase (SCD)
transporter
VDA
Taste receptor
Drug-Linker Conjugates for ADC
Epoxide Hydrolase
IRE1
LDL
MLK
Oxytocin Receptor
ACK
Arrestin
Glutaminase
c-Myc
Anti-infection
Aromatase
advanced glycation end products
Aquaporin
DYRK
MNK
MTH1
PI4K
PKM
Adenylyl cyclase
Anion Exchanger
BMI-1
Fas/FasL
RAR/RXR 
AAK1 (AP2 associated kinase 1)
GSNOR
TOPK
Vitamin
Hydrogenase
Monocarboxylate transporter
PAFR
MALT
GTPase
KLF
Lipase
MELK
Methionine Adenosyltransferase (MAT)
Motilin Receptor
ASK
CRISPR/Cas9
FLAP
GluCls
Hck
Hippo pathway
Histone Acetyltransferase
N-Acetylglucosaminyltransferase
NOD
NPC1L1
Pyroptosis
Survivin
Phosphorylase
PROTAC Linker
GRK
HCN Channel
SGK
Stemness kinase
Thioredoxin
VDAC
Adenylyl cyclase
Anion Exchanger
advanced glycation end products
Aquaporin
ACK
Arrestin
AAK1 (AP2 associated kinase 1)
Anti-infection
BMI-1
Aromatase
ASK
DYRK
CRISPR/Cas9
Fas/FasL
GTPase
GSNOR
Hck
Hippo pathway
Histone Acetyltransferase
FLAP
Glutaminase
Hydrogenase
c-Myc
MALT
KLF
Lipase
MELK
Methionine Adenosyltransferase (MAT)
Motilin Receptor
GluCls
GRK
HCN Channel
N-Acetylglucosaminyltransferase
NOD
NPC1L1
Monocarboxylate transporter
PAFR
MNK
MTH1
Phosphorylase
PROTAC Linker
PI4K
PKM
Pyroptosis
SGK
Survivin
Stemness kinase
Thioredoxin
VDAC
RAR/RXR 
TOPK
Vitamin
Anti-infection
Adenylyl cyclase
Anion Exchanger
ACK
Arrestin
advanced glycation end products
Aquaporin
AAK1 (AP2 associated kinase 1)
ASK
BMI-1
Aromatase
Glutaminase
c-Myc
Hydrogenase
CRISPR/Cas9
Fas/FasL
GTPase
GSNOR
Hck
Hippo pathway
Histone Acetyltransferase
FLAP
GluCls
GRK
HCN Channel
KLF
Monocarboxylate transporter
PAFR
Lipase
MELK
Methionine Adenosyltransferase (MAT)
Motilin Receptor
MNK
MTH1
Phosphorylase
N-Acetylglucosaminyltransferase
NOD
NPC1L1
PI4K
PKM
Survivin
RAR/RXR 
PROTAC Linker
Stemness kinase
TOPK
Vitamin
Pyroptosis
SGK
Thioredoxin
VDAC
DYRK
MALT
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