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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3550 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3550 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
Antibiotic
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Parasite
Dopamine Receptor
HIV Protease
AChR
VEGFR
COX
Potassium Channel
Histamine Receptor
Sodium Channel
Calcium Channel
EGFR
PI3K
PDE
Reactive Oxygen Species
Antifungal
Cytochromes P450
Topoisomerase
CDK
Virus Protease
SARS-CoV
FLT
HCV Protease
PDGFR
NF-κB
Dehydrogenase
PPAR
FGFR
JAK
Microtubule Associated
c-Kit
Ferroptosis
c-Met/HGFR
Glucocorticoid Receptor
mTOR
Influenza Virus
HDAC
HBV
Nucleoside Antimetabolite/Analog
iGluR
GABA Receptor
Src
Mitophagy
Reverse Transcriptase
Estrogen/progestogen Receptor
Prostaglandin Receptor
RAAS
Tyrosine Kinases
Akt
GPCR
p38 MAPK
Adenosine Receptor
Androgen Receptor
Interleukin
TNF
Serotonin Transporter
Caspase
Bcr-Abl
Bcl-2 Family
Raf
HSV
Epigenetic Reader Domain
Ras
Proteasome
Phosphatase
NMDAR
GluR
Beta Amyloid
PARP
TRP/TRPV Channel
ERK
Transferase
Estrogen Receptor/ERR
ROS
HSP
Cholinesterase (ChE)
MMP
Aurora Kinase
HIF/HIF Prolyl-Hydroxylase
ATPase
Norepinephrine
Progesterone Receptor
Mitochondrial Metabolism
Opioid Receptor
IL Receptor
P-gp
ALK
MEK
MDM-2/p53
Antiviral
TLR
c-Fms
c-RET
NO Synthase
Histone Methyltransferase
Antioxidant
Antifection
DPP-4
Trk receptor
HER
Carbonic Anhydrase
PKC
STAT
ribosome
AMPK
Proton pump
LPL Receptor
MAO
E1/E2/E3 Enzyme
CXCR
Endothelin Receptor
Retinoid Receptor
DNA Alkylator/Crosslinker
GSK-3
Wnt/beta-catenin
Gamma-secretase
CCR
Chk
Phospholipase
TAM Receptor
S1P Receptor
Thyroid hormone receptor(THR)
Drug Metabolite
Angiotensin-converting Enzyme (ACE)
IGF-1R
Nrf2
Syk
CFTR
p53
DNA-PK
Integrin
JNK
Antifolate
SGLT
HIF
Thrombin
FAK
ROS Kinase
Monoamine Oxidase
Reductase
NADPH
Serine Protease
Molecular Glues
Guanylate cyclase
Lipoxygenase
Hydroxylase
Neurokinin receptor
Anti-infection
S6 Kinase
Kras
P2Y Receptor
PKA
ROCK
CSF-1R
P2X Receptor
BTK
Hedgehog/Smoothened
DNA Alkylation
OX Receptor
TGF-beta/Smad
ATM/ATR
PLK
DHFR
Glutathione Peroxidase
MRP
Leukotriene Receptor
FXR
IDO
IAP
Glucosidase
Vasopressin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
RSV
IκB/IKK
Cannabinoid Receptor
HMG-CoA Reductase
ADC Cytotoxin
Mdm2
GNRH Receptor
Aryl Hydrocarbon Receptor
Isocitrate Dehydrogenase (IDH)
Xanthine Oxidase
Beta-Secretase
Sirtuin
Sigma receptor
Amino Acids and Derivatives
Histone Demethylase
Tie-2
Factor Xa
Pim
RIP kinase
Smo
PAK
DNA
MAPK
Aminopeptidase
Casein Kinase
Ligand for E3 Ligase
Complement System
DNA Methyltransferase
NOD-like Receptor (NLR)
Kinesin
NOS
ROR
Melatonin Receptor
Glucokinase
Glucagon Receptor
Fatty Acid Synthase
Telomerase
GHSR
IRAK
AhR
CRM1
BACE
CETP
Photosensitizer
MT Receptor
Monoamine Transporter
Bradykinin Receptor
CaMK
OAT
Acyltransferase
Ephrin Receptor
CRFR
Gap Junction Protein
PD-1/PD-L1
Chloride channel
PROTACs
MTP
DprE1
YAP
LTR
IFNAR
c-Myc
Cholecystokinin Receptor
Serine/threonin kinase
Cysteine Protease
Liver X Receptor
PYK2
Glutaminase
Myosin
UGT
DNA gyrase
GlyT
IKZF
Neuropeptide Y Receptor
FAAH
Wee1
PGE Synthase
GPCR19
Decarboxylase
Neprilysin
GST
Acetyl-CoA Carboxylase
Melanocortin Receptor
CGRP Receptor
NADPH-oxidase
Tyrosinase
ASBT
NEDD8
Arginase
Cell wall
PERK
Galectin
CaSR
Rho
NAMPT
Annexin A
ABC Transporter
Na-K-Cl cotransporter
Stearoyl-CoA Desaturase (SCD)
Somatostatin
Thrombopoietin Receptor
DUB
ATP Citrate Lyase
BCRP
OXPHOS
STING
Free radical scavengers
FKBP
LPA Receptor
PDK
Oxytocin Receptor
Adenosine Deaminase
Cuproptosis
Discoidin Domain Receptor (DDR)
NOD
Protease-activated Receptor
Imidazoline Receptor
Apelin receptor
Taste receptor
GSNOR
Ligands for Target Protein for PROTAC
DYRK
VDA
Neurotensin Receptor
IRE1
LDL
Hexokinase
Integrase
HCN Channel
Epoxide Hydrolase
KSP
Mucin
Lipid
Survivin
Porcupine
CD73
Histone Acetyltransferase
transporter
PAI-1
Pyroptosis
SGK
p97
MLK
Vitamin
Advanced Glycation End Products
Adenylyl Cyclase
MicroRNA
NPC1L1
Monocarboxylate transporter
Hydrogenase
MALT
Factor VIIa
Arrestin
Lipase
Necroptosis
MIF
TOPK
GTPase
OCT
Kisspeptin
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
Stemness kinase
NR4A
Immunology/Inflammation related
SIK
FLAP
PAFR
Fas/FasL
GRK
Phosphorylase
AAK1 (AP2 associated kinase 1)
Anion Exchanger
PROTAC Linker
MAGL
Thioredoxin
ACK1
Cadherin
Huntingtin
PSMA
MNK
ASK
GluCls
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aromatase
PI4K
KLF
CRISPR/Cas9
Aquaporin
FOXO
RXFP receptor
BMI-1
PKM
Drug-Linker Conjugates for ADC
PGC-1α
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