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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3550 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3550 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Supporting Files | TargetMol Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (60.2 MB)

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
Antibiotic
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
Parasite
Dopamine Receptor
HIV Protease
AChR
VEGFR
Potassium Channel
COX
Histamine Receptor
Sodium Channel
Calcium Channel
EGFR
PI3K
PDE
Antifungal
Cytochromes P450
Reactive Oxygen Species
Topoisomerase
CDK
Virus Protease
SARS-CoV
FLT
HCV Protease
NF-κB
PDGFR
Dehydrogenase
FGFR
PPAR
Microtubule Associated
JAK
c-Kit
Ferroptosis
Influenza Virus
Glucocorticoid Receptor
mTOR
HDAC
c-Met/HGFR
HBV
Nucleoside Antimetabolite/Analog
iGluR
GABA Receptor
Estrogen/progestogen Receptor
Src
Mitophagy
Reverse Transcriptase
Prostaglandin Receptor
Tyrosine Kinases
RAAS
Akt
p38 MAPK
GPCR
Adenosine Receptor
Androgen Receptor
Interleukin
TNF
Caspase
Bcr-Abl
Serotonin Transporter
Bcl-2 Family
Raf
HSV
Epigenetic Reader Domain
Ras
NMDAR
Phosphatase
Proteasome
Beta Amyloid
GluR
TRP/TRPV Channel
Estrogen Receptor/ERR
PARP
ERK
ROS
Transferase
HSP
Aurora Kinase
MMP
HIF/HIF Prolyl-Hydroxylase
Cholinesterase (ChE)
Norepinephrine
ATPase
Mitochondrial Metabolism
IL Receptor
Opioid Receptor
P-gp
MEK
Progesterone Receptor
ALK
MDM-2/p53
c-Fms
TLR
NO Synthase
Antiviral
c-RET
Histone Methyltransferase
Antifection
DPP-4
Trk receptor
Antioxidant
HER
PKC
STAT
Carbonic Anhydrase
ribosome
AMPK
LPL Receptor
Proton pump
CXCR
Retinoid Receptor
E1/E2/E3 Enzyme
Endothelin Receptor
MAO
Gamma-secretase
Chk
S1P Receptor
DNA Alkylator/Crosslinker
Wnt/beta-catenin
CCR
GSK-3
Phospholipase
TAM Receptor
Drug Metabolite
Syk
Nrf2
p53
Thrombin
IGF-1R
CFTR
Thyroid hormone receptor(THR)
Antifolate
FAK
Angiotensin-converting Enzyme (ACE)
SGLT
Monoamine Oxidase
DNA-PK
JNK
HIF
ROS Kinase
Serine Protease
Guanylate cyclase
NADPH
Molecular Glues
Anti-infection
S6 Kinase
Hydroxylase
Integrin
Neurokinin receptor
Lipoxygenase
KRas
P2X Receptor
OX Receptor
P2Y Receptor
PLK
ROCK
PKA
CSF-1R
Hedgehog/Smoothened
DNA Alkylation
TGF-beta/Smad
ATM/ATR
BTK
MRP
Indoleamine 2,3-Dioxygenase (IDO)
HMG-CoA Reductase
RSV
Glutathione Peroxidase
Leukotriene Receptor
FXR
Cannabinoid Receptor
IDO
IAP
DHFR
Reductase
Glucosidase
IκB/IKK
Vasopressin Receptor
ADC Cytotoxin
Kinesin
Aryl Hydrocarbon Receptor
Xanthine Oxidase
Sirtuin
Sigma receptor
Beta-Secretase
Mdm2
GNRH Receptor
Isocitrate Dehydrogenase (IDH)
RIP kinase
Aminopeptidase
Amino Acids and Derivatives
MAPK
Complement System
Pim
DNA Methyltransferase
NOD-like Receptor (NLR)
Histone Demethylase
DNA
Casein Kinase
Tie-2
Smo
Ligand for E3 Ligase
Factor Xa
PAK
Fatty Acid Synthase
ROR
Glucokinase
Glucagon Receptor
NOS
Melatonin Receptor
Telomerase
AhR
GHSR
IRAK
CRM1
OAT
Bradykinin Receptor
BACE
CETP
MT Receptor
CaMK
Monoamine Transporter
Acyltransferase
Photosensitizer
Ephrin Receptor
CRFR
Gap Junction Protein
PD-1/PD-L1
PYK2
Glutaminase
UGT
GlyT
Wee1
PGE Synthase
GPCR19
Chloride channel
MTP
DprE1
Serine/threonin kinase
Cysteine Protease
DNA gyrase
Acetyl-CoA Carboxylase
CGRP Receptor
NADPH-oxidase
Tyrosinase
YAP
IFNAR
Neuropeptide Y Receptor
PROTACs
LTR
FAAH
Cholecystokinin Receptor
Myosin
IKZF
Decarboxylase
Neprilysin
c-Myc
Liver X Receptor
GST
Melanocortin Receptor
ASBT
Somatostatin
Thrombopoietin Receptor
BCRP
Cuproptosis
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Galectin
DUB
KSP
OXPHOS
STING
Free radical scavengers
FKBP
Cell wall
Annexin A
Na-K-Cl cotransporter
Stearoyl-CoA Desaturase (SCD)
LPA Receptor
PDK
NEDD8
PERK
ABC Transporter
ATP Citrate Lyase
Imidazoline Receptor
Adenosine Deaminase
Arginase
CaSR
Rho
NAMPT
Oxytocin Receptor
NOD
Neurotensin Receptor
Mucin
Survivin
p97
Apelin receptor
Ligands for Target Protein for PROTAC
Hexokinase
IRE1
LDL
Epoxide Hydrolase
Pyroptosis
MLK
Lipid
transporter
SGK
VDA
Porcupine
CD73
Taste receptor
Integrase
GSNOR
DYRK
HCN Channel
Histone Acetyltransferase
PAI-1
Vitamin
Adenylyl Cyclase
MIF
ASK
Methionine Adenosyltransferase (MAT)
Aquaporin
MicroRNA
Lipase
Immunology/Inflammation related
PAFR
MNK
KLF
PI4K
Monocarboxylate transporter
MALT
Arrestin
MAGL
Cadherin
Huntingtin
GluCls
RXFP receptor
PKM
Advanced Glycation End Products
Necroptosis
OCT
Hck
Stemness kinase
Fas/FasL
GRK
AAK1 (AP2 associated kinase 1)
Phosphorylase
ACK1
PSMA
BMI-1
Hydrogenase
Factor VIIa
N-Acetylglucosaminyltransferase
VDAC
NR4A
Anion Exchanger
PROTAC Linker
Hippo pathway
CRISPR/Cas9
NPC1L1
TOPK
Kisspeptin
AAK1
SIK
FLAP
Thioredoxin
FOXO
GTPase
MELK
Aromatase
Drug-Linker Conjugates for ADC
PGC-1α
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