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TOPProduct DescriptionPackaging & StorageSupporting FilesLibrary CustomizationLibrary Composition
TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3404 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence. Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Sci Citations

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
AChR
HIV Protease
Dopamine Receptor
COX
Histamine Receptor
VEGFR
Parasite
Sodium Channel
PI3K
EGFR
Calcium Channel
Potassium Channel
Antifungal
PDE
Topoisomerase
FLT
CDK
HCV Protease
Cytochromes P450
PDGFR
Dehydrogenase
JAK
SARS-CoV
Microtubule Associated
Reactive Oxygen Species
PPAR
FGFR
c-Kit
Glucocorticoid Receptor
mTOR
Ferroptosis
HDAC
Influenza Virus
c-Met/HGFR
Src
GABA Receptor
Estrogen/progestogen Receptor
RAAS
HBV
NF-κB
Mitophagy
Prostaglandin Receptor
Reverse Transcriptase
Tyrosine Kinases
Nucleoside Antimetabolite/Analog
GPR
Adenosine Receptor
Bcr-Abl
Raf
Proteasome
Androgen Receptor
Serotonin Transporter
iGluR
Epigenetic Reader Domain
Aurora Kinase
Akt
Phosphatase
Virus Protease
TRP/TRPV Channel
ROS
HSV
Transferase
p38 MAPK
Progesterone Receptor
Estrogen Receptor/ERR
PARP
GluR
Norepinephrine
ALK
MEK
ATPase
NMDAR
Opioid Receptor
IL Receptor
HSP
Beta Amyloid
c-RET
TNF
HIF/HIF Prolyl-Hydroxylase
DPP-4
Cholinesterase (ChE)
Trk receptor
HER
Carbonic Anhydrase
Antioxidant
Antifection
P-gp
Histone Methyltransferase
GSK-3
ERK
CXCR
MMP
Antiviral
c-Fms
ribosome
DNA Alkylator/Crosslinker
PKC
Mitochondrial Metabolism
Endothelin Receptor
Chk
Interleukin
TLR
Retinoid Receptor
Thrombin
S1P Receptor
Proton pump
DNA-PK
MAO
CCR
Bcl-2 Family
Thyroid hormone receptor(THR)
LPL Receptor
E1/E2/E3 Enzyme
Gamma-secretase
SGLT
STAT
AMPK
Phospholipase
HIF
Syk
CFTR
p53
NO Synthase
Antifolate
Caspase
Guanylate cyclase
TAM Receptor
Integrin
NADPH
Wnt/beta-catenin
CSF-1R
Hedgehog/Smoothened
DNA Alkylation
IGF-1R
Nrf2
Neurokinin receptor
FAK
CETP
Glutathione Peroxidase
MRP
PKA
ROCK
P2X Receptor
Lipoxygenase
TGF-beta/Smad
Hydroxylase
PLK
Cannabinoid Receptor
Monoamine Oxidase
BTK
Mdm2
DHFR
P2Y Receptor
Reductase
GNRH Receptor
IAP
Drug Metabolite
Vasopressin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
RSV
ATM/ATR
HMG-CoA Reductase
S6 Kinase
ROS Kinase
ADC Cytotoxin
Histone Demethylase
JNK
Serine Protease
FXR
Aryl Hydrocarbon Receptor
RIP kinase
Glucosidase
Smo
OX Receptor
Xanthine Oxidase
DNA
Beta-Secretase
Aminopeptidase
Sirtuin
Casein Kinase
Sigma receptor
ROR
Amino Acids and Derivatives
BACE
Factor Xa
Pim
Glucokinase
Glucagon Receptor
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
DNA Methyltransferase
IRAK
AhR
Kinesin
Leukotriene Receptor
IDO
DNA gyrase
Fatty Acid Synthase
Acyltransferase
Ephrin Receptor
Ligand for E3 Ligase
Complement System
Chloride channel
NOS
DprE1
YAP
LTR
IFNAR
Tie-2
Melatonin Receptor
Cholecystokinin Receptor
MT Receptor
GlyT
Monoamine Transporter
Molecular Glues
Neuropeptide Y Receptor
FAAH
CaMK
Wee1
PGE Synthase
OAT
Decarboxylase
CRFR
Neprilysin
Acetyl-CoA Carboxylase
Melanocortin Receptor
GHSR
CGRP Receptor
Gap Junction Protein
NADPH-oxidase
Kras
PROTACs
CRM1
Arginase
Cell wall
CaSR
Rho
Cysteine Protease
NAMPT
PYK2
Myosin
Annexin A
ABC Transporter
Somatostatin
KSP
DUB
Telomerase
MAPK
STING
Free radical scavengers
GPCR19
LPA Receptor
PDK
Adenosine Deaminase
Ras
Tyrosinase
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
PD-1/PD-L1
Taste receptor
GSNOR
NEDD8
Ligands for Target Protein for PROTAC
PERK
VDA
Galectin
Serine/threonin kinase
Liver X Receptor
Glutaminase
IRE1
UGT
LDL
Na-K-Cl cotransporter
Hexokinase
Integrase
HCN Channel
Stearoyl-CoA Desaturase (SCD)
Epoxide Hydrolase
ATP Citrate Lyase
BCRP
Porcupine
CD73
transporter
PAI-1
GST
Oxytocin Receptor
Discoidin Domain Receptor (DDR)
p97
MLK
Advanced Glycation End Products
Adenylyl Cyclase
MicroRNA
NPC1L1
Monocarboxylate transporter
Hydrogenase
RAR/RXR
MALT
Arrestin
DYRK
Lipase
GTPase
c-Myc
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
Stemness kinase
FLAP
PAFR
Fas/FasL
GRK
Phosphorylase
Anion Exchanger
PROTAC Linker
Thioredoxin
ACK1
Lipid
PSMA
MNK
Survivin
Histone Acetyltransferase
ASK
GluCls
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aromatase
PI4K
KLF
CRISPR/Cas9
Aquaporin
RXFP receptor
SGK
Anti-infection
BMI-1
NOD
PKM
Vitamin
Drug-Linker Conjugates for ADC
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